NO2009028I2 - Gefitinib eller et farmasøytisk akseptabelt salt derav - Google Patents

Gefitinib eller et farmasøytisk akseptabelt salt derav

Info

Publication number
NO2009028I2
NO2009028I2 NO2009028C NO2009028C NO2009028I2 NO 2009028 I2 NO2009028 I2 NO 2009028I2 NO 2009028 C NO2009028 C NO 2009028C NO 2009028 C NO2009028 C NO 2009028C NO 2009028 I2 NO2009028 I2 NO 2009028I2
Authority
NO
Norway
Prior art keywords
gefitinib
pharmaceutically acceptable
acceptable salt
salt
pharmaceutically
Prior art date
Application number
NO2009028C
Other languages
English (en)
Other versions
NO2009028I1 (no
Original Assignee
Astrazeneca Uk Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=10773597&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO2009028(I2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astrazeneca Uk Ltd filed Critical Astrazeneca Uk Ltd
Publication of NO2009028I2 publication Critical patent/NO2009028I2/no
Publication of NO2009028I1 publication Critical patent/NO2009028I1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/94—Nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
NO2009028C 1995-04-27 2009-12-16 Kinazolin-derivater, anvendelse og fremstilling derav, samt farmasøytisk preparat NO2009028I1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9508538.7A GB9508538D0 (en) 1995-04-27 1995-04-27 Quinazoline derivatives
PCT/GB1996/000961 WO1996033980A1 (en) 1995-04-27 1996-04-23 Quinazoline derivatives

Publications (2)

Publication Number Publication Date
NO2009028I2 true NO2009028I2 (no) 2011-10-17
NO2009028I1 NO2009028I1 (no) 2014-05-19

Family

ID=10773597

Family Applications (2)

Application Number Title Priority Date Filing Date
NO974940A NO309472B1 (no) 1995-04-27 1997-10-24 Kinazolin-derivater, anvendelse og fremstilling derav, samt farmasöytisk preparat
NO2009028C NO2009028I1 (no) 1995-04-27 2009-12-16 Kinazolin-derivater, anvendelse og fremstilling derav, samt farmasøytisk preparat

Family Applications Before (1)

Application Number Title Priority Date Filing Date
NO974940A NO309472B1 (no) 1995-04-27 1997-10-24 Kinazolin-derivater, anvendelse og fremstilling derav, samt farmasöytisk preparat

Country Status (39)

Country Link
US (1) US5770599A (no)
EP (1) EP0823900B1 (no)
JP (1) JP3040486B2 (no)
KR (1) KR100296656B1 (no)
CN (1) CN1100046C (no)
AR (1) AR003944A1 (no)
AT (1) ATE198329T1 (no)
AU (1) AU699163B2 (no)
BG (1) BG62730B1 (no)
BR (1) BRPI9608082B8 (no)
CA (1) CA2215732C (no)
CZ (1) CZ288489B6 (no)
DE (2) DE122009000076I1 (no)
DK (1) DK0823900T3 (no)
EE (1) EE03482B1 (no)
EG (1) EG24134A (no)
ES (1) ES2153098T3 (no)
FR (1) FR09C0065I2 (no)
GB (1) GB9508538D0 (no)
GR (1) GR3035211T3 (no)
HK (1) HK1005371A1 (no)
HR (1) HRP960204B1 (no)
HU (1) HU223313B1 (no)
IL (1) IL118045A (no)
LU (1) LU91631I2 (no)
MY (1) MY114425A (no)
NL (1) NL300429I1 (no)
NO (2) NO309472B1 (no)
NZ (1) NZ305444A (no)
PL (1) PL189182B1 (no)
PT (1) PT823900E (no)
RO (1) RO117849B1 (no)
RU (1) RU2153495C2 (no)
SI (1) SI0823900T1 (no)
SK (1) SK282236B6 (no)
TW (1) TW436486B (no)
UA (1) UA52602C2 (no)
WO (1) WO1996033980A1 (no)
ZA (1) ZA963358B (no)

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UA52602C2 (uk) 2003-01-15
IL118045A0 (en) 1996-08-04
WO1996033980A1 (en) 1996-10-31
MY114425A (en) 2002-10-31
EP0823900A1 (en) 1998-02-18
BG62730B1 (bg) 2000-06-30
US5770599A (en) 1998-06-23
CZ288489B6 (en) 2001-06-13
CA2215732A1 (en) 1996-10-31
CA2215732C (en) 2002-04-09
PL189182B1 (pl) 2005-07-29
BRPI9608082B8 (pt) 2021-07-06
IL118045A (en) 2001-10-31
CN1100046C (zh) 2003-01-29
HUP9802839A3 (en) 2001-02-28
BG102052A (en) 1998-08-31
EE03482B1 (et) 2001-08-15
SK145497A3 (en) 1998-02-04
GB9508538D0 (en) 1995-06-14
LU91631I2 (fr) 2010-02-17
KR19990007987A (ko) 1999-01-25
TW436486B (en) 2001-05-28
HRP960204A2 (en) 1997-08-31
BRPI9608082B1 (pt) 2019-04-30
RO117849B1 (ro) 2002-08-30
GR3035211T3 (en) 2001-04-30
JPH11504033A (ja) 1999-04-06
CZ339697A3 (cs) 1998-02-18
SK282236B6 (sk) 2001-12-03
ZA963358B (en) 1996-10-28
HU223313B1 (hu) 2004-05-28
PL323066A1 (en) 1998-03-02
EE9700252A (et) 1998-04-15
NO309472B1 (no) 2001-02-05
NL300429I1 (nl) 2010-03-01
SI0823900T1 (no) 2001-06-30
HK1005371A1 (en) 1999-01-08
RU2153495C2 (ru) 2000-07-27
HRP960204B1 (en) 2001-10-31
NO2009028I1 (no) 2014-05-19
AU699163B2 (en) 1998-11-26
DE122009000076I1 (de) 2010-05-06
EP0823900B1 (en) 2000-12-27
BRPI9608082A (pt) 1999-01-26
DE69611361D1 (de) 2001-02-01
JP3040486B2 (ja) 2000-05-15
FR09C0065I2 (fr) 2014-03-28
HUP9802839A2 (hu) 1999-03-29
EG24134A (en) 2008-08-06
FR09C0065I1 (no) 2010-01-22
KR100296656B1 (ko) 2001-08-07
NZ305444A (en) 1999-03-29
NO974940D0 (no) 1997-10-24
CN1182421A (zh) 1998-05-20
ATE198329T1 (de) 2001-01-15
DK0823900T3 (da) 2001-04-02
ES2153098T3 (es) 2001-02-16

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