AP735A - Quinazoline derivatives. - Google Patents

Quinazoline derivatives. Download PDF

Info

Publication number
AP735A
AP735A APAP/P/1996/000788A AP9600788A AP735A AP 735 A AP735 A AP 735A AP 9600788 A AP9600788 A AP 9600788A AP 735 A AP735 A AP 735A
Authority
AP
ARIPO
Prior art keywords
amine
quinazolin
phenyl
ethynyl
ethoxy
Prior art date
Application number
APAP/P/1996/000788A
Other languages
English (en)
Other versions
AP9600788A0 (en
Inventor
Rodney Caughren Schnur
Lee Daniel Arnold
Original Assignee
Pfizer
Pfizer Prod Inc
Osi Pharm Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=23636708&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AP735(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer, Pfizer Prod Inc, Osi Pharm Inc filed Critical Pfizer
Publication of AP9600788A0 publication Critical patent/AP9600788A0/xx
Application granted granted Critical
Publication of AP735A publication Critical patent/AP735A/en

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/94—Nitrogen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/08—Drugs for disorders of the urinary system of the prostate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Dermatology (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
APAP/P/1996/000788A 1995-03-30 1996-03-07 Quinazoline derivatives. AP735A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US41330095A 1995-03-30 1995-03-30
PCT/IB1995/000436 WO1996030347A1 (en) 1995-03-30 1995-06-06 Quinazoline derivatives

Publications (2)

Publication Number Publication Date
AP9600788A0 AP9600788A0 (en) 1996-04-30
AP735A true AP735A (en) 1999-02-25

Family

ID=23636708

Family Applications (1)

Application Number Title Priority Date Filing Date
APAP/P/1996/000788A AP735A (en) 1995-03-30 1996-03-07 Quinazoline derivatives.

Country Status (43)

Country Link
EP (5) EP0817775B1 (cs)
JP (1) JP3088018B2 (cs)
KR (1) KR100232335B1 (cs)
CN (1) CN1066142C (cs)
AP (1) AP735A (cs)
AR (1) AR002723A1 (cs)
AT (2) ATE446955T1 (cs)
AU (2) AU703638B2 (cs)
BR (1) BR9601200B1 (cs)
CA (1) CA2216796C (cs)
CO (1) CO4410333A1 (cs)
CZ (2) CZ294967B6 (cs)
DE (3) DE122005000053I2 (cs)
DK (1) DK0817775T3 (cs)
EG (1) EG24229A (cs)
ES (2) ES2161290T3 (cs)
FI (1) FI120646B (cs)
FR (1) FR06C0010I2 (cs)
GR (1) GR3037070T3 (cs)
HR (1) HRP960147B1 (cs)
HU (2) HU229120B1 (cs)
IL (7) IL189037A (cs)
LU (1) LU91209I2 (cs)
MA (1) MA23831A1 (cs)
MX (1) MX9707453A (cs)
MY (1) MY117896A (cs)
NL (1) NL300214I2 (cs)
NO (2) NO308740B1 (cs)
NZ (1) NZ286263A (cs)
OA (1) OA10277A (cs)
PE (1) PE43897A1 (cs)
PL (1) PL186843B1 (cs)
PT (1) PT817775E (cs)
RU (2) RU2694252C3 (cs)
SA (1) SA96160707B1 (cs)
SG (1) SG43262A1 (cs)
SI (1) SI9600102A (cs)
SK (2) SK283762B6 (cs)
TR (1) TR199600265A1 (cs)
TW (1) TW454000B (cs)
UA (1) UA44254C2 (cs)
WO (1) WO1996030347A1 (cs)
ZA (1) ZA962522B (cs)

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* Cited by examiner, † Cited by third party
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HRP960147B1 (en) 2002-04-30
EP3103799A1 (en) 2016-12-14
DE69522717D1 (de) 2001-10-18
FI120646B (fi) 2010-01-15
PL313541A1 (en) 1996-10-14
EP2163546B1 (en) 2016-06-01
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CA2216796A1 (en) 1996-10-03
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FI973832A0 (fi) 1997-09-29
MA23831A1 (fr) 1996-10-01
IL129995A (en) 2005-11-20
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SK38796A3 (en) 1997-08-06
PE43897A1 (es) 1997-10-10
AU703638B2 (en) 1999-03-25
BR9601200B1 (pt) 2010-12-14
DE69522717T2 (de) 2002-02-14
IL189037A (en) 2011-03-31
SK283762B6 (sk) 2004-01-08
CN1137037A (zh) 1996-12-04

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