ES2516815T3 - Análogos de ácidos nucleicos bicíclicos modificados en la posición 6 - Google Patents

Análogos de ácidos nucleicos bicíclicos modificados en la posición 6 Download PDF

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Publication number
ES2516815T3
ES2516815T3 ES10176867.9T ES10176867T ES2516815T3 ES 2516815 T3 ES2516815 T3 ES 2516815T3 ES 10176867 T ES10176867 T ES 10176867T ES 2516815 T3 ES2516815 T3 ES 2516815T3
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oligomeric compound
mmol
nucleoside
substituted
reaction
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English (en)
Spanish (es)
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Eric E. Swayze
Punit P. Seth
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Ionis Pharmaceuticals Inc
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Isis Pharmaceuticals Inc
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H21/00Compounds containing two or more mononucleotide units having separate phosphate or polyphosphate groups linked by saccharide radicals of nucleoside groups, e.g. nucleic acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
ES10176867.9T 2006-01-27 2007-01-27 Análogos de ácidos nucleicos bicíclicos modificados en la posición 6 Active ES2516815T3 (es)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US76272206P 2006-01-27 2006-01-27
US762722P 2006-01-27
US80566006P 2006-06-23 2006-06-23
US805660P 2006-06-23

Publications (1)

Publication Number Publication Date
ES2516815T3 true ES2516815T3 (es) 2014-10-31

Family

ID=38328111

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ES10176867.9T Active ES2516815T3 (es) 2006-01-27 2007-01-27 Análogos de ácidos nucleicos bicíclicos modificados en la posición 6

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US (3) US7399845B2 (US07741457-20100622-C00066.png)
EP (3) EP1984381B1 (US07741457-20100622-C00066.png)
JP (2) JP5342881B2 (US07741457-20100622-C00066.png)
KR (2) KR101304071B1 (US07741457-20100622-C00066.png)
CN (2) CN102766630B (US07741457-20100622-C00066.png)
AT (1) ATE482965T1 (US07741457-20100622-C00066.png)
AU (1) AU2007211080B9 (US07741457-20100622-C00066.png)
CA (1) CA2640171C (US07741457-20100622-C00066.png)
DE (1) DE602007009487D1 (US07741457-20100622-C00066.png)
DK (2) DK2314594T3 (US07741457-20100622-C00066.png)
ES (1) ES2516815T3 (US07741457-20100622-C00066.png)
PL (2) PL1984381T3 (US07741457-20100622-C00066.png)
WO (1) WO2007090071A2 (US07741457-20100622-C00066.png)

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AU2007211080B2 (en) 2012-04-12
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US20070249049A1 (en) 2007-10-25
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US7741457B2 (en) 2010-06-22
ATE482965T1 (de) 2010-10-15
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