SK282236B6 - Chinazolínové deriváty, spôsob ich prípravy, farmaceutický prostriedok, ktorý ich obsahuje a ich použitie - Google Patents

Chinazolínové deriváty, spôsob ich prípravy, farmaceutický prostriedok, ktorý ich obsahuje a ich použitie Download PDF

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Publication number
SK282236B6
SK282236B6 SK1454-97A SK145497A SK282236B6 SK 282236 B6 SK282236 B6 SK 282236B6 SK 145497 A SK145497 A SK 145497A SK 282236 B6 SK282236 B6 SK 282236B6
Authority
SK
Slovakia
Prior art keywords
formula
chloro
quinazoline
pharmaceutically acceptable
fluoroanilino
Prior art date
Application number
SK1454-97A
Other languages
English (en)
Slovak (sk)
Other versions
SK145497A3 (en
Inventor
Keith Hopkinson Gibson
Original Assignee
Zeneca Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=10773597&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SK282236(B6) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Zeneca Limited filed Critical Zeneca Limited
Publication of SK145497A3 publication Critical patent/SK145497A3/sk
Publication of SK282236B6 publication Critical patent/SK282236B6/sk

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/94—Nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
SK1454-97A 1995-04-27 1996-04-23 Chinazolínové deriváty, spôsob ich prípravy, farmaceutický prostriedok, ktorý ich obsahuje a ich použitie SK282236B6 (sk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9508538.7A GB9508538D0 (en) 1995-04-27 1995-04-27 Quinazoline derivatives
PCT/GB1996/000961 WO1996033980A1 (en) 1995-04-27 1996-04-23 Quinazoline derivatives

Publications (2)

Publication Number Publication Date
SK145497A3 SK145497A3 (en) 1998-02-04
SK282236B6 true SK282236B6 (sk) 2001-12-03

Family

ID=10773597

Family Applications (1)

Application Number Title Priority Date Filing Date
SK1454-97A SK282236B6 (sk) 1995-04-27 1996-04-23 Chinazolínové deriváty, spôsob ich prípravy, farmaceutický prostriedok, ktorý ich obsahuje a ich použitie

Country Status (39)

Country Link
US (1) US5770599A (hu)
EP (1) EP0823900B1 (hu)
JP (1) JP3040486B2 (hu)
KR (1) KR100296656B1 (hu)
CN (1) CN1100046C (hu)
AR (1) AR003944A1 (hu)
AT (1) ATE198329T1 (hu)
AU (1) AU699163B2 (hu)
BG (1) BG62730B1 (hu)
BR (1) BRPI9608082B8 (hu)
CA (1) CA2215732C (hu)
CZ (1) CZ288489B6 (hu)
DE (2) DE122009000076I1 (hu)
DK (1) DK0823900T3 (hu)
EE (1) EE03482B1 (hu)
EG (1) EG24134A (hu)
ES (1) ES2153098T3 (hu)
FR (1) FR09C0065I2 (hu)
GB (1) GB9508538D0 (hu)
GR (1) GR3035211T3 (hu)
HK (1) HK1005371A1 (hu)
HR (1) HRP960204B1 (hu)
HU (1) HU223313B1 (hu)
IL (1) IL118045A (hu)
LU (1) LU91631I2 (hu)
MY (1) MY114425A (hu)
NL (1) NL300429I1 (hu)
NO (2) NO309472B1 (hu)
NZ (1) NZ305444A (hu)
PL (1) PL189182B1 (hu)
PT (1) PT823900E (hu)
RO (1) RO117849B1 (hu)
RU (1) RU2153495C2 (hu)
SI (1) SI0823900T1 (hu)
SK (1) SK282236B6 (hu)
TW (1) TW436486B (hu)
UA (1) UA52602C2 (hu)
WO (1) WO1996033980A1 (hu)
ZA (1) ZA963358B (hu)

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DE122009000076I1 (de) 2010-05-06
PL189182B1 (pl) 2005-07-29
DE69611361T2 (de) 2001-04-26
RO117849B1 (ro) 2002-08-30
EP0823900A1 (en) 1998-02-18
NO2009028I2 (no) 2011-10-17
WO1996033980A1 (en) 1996-10-31
HUP9802839A3 (en) 2001-02-28
LU91631I2 (fr) 2010-02-17
CA2215732A1 (en) 1996-10-31
PT823900E (pt) 2001-04-30
BRPI9608082B8 (pt) 2021-07-06
JP3040486B2 (ja) 2000-05-15
PL323066A1 (en) 1998-03-02
IL118045A (en) 2001-10-31
CN1182421A (zh) 1998-05-20
NZ305444A (en) 1999-03-29
ES2153098T3 (es) 2001-02-16
FR09C0065I2 (fr) 2014-03-28
UA52602C2 (uk) 2003-01-15
IL118045A0 (en) 1996-08-04
NO974940L (no) 1997-10-24
ATE198329T1 (de) 2001-01-15
NO309472B1 (no) 2001-02-05
EP0823900B1 (en) 2000-12-27
HUP9802839A2 (hu) 1999-03-29

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