EA024255B1 - Синтез ингибиторов тирозинкиназы брутона - Google Patents

Синтез ингибиторов тирозинкиназы брутона Download PDF

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Publication number
EA024255B1
EA024255B1 EA201300246A EA201300246A EA024255B1 EA 024255 B1 EA024255 B1 EA 024255B1 EA 201300246 A EA201300246 A EA 201300246A EA 201300246 A EA201300246 A EA 201300246A EA 024255 B1 EA024255 B1 EA 024255B1
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EA
Eurasian Patent Office
Prior art keywords
acid
compound
pharmaceutically acceptable
acceptable salt
present
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Application number
EA201300246A
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English (en)
Russian (ru)
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EA201300246A1 (ru
Inventor
Ли Хонигберг
Эрик Вернер
Женгьинг Пан
Original Assignee
Фармасайкликс Элэлси
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39225888&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EA024255(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Фармасайкликс Элэлси filed Critical Фармасайкликс Элэлси
Publication of EA201300246A1 publication Critical patent/EA201300246A1/ru
Publication of EA024255B1 publication Critical patent/EA024255B1/ru

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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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  • Urology & Nephrology (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Pulmonology (AREA)
  • Neurosurgery (AREA)
  • Obesity (AREA)
  • Dermatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
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  • Reproductive Health (AREA)
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EA201300246A 2006-09-22 2006-12-28 Синтез ингибиторов тирозинкиназы брутона EA024255B1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US82672006P 2006-09-22 2006-09-22
US82859006P 2006-10-06 2006-10-06

Publications (2)

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EA201300246A1 EA201300246A1 (ru) 2014-01-30
EA024255B1 true EA024255B1 (ru) 2016-08-31

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EA201300246A EA024255B1 (ru) 2006-09-22 2006-12-28 Синтез ингибиторов тирозинкиназы брутона
EA201000599A EA020001B1 (ru) 2006-09-22 2006-12-28 Ингибиторы тирозинкиназы брутона
EA200900351A EA018573B1 (ru) 2006-09-22 2006-12-28 Ингибиторы тирозинкиназы брутона

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EA201000599A EA020001B1 (ru) 2006-09-22 2006-12-28 Ингибиторы тирозинкиназы брутона
EA200900351A EA018573B1 (ru) 2006-09-22 2006-12-28 Ингибиторы тирозинкиназы брутона

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US (49) US7514444B2 (OSRAM)
EP (11) EP2532235A1 (OSRAM)
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HUS1600049I1 (hu) 2017-01-30
LT2526771T (lt) 2017-06-12
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US8008309B2 (en) 2011-08-30
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AU2010201052B2 (en) 2012-03-15
ATE531263T1 (de) 2011-11-15
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LTPA2016034I1 (lt) 2016-12-27
LT2529622T (lt) 2018-05-10
US8748439B2 (en) 2014-06-10
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US8497277B2 (en) 2013-07-30
US8501751B2 (en) 2013-08-06
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