BR9601200B1 - composto e seus sais farmaceuticamente aceitÁveis e composiÇço farmacÊutica para o tratamento de doenÇas hiperproliferativas compreendendo os mesmos. - Google Patents

composto e seus sais farmaceuticamente aceitÁveis e composiÇço farmacÊutica para o tratamento de doenÇas hiperproliferativas compreendendo os mesmos. Download PDF

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Publication number
BR9601200B1
BR9601200B1 BRPI9601200-5A BR9601200A BR9601200B1 BR 9601200 B1 BR9601200 B1 BR 9601200B1 BR 9601200 A BR9601200 A BR 9601200A BR 9601200 B1 BR9601200 B1 BR 9601200B1
Authority
BR
Brazil
Prior art keywords
mmol
amine
vacuo
quinazolin
ethoxy
Prior art date
Application number
BRPI9601200-5A
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English (en)
Portuguese (pt)
Other versions
BR9601200A (pt
Inventor
Rodney Caughren
Lee Daniel Arnold
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Publication date
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=23636708&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BR9601200(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed filed Critical
Publication of BR9601200A publication Critical patent/BR9601200A/pt
Publication of BR9601200B1 publication Critical patent/BR9601200B1/pt

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/94—Nitrogen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/08—Drugs for disorders of the urinary system of the prostate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Dermatology (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
BRPI9601200-5A 1995-03-30 1996-03-29 composto e seus sais farmaceuticamente aceitÁveis e composiÇço farmacÊutica para o tratamento de doenÇas hiperproliferativas compreendendo os mesmos. BR9601200B1 (pt)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US41330095A 1995-03-30 1995-03-30
US413300 1995-03-30
USPCT/IB95/00436 1995-06-06
PCT/IB1995/000436 WO1996030347A1 (en) 1995-03-30 1995-06-06 Quinazoline derivatives

Publications (2)

Publication Number Publication Date
BR9601200A BR9601200A (pt) 1998-01-06
BR9601200B1 true BR9601200B1 (pt) 2010-12-14

Family

ID=23636708

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI9601200-5A BR9601200B1 (pt) 1995-03-30 1996-03-29 composto e seus sais farmaceuticamente aceitÁveis e composiÇço farmacÊutica para o tratamento de doenÇas hiperproliferativas compreendendo os mesmos.

Country Status (43)

Country Link
EP (5) EP1110953B1 (enExample)
JP (1) JP3088018B2 (enExample)
KR (1) KR100232335B1 (enExample)
CN (1) CN1066142C (enExample)
AP (1) AP735A (enExample)
AR (1) AR002723A1 (enExample)
AT (2) ATE205483T1 (enExample)
AU (2) AU703638B2 (enExample)
BR (1) BR9601200B1 (enExample)
CA (1) CA2216796C (enExample)
CO (1) CO4410333A1 (enExample)
CZ (2) CZ294967B6 (enExample)
DE (3) DE69536015D1 (enExample)
DK (1) DK0817775T3 (enExample)
EG (1) EG24229A (enExample)
ES (2) ES2332984T3 (enExample)
FI (1) FI120646B (enExample)
FR (1) FR06C0010I2 (enExample)
GR (1) GR3037070T3 (enExample)
HR (1) HRP960147B1 (enExample)
HU (2) HU229120B1 (enExample)
IL (7) IL129995A (enExample)
LU (1) LU91209I2 (enExample)
MA (1) MA23831A1 (enExample)
MX (1) MX9707453A (enExample)
MY (1) MY117896A (enExample)
NL (1) NL300214I2 (enExample)
NO (2) NO308740B1 (enExample)
NZ (1) NZ286263A (enExample)
OA (1) OA10277A (enExample)
PE (1) PE43897A1 (enExample)
PL (1) PL186843B1 (enExample)
PT (1) PT817775E (enExample)
RU (2) RU2694252C2 (enExample)
SA (1) SA96160707B1 (enExample)
SG (1) SG43262A1 (enExample)
SI (1) SI9600102A (enExample)
SK (2) SK283762B6 (enExample)
TR (1) TR199600265A1 (enExample)
TW (1) TW454000B (enExample)
UA (1) UA44254C2 (enExample)
WO (1) WO1996030347A1 (enExample)
ZA (1) ZA962522B (enExample)

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RU2174977C2 (ru) 2001-10-20
PL186843B1 (pl) 2004-03-31
WO1996030347A1 (en) 1996-10-03
KR960034184A (ko) 1996-10-22
SG43262A1 (en) 1997-10-17
CZ294967B6 (cs) 2005-04-13
NO308740B1 (no) 2000-10-23
PT817775E (pt) 2002-01-30
TR199600265A1 (tr) 1997-03-21
LU91209I2 (fr) 2006-10-05
HRP960147B1 (en) 2002-04-30
EG24229A (enExample) 2008-11-10
KR100232335B1 (ko) 1999-12-01
IL117598A (en) 2005-11-20
CA2216796A1 (en) 1996-10-03
MA23831A1 (fr) 1996-10-01
EP0817775B1 (en) 2001-09-12
IL117598A0 (en) 1996-07-23
CA2216796C (en) 2003-09-02
DE69522717D1 (de) 2001-10-18

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