JP5342881B2 - 6−修飾された二環式核酸類似体 - Google Patents
6−修飾された二環式核酸類似体 Download PDFInfo
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- JP5342881B2 JP5342881B2 JP2008552604A JP2008552604A JP5342881B2 JP 5342881 B2 JP5342881 B2 JP 5342881B2 JP 2008552604 A JP2008552604 A JP 2008552604A JP 2008552604 A JP2008552604 A JP 2008552604A JP 5342881 B2 JP5342881 B2 JP 5342881B2
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- Prior art keywords
- oligomeric compound
- nucleoside
- mmol
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- nucleosides
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H21/00—Compounds containing two or more mononucleotide units having separate phosphate or polyphosphate groups linked by saccharide radicals of nucleoside groups, e.g. nucleic acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
- C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Applications Claiming Priority (5)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US76272206P | 2006-01-27 | 2006-01-27 | |
US60/762,722 | 2006-01-27 | ||
US80566006P | 2006-06-23 | 2006-06-23 | |
US60/805,660 | 2006-06-23 | ||
PCT/US2007/061183 WO2007090071A2 (en) | 2006-01-27 | 2007-01-27 | 6-modified bicyclic nucleic acid analogs |
Related Child Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP2013017584A Division JP2013147498A (ja) | 2006-01-27 | 2013-01-31 | 6−修飾された二環式核酸類似体 |
Publications (3)
Publication Number | Publication Date |
---|---|
JP2009524695A JP2009524695A (ja) | 2009-07-02 |
JP2009524695A5 JP2009524695A5 (US07741457-20100622-C00015.png) | 2009-12-17 |
JP5342881B2 true JP5342881B2 (ja) | 2013-11-13 |
Family
ID=38328111
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP2008552604A Active JP5342881B2 (ja) | 2006-01-27 | 2007-01-27 | 6−修飾された二環式核酸類似体 |
JP2013017584A Pending JP2013147498A (ja) | 2006-01-27 | 2013-01-31 | 6−修飾された二環式核酸類似体 |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP2013017584A Pending JP2013147498A (ja) | 2006-01-27 | 2013-01-31 | 6−修飾された二環式核酸類似体 |
Country Status (13)
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2013147498A (ja) * | 2006-01-27 | 2013-08-01 | Isis Pharmaceuticals Inc | 6−修飾された二環式核酸類似体 |
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