NO308740B1 - Kinazolinderivater, anvendelse derav og farmasøytisk blanding - Google Patents
Kinazolinderivater, anvendelse derav og farmasøytisk blandingInfo
- Publication number
- NO308740B1 NO308740B1 NO961299A NO961299A NO308740B1 NO 308740 B1 NO308740 B1 NO 308740B1 NO 961299 A NO961299 A NO 961299A NO 961299 A NO961299 A NO 961299A NO 308740 B1 NO308740 B1 NO 308740B1
- Authority
- NO
- Norway
- Prior art keywords
- quinazoline derivatives
- pharmaceutical admixture
- admixture
- pharmaceutical
- quinazoline
- Prior art date
Links
- 125000002294 quinazolinyl group Chemical class N1=C(N=CC2=CC=CC=C12)* 0.000 title 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
- C07D239/72—Quinazolines; Hydrogenated quinazolines
- C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
- C07D239/94—Nitrogen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/08—Drugs for disorders of the urinary system of the prostate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Urology & Nephrology (AREA)
- Dermatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US41330095A | 1995-03-30 | 1995-03-30 | |
| PCT/IB1995/000436 WO1996030347A1 (en) | 1995-03-30 | 1995-06-06 | Quinazoline derivatives |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NO961299D0 NO961299D0 (no) | 1996-03-29 |
| NO961299L NO961299L (no) | 1996-10-01 |
| NO308740B1 true NO308740B1 (no) | 2000-10-23 |
Family
ID=23636708
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO961299A NO308740B1 (no) | 1995-03-30 | 1996-03-29 | Kinazolinderivater, anvendelse derav og farmasøytisk blanding |
| NO2006004C NO2006004I2 (no) | 1995-03-30 | 2006-03-06 | Erlotinib hydroklorid og farmasøytisk akseptable salter derav |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO2006004C NO2006004I2 (no) | 1995-03-30 | 2006-03-06 | Erlotinib hydroklorid og farmasøytisk akseptable salter derav |
Country Status (43)
Families Citing this family (549)
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| SU400048A1 (cs) * | 1970-12-14 | 1973-10-03 | ||
| SU466233A1 (ru) * | 1973-06-08 | 1975-04-05 | Всесоюзный научно-исследовательский химико-фармацевтический институт им. С.Орджоникидзе | Способ получени производных 2-метил-4-диалкиламиноалкиламинохиназолина |
| US5710158A (en) * | 1991-05-10 | 1998-01-20 | Rhone-Poulenc Rorer Pharmaceuticals Inc. | Aryl and heteroaryl quinazoline compounds which inhibit EGF and/or PDGF receptor tyrosine kinase |
| DE69222637T2 (de) | 1991-05-10 | 1998-02-26 | Rhone Poulenc Rorer Int | Bis mono- und bicyclische aryl- und heteroarylderivate mit inhibierender wirkung auf die egf und/oder pdgf-rezeptor tyrosinkinase |
| NZ243082A (en) | 1991-06-28 | 1995-02-24 | Ici Plc | 4-anilino-quinazoline derivatives; pharmaceutical compositions, preparatory processes, and use thereof |
| GB9300059D0 (en) | 1992-01-20 | 1993-03-03 | Zeneca Ltd | Quinazoline derivatives |
| US5258518A (en) * | 1992-04-01 | 1993-11-02 | G. D. Searle & Co. | 2-substituted tertiary carbinol derivatives of deoxynojirimycin |
| GB9323290D0 (en) | 1992-12-10 | 1994-01-05 | Zeneca Ltd | Quinazoline derivatives |
| GB9314884D0 (en) | 1993-07-19 | 1993-09-01 | Zeneca Ltd | Tricyclic derivatives |
| GB9314893D0 (en) | 1993-07-19 | 1993-09-01 | Zeneca Ltd | Quinazoline derivatives |
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1995
- 1995-06-06 MX MX9707453A patent/MX9707453A/es active IP Right Grant
- 1995-06-06 DK DK95918713T patent/DK0817775T3/da active
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- 1995-06-06 EP EP01104696A patent/EP1110953B1/en not_active Expired - Lifetime
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1996
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- 1996-03-07 AP APAP/P/1996/000788A patent/AP735A/en active
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- 1996-03-29 AU AU50406/96A patent/AU703638B2/en not_active Expired
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- 1996-03-29 BR BRPI9601200-5A patent/BR9601200B1/pt not_active IP Right Cessation
- 1996-03-29 TR TR96/00265A patent/TR199600265A1/xx unknown
- 1996-03-29 MY MYPI96001194A patent/MY117896A/en unknown
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- 1996-03-29 RU RU0096106055A patent/RU2694252C3/ru active IP Right Grant
- 1996-03-29 CZ CZ1996931A patent/CZ294967B6/cs not_active IP Right Cessation
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- 1996-03-29 CZ CZ19972067A patent/CZ295145B6/cs not_active IP Right Cessation
- 1996-03-29 CO CO96015833A patent/CO4410333A1/es unknown
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- 1996-03-30 KR KR1019960009659A patent/KR100232335B1/ko not_active Expired - Lifetime
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1997
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1999
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2001
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2005
- 2005-12-14 LU LU91209C patent/LU91209I2/fr unknown
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2006
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2014
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