JO3598B1 - الاحماض والاسترات البورونية كمثبطات اميد هيدروليز الحامض الدهني - Google Patents

الاحماض والاسترات البورونية كمثبطات اميد هيدروليز الحامض الدهني

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Publication number
JO3598B1
JO3598B1 JOP/2007/0420A JOP20070420A JO3598B1 JO 3598 B1 JO3598 B1 JO 3598B1 JO P20070420 A JOP20070420 A JO P20070420A JO 3598 B1 JO3598 B1 JO 3598B1
Authority
JO
Jordan
Prior art keywords
inhibitors
esters
fatty acid
acid amide
boronic acids
Prior art date
Application number
JOP/2007/0420A
Other languages
English (en)
Inventor
A Snyder Daniel
A Evans Catherine
Grenier Louis
C Castro Alfredo
J Grogan Michael
Liu Tao
Adams Julian
T Tibbitts Thomas
L Behnke Mark
Original Assignee
Infinity Discovery Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39323893&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=JO3598(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Infinity Discovery Inc filed Critical Infinity Discovery Inc
Application granted granted Critical
Publication of JO3598B1 publication Critical patent/JO3598B1/ar

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    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C07F5/025—Boronic and borinic acid compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/69—Boron compounds
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C07F5/05—Cyclic compounds having at least one ring containing boron but no carbon in the ring

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  • Health & Medical Sciences (AREA)
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  • Life Sciences & Earth Sciences (AREA)
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  • Physical Education & Sports Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Diabetes (AREA)
  • Ophthalmology & Optometry (AREA)
  • Hematology (AREA)
  • Rheumatology (AREA)
  • Epidemiology (AREA)
  • Psychiatry (AREA)
  • Oncology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Immunology (AREA)
  • Obesity (AREA)
  • Virology (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Endocrinology (AREA)
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  • Communicable Diseases (AREA)
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Abstract

الاختراع الحالي يوفر مركبات، وتركيبات صيدلية مشتقة منها، تشمل عن طريق الصيغ (I)، (II) أو (III) الاختراع الحالي ايضا يوفر طرق لعلاج الظروف المصاحبة مع الفعالية المتزايدة من FAAH عن طريق تناول كمية فعالة علاجيا من المركب المتوفر من الصيغ (I)، (II) أو (III)، او تركيب صيدلي مشتق منه، تجاه شخص مريض بحاجة اليه. اضافيا، الاختراع الحالي يوفر طرق لتثبيط FAAH في شخص مريض عن طريق تناول كمية فعالة علاجيا من مركب الصيغة (I)، (II) أو (III)، او تركيب مشتق مقبول صيدليا، لشخص مريض بحاجة اليها.
JOP/2007/0420A 2006-10-10 2007-10-07 الاحماض والاسترات البورونية كمثبطات اميد هيدروليز الحامض الدهني JO3598B1 (ar)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US85052006P 2006-10-10 2006-10-10

Publications (1)

Publication Number Publication Date
JO3598B1 true JO3598B1 (ar) 2020-07-05

Family

ID=39323893

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Country Status (26)

Country Link
US (6) US7947663B2 (ar)
EP (4) EP2399585A1 (ar)
JP (2) JP5641600B2 (ar)
KR (2) KR20150038363A (ar)
CN (2) CN101563089A (ar)
AR (1) AR063165A1 (ar)
AT (1) ATE524188T1 (ar)
AU (1) AU2007322268B2 (ar)
BR (1) BRPI0719218A2 (ar)
CA (1) CA2666224C (ar)
CL (1) CL2007002910A1 (ar)
DK (1) DK2073816T3 (ar)
ES (1) ES2373697T3 (ar)
IL (2) IL197932A (ar)
JO (1) JO3598B1 (ar)
MX (1) MX2009003727A (ar)
NO (1) NO342439B1 (ar)
NZ (1) NZ576851A (ar)
PE (1) PE20081172A1 (ar)
PH (1) PH12012500765A1 (ar)
PT (1) PT2073816E (ar)
RU (1) RU2492174C2 (ar)
SG (3) SG10201502266RA (ar)
TW (1) TWI451870B (ar)
UA (1) UA101601C2 (ar)
WO (1) WO2008063300A2 (ar)

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