EE03482B1 - Kinasoliiniderivaadid, nende valmistamismeetod ja kasutamine - Google Patents

Kinasoliiniderivaadid, nende valmistamismeetod ja kasutamine

Info

Publication number
EE03482B1
EE03482B1 EE9700252A EE9700252A EE03482B1 EE 03482 B1 EE03482 B1 EE 03482B1 EE 9700252 A EE9700252 A EE 9700252A EE 9700252 A EE9700252 A EE 9700252A EE 03482 B1 EE03482 B1 EE 03482B1
Authority
EE
Estonia
Prior art keywords
preparation
quinazoline derivatives
quinazoline
derivatives
Prior art date
Application number
EE9700252A
Other languages
English (en)
Estonian (et)
Other versions
EE9700252A (et
Inventor
Hopkinson Gibson Keith
Original Assignee
Zeneca Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=10773597&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EE03482(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Zeneca Limited filed Critical Zeneca Limited
Publication of EE9700252A publication Critical patent/EE9700252A/xx
Publication of EE03482B1 publication Critical patent/EE03482B1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/94—Nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
EE9700252A 1995-04-27 1996-04-23 Kinasoliiniderivaadid, nende valmistamismeetod ja kasutamine EE03482B1 (et)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9508538.7A GB9508538D0 (en) 1995-04-27 1995-04-27 Quinazoline derivatives
PCT/GB1996/000961 WO1996033980A1 (en) 1995-04-27 1996-04-23 Quinazoline derivatives

Publications (2)

Publication Number Publication Date
EE9700252A EE9700252A (et) 1998-04-15
EE03482B1 true EE03482B1 (et) 2001-08-15

Family

ID=10773597

Family Applications (1)

Application Number Title Priority Date Filing Date
EE9700252A EE03482B1 (et) 1995-04-27 1996-04-23 Kinasoliiniderivaadid, nende valmistamismeetod ja kasutamine

Country Status (39)

Country Link
US (1) US5770599A (no)
EP (1) EP0823900B1 (no)
JP (1) JP3040486B2 (no)
KR (1) KR100296656B1 (no)
CN (1) CN1100046C (no)
AR (1) AR003944A1 (no)
AT (1) ATE198329T1 (no)
AU (1) AU699163B2 (no)
BG (1) BG62730B1 (no)
BR (1) BRPI9608082B8 (no)
CA (1) CA2215732C (no)
CZ (1) CZ288489B6 (no)
DE (2) DE122009000076I1 (no)
DK (1) DK0823900T3 (no)
EE (1) EE03482B1 (no)
EG (1) EG24134A (no)
ES (1) ES2153098T3 (no)
FR (1) FR09C0065I2 (no)
GB (1) GB9508538D0 (no)
GR (1) GR3035211T3 (no)
HK (1) HK1005371A1 (no)
HR (1) HRP960204B1 (no)
HU (1) HU223313B1 (no)
IL (1) IL118045A (no)
LU (1) LU91631I2 (no)
MY (1) MY114425A (no)
NL (1) NL300429I1 (no)
NO (2) NO309472B1 (no)
NZ (1) NZ305444A (no)
PL (1) PL189182B1 (no)
PT (1) PT823900E (no)
RO (1) RO117849B1 (no)
RU (1) RU2153495C2 (no)
SI (1) SI0823900T1 (no)
SK (1) SK282236B6 (no)
TW (1) TW436486B (no)
UA (1) UA52602C2 (no)
WO (1) WO1996033980A1 (no)
ZA (1) ZA963358B (no)

Families Citing this family (711)

* Cited by examiner, † Cited by third party
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AU699163B2 (en) 1998-11-26
HUP9802839A3 (en) 2001-02-28
FR09C0065I1 (no) 2010-01-22
AU5343396A (en) 1996-11-18
NO2009028I2 (no) 2011-10-17
FR09C0065I2 (fr) 2014-03-28
DK0823900T3 (da) 2001-04-02
EP0823900B1 (en) 2000-12-27
PL189182B1 (pl) 2005-07-29
IL118045A (en) 2001-10-31
PT823900E (pt) 2001-04-30
DE69611361D1 (de) 2001-02-01
CN1182421A (zh) 1998-05-20
HU223313B1 (hu) 2004-05-28
CN1100046C (zh) 2003-01-29
EP0823900A1 (en) 1998-02-18
IL118045A0 (en) 1996-08-04
EG24134A (en) 2008-08-06
SK145497A3 (en) 1998-02-04
ZA963358B (en) 1996-10-28
DE122009000076I1 (de) 2010-05-06
PL323066A1 (en) 1998-03-02
DE69611361T2 (de) 2001-04-26
JP3040486B2 (ja) 2000-05-15
BRPI9608082B8 (pt) 2021-07-06
NO974940L (no) 1997-10-24
ATE198329T1 (de) 2001-01-15
CZ288489B6 (en) 2001-06-13
SI0823900T1 (no) 2001-06-30
GR3035211T3 (en) 2001-04-30
SK282236B6 (sk) 2001-12-03
HRP960204A2 (en) 1997-08-31
BG102052A (en) 1998-08-31
JPH11504033A (ja) 1999-04-06
US5770599A (en) 1998-06-23
CA2215732C (en) 2002-04-09
BRPI9608082B1 (pt) 2019-04-30
NO309472B1 (no) 2001-02-05
MY114425A (en) 2002-10-31
WO1996033980A1 (en) 1996-10-31
CZ339697A3 (cs) 1998-02-18
NL300429I1 (nl) 2010-03-01
HRP960204B1 (en) 2001-10-31
ES2153098T3 (es) 2001-02-16
AR003944A1 (es) 1998-09-30
NZ305444A (en) 1999-03-29
NO974940D0 (no) 1997-10-24
BRPI9608082A (pt) 1999-01-26
GB9508538D0 (en) 1995-06-14
KR100296656B1 (ko) 2001-08-07
EE9700252A (et) 1998-04-15
RO117849B1 (ro) 2002-08-30
BG62730B1 (bg) 2000-06-30
TW436486B (en) 2001-05-28
RU2153495C2 (ru) 2000-07-27
NO2009028I1 (no) 2014-05-19
HUP9802839A2 (hu) 1999-03-29
LU91631I2 (fr) 2010-02-17
UA52602C2 (uk) 2003-01-15
CA2215732A1 (en) 1996-10-31
HK1005371A1 (en) 1999-01-08

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