IL104479A - History of quinazoline, the processes for their preparation and pharmacy preparations containing them and their use - Google Patents

History of quinazoline, the processes for their preparation and pharmacy preparations containing them and their use

Info

Publication number
IL104479A
IL104479A IL10447993A IL10447993A IL104479A IL 104479 A IL104479 A IL 104479A IL 10447993 A IL10447993 A IL 10447993A IL 10447993 A IL10447993 A IL 10447993A IL 104479 A IL104479 A IL 104479A
Authority
IL
Israel
Prior art keywords
quinazoline
mixture
formula
alkyl
alkoxy
Prior art date
Application number
IL10447993A
Other languages
English (en)
Hebrew (he)
Other versions
IL104479A0 (en
Original Assignee
Zeneca Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB929201095A external-priority patent/GB9201095D0/en
Priority claimed from GB929213572A external-priority patent/GB9213572D0/en
Priority claimed from GB929223735A external-priority patent/GB9223735D0/en
Application filed by Zeneca Ltd filed Critical Zeneca Ltd
Publication of IL104479A0 publication Critical patent/IL104479A0/xx
Publication of IL104479A publication Critical patent/IL104479A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/94—Nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04—Ortho-condensed systems

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
  • Cosmetics (AREA)
  • Treatments For Attaching Organic Compounds To Fibrous Goods (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
IL10447993A 1992-01-20 1993-01-21 History of quinazoline, the processes for their preparation and pharmacy preparations containing them and their use IL104479A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB929201095A GB9201095D0 (en) 1992-01-20 1992-01-20 Quinazoline derivatives
GB929213572A GB9213572D0 (en) 1992-06-26 1992-06-26 Quinazoline derivatives
GB929223735A GB9223735D0 (en) 1992-11-12 1992-11-12 Quinazoline derivatives

Publications (2)

Publication Number Publication Date
IL104479A0 IL104479A0 (en) 1993-05-13
IL104479A true IL104479A (en) 1999-12-22

Family

ID=27266013

Family Applications (1)

Application Number Title Priority Date Filing Date
IL10447993A IL104479A (en) 1992-01-20 1993-01-21 History of quinazoline, the processes for their preparation and pharmacy preparations containing them and their use

Country Status (22)

Country Link
US (2) US5457105A (de)
EP (1) EP0566226B1 (de)
KR (1) KR100229294B1 (de)
AT (1) ATE130000T1 (de)
AU (1) AU661533B2 (de)
CA (1) CA2086968C (de)
CZ (1) CZ282038B6 (de)
DE (1) DE69300754T2 (de)
DK (1) DK0566226T3 (de)
ES (1) ES2078798T3 (de)
FI (1) FI111631B (de)
GB (1) GB9300059D0 (de)
GR (1) GR3018143T3 (de)
HK (1) HK36497A (de)
HU (2) HU221622B1 (de)
IL (1) IL104479A (de)
NO (1) NO301541B1 (de)
NZ (1) NZ245662A (de)
RU (1) RU2127263C1 (de)
SK (1) SK281551B6 (de)
TW (1) TW283146B (de)
UA (1) UA34426C2 (de)

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* Cited by examiner, † Cited by third party
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