FR2758329B1 - Derives d'imidazole-4-butane boronique, leur preparation et leur utilisation en therapeutique - Google Patents
Derives d'imidazole-4-butane boronique, leur preparation et leur utilisation en therapeutiqueInfo
- Publication number
- FR2758329B1 FR2758329B1 FR9700379A FR9700379A FR2758329B1 FR 2758329 B1 FR2758329 B1 FR 2758329B1 FR 9700379 A FR9700379 A FR 9700379A FR 9700379 A FR9700379 A FR 9700379A FR 2758329 B1 FR2758329 B1 FR 2758329B1
- Authority
- FR
- France
- Prior art keywords
- boronic
- imidazole
- preparation
- therapeutic use
- butane derivatives
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
- 230000001225 therapeutic effect Effects 0.000 title 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K33/00—Medicinal preparations containing inorganic active ingredients
- A61K33/22—Boron compounds
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
- C07F5/02—Boron compounds
- C07F5/025—Boronic and borinic acid compounds
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Epidemiology (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Inorganic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9700379A FR2758329B1 (fr) | 1997-01-16 | 1997-01-16 | Derives d'imidazole-4-butane boronique, leur preparation et leur utilisation en therapeutique |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9700379A FR2758329B1 (fr) | 1997-01-16 | 1997-01-16 | Derives d'imidazole-4-butane boronique, leur preparation et leur utilisation en therapeutique |
Publications (2)
Publication Number | Publication Date |
---|---|
FR2758329A1 FR2758329A1 (fr) | 1998-07-17 |
FR2758329B1 true FR2758329B1 (fr) | 1999-02-12 |
Family
ID=9502641
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR9700379A Expired - Fee Related FR2758329B1 (fr) | 1997-01-16 | 1997-01-16 | Derives d'imidazole-4-butane boronique, leur preparation et leur utilisation en therapeutique |
Country Status (1)
Country | Link |
---|---|
FR (1) | FR2758329B1 (fr) |
Cited By (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US8329675B2 (en) | 2006-10-10 | 2012-12-11 | Infinity Pharmaceuticals, Inc. | Inhibitors of fatty acid amide hydrolase |
US8541581B2 (en) | 2009-04-07 | 2013-09-24 | Infinity Pharmaceuticals, Inc. | Inhibitors of fatty acid amide hydrolase |
US8546564B2 (en) | 2009-04-07 | 2013-10-01 | Infinity Pharmaceuticals, Inc. | Inhibitors of fatty acid amide hydrolase |
US9034849B2 (en) | 2010-02-03 | 2015-05-19 | Infinity Pharmaceuticals, Inc. | Fatty acid amide hydrolase inhibitors |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7122627B2 (en) | 1999-07-26 | 2006-10-17 | Bristol-Myers Squibb Company | Lactam inhibitors of Hepatitis C virus NS3 protease |
EP1206449A1 (fr) * | 1999-07-26 | 2002-05-22 | Bristol-Myers Squibb Company | Inhibiteurs lactame de la protease ns3 du virus de l'hepatite c |
WO2003105860A1 (fr) | 2002-06-14 | 2003-12-24 | Novo Nordisk A/S | Utilisation pharmaceutique d'acides boroniques et de leurs esters |
EP2282742A1 (fr) | 2008-04-09 | 2011-02-16 | Infinity Pharmaceuticals, Inc. | Inhibiteurs d'hydrolase d'amide d'acide gras |
WO2013053372A1 (fr) * | 2011-10-13 | 2013-04-18 | Therabor Pharmaceuticals | Inhibiteurs de type acide boronique de bêta-lactamases |
CA2963186A1 (fr) * | 2014-10-01 | 2016-04-07 | Merck Patent Gmbh | Derives d'acide boronique |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2701951B1 (fr) * | 1993-02-24 | 1995-06-09 | Adir | Nouveaux derives peptidiques de l'acide boronique, leur procede de preparation et les compositions pharmaceutiques qui les contiennent. |
FR2718451B1 (fr) * | 1994-04-12 | 1996-05-10 | Synthelabo | Dérivés de peptides boroniques, leur préparation et leur application en thérapeutique. |
US6083903A (en) * | 1994-10-28 | 2000-07-04 | Leukosite, Inc. | Boronic ester and acid compounds, synthesis and uses |
-
1997
- 1997-01-16 FR FR9700379A patent/FR2758329B1/fr not_active Expired - Fee Related
Cited By (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US8329675B2 (en) | 2006-10-10 | 2012-12-11 | Infinity Pharmaceuticals, Inc. | Inhibitors of fatty acid amide hydrolase |
US8349814B2 (en) | 2006-10-10 | 2013-01-08 | Infinity Pharmaceuticals, Inc. | Inhibitors of fatty acid amide hydrolase |
US8629125B2 (en) | 2006-10-10 | 2014-01-14 | Infinty Pharmaceuticals, Inc. | Inhibitors of fatty acid amide hydrolase |
US9108989B2 (en) | 2006-10-10 | 2015-08-18 | Infinity Pharmaceuticals, Inc. | Inhibitors of fatty acid amide hydrolase |
US8541581B2 (en) | 2009-04-07 | 2013-09-24 | Infinity Pharmaceuticals, Inc. | Inhibitors of fatty acid amide hydrolase |
US8546564B2 (en) | 2009-04-07 | 2013-10-01 | Infinity Pharmaceuticals, Inc. | Inhibitors of fatty acid amide hydrolase |
US8802119B2 (en) | 2009-04-07 | 2014-08-12 | Infinity Pharmaceuticals, Inc. | Inhibitors of fatty acid amide hydrolase |
US8802064B2 (en) | 2009-04-07 | 2014-08-12 | Infinity Pharmaceuticals, Inc. | Inhibitors of fatty acid amide hydrolase |
US9034849B2 (en) | 2010-02-03 | 2015-05-19 | Infinity Pharmaceuticals, Inc. | Fatty acid amide hydrolase inhibitors |
Also Published As
Publication number | Publication date |
---|---|
FR2758329A1 (fr) | 1998-07-17 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
TP | Transmission of property | ||
ST | Notification of lapse |