JP5934645B2 - グルタミニルシクラーゼ阻害剤としてのヘテロ環式誘導体 - Google Patents

グルタミニルシクラーゼ阻害剤としてのヘテロ環式誘導体 Download PDF

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JP5934645B2
JP5934645B2 JP2012528379A JP2012528379A JP5934645B2 JP 5934645 B2 JP5934645 B2 JP 5934645B2 JP 2012528379 A JP2012528379 A JP 2012528379A JP 2012528379 A JP2012528379 A JP 2012528379A JP 5934645 B2 JP5934645 B2 JP 5934645B2
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phenyl
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JP2013504544A5 (enExample
JP2013504544A (ja
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ヘイセル ウルリクフ
ヘイセル ウルリクフ
ソムメル ロベルト
ソムメル ロベルト
ラムスベクク ダニエル
ラムスベクク ダニエル
メイエル アントジェ
メイエル アントジェ
トルステン　ホフマン
ホフマン トルステン
ボエフメ ルイブイア
ボエフメ ルイブイア
デムトフ ハンス−ウルリクフ
デムトフ ハンス−ウルリクフ
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プロビオドルグ エージー
プロビオドルグ エージー
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    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
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JP2012528379A 2009-09-11 2010-09-13 グルタミニルシクラーゼ阻害剤としてのヘテロ環式誘導体 Active JP5934645B2 (ja)

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US24143209P 2009-09-11 2009-09-11
US61/241,432 2009-09-11
PCT/EP2010/063341 WO2011029920A1 (en) 2009-09-11 2010-09-13 Heterocylcic derivatives as inhibitors of glutaminyl cyclase

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JP2013504544A JP2013504544A (ja) 2013-02-07
JP2013504544A5 JP2013504544A5 (enExample) 2013-10-31
JP5934645B2 true JP5934645B2 (ja) 2016-06-15

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CA2772488A1 (en) 2011-03-17
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