MA52780A - Inhibiteurs de kras g12c pour le traitement du cancer - Google Patents

Inhibiteurs de kras g12c pour le traitement du cancer

Info

Publication number
MA52780A
MA52780A MA052780A MA52780A MA52780A MA 52780 A MA52780 A MA 52780A MA 052780 A MA052780 A MA 052780A MA 52780 A MA52780 A MA 52780A MA 52780 A MA52780 A MA 52780A
Authority
MA
Morocco
Prior art keywords
kras
inhibitors
cancer treatment
cancer
treatment
Prior art date
Application number
MA052780A
Other languages
English (en)
Inventor
Victor J Cee
Jian Chen
Brian Alan Lanman
Longbin Liu
Youngsook Shin
Nuria A Tamayo
Hui-Ling Wang
Ryan Paul Wurz
Original Assignee
Amgen Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Amgen Inc filed Critical Amgen Inc
Publication of MA52780A publication Critical patent/MA52780A/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/16Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Peptides Or Proteins (AREA)
MA052780A 2018-06-11 2019-06-10 Inhibiteurs de kras g12c pour le traitement du cancer MA52780A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201862683263P 2018-06-11 2018-06-11

Publications (1)

Publication Number Publication Date
MA52780A true MA52780A (fr) 2021-04-14

Family

ID=67253966

Family Applications (1)

Application Number Title Priority Date Filing Date
MA052780A MA52780A (fr) 2018-06-11 2019-06-10 Inhibiteurs de kras g12c pour le traitement du cancer

Country Status (8)

Country Link
US (2) US20190375749A1 (fr)
EP (2) EP4268898A3 (fr)
JP (2) JP7357644B2 (fr)
AU (1) AU2019284472B2 (fr)
CA (1) CA3099799A1 (fr)
MA (1) MA52780A (fr)
MX (1) MX2020012204A (fr)
WO (1) WO2019241157A1 (fr)

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TW202340214A (zh) 2021-12-17 2023-10-16 美商健臻公司 做為shp2抑制劑之吡唑并吡𠯤化合物
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EP4268898A2 (fr) 2023-11-01
AU2019284472A1 (en) 2020-11-26
JP7357644B2 (ja) 2023-10-06
US20190375749A1 (en) 2019-12-12
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US20220002298A1 (en) 2022-01-06

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