LU92692I2 - Ibrutinib, ou un sel pharmaceutiquement acceptablede celui-ci - Google Patents

Ibrutinib, ou un sel pharmaceutiquement acceptablede celui-ci Download PDF

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Publication number
LU92692I2
LU92692I2 LU92662C LU92662C LU92692I2 LU 92692 I2 LU92692 I2 LU 92692I2 LU 92662 C LU92662 C LU 92662C LU 92662 C LU92662 C LU 92662C LU 92692 I2 LU92692 I2 LU 92692I2
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Luxembourg
Prior art keywords
disclosed
compounds
conditions
btk
ibrutinib
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LU92662C
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Pharmacyclics Inc
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39225888&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=LU92692(I2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pharmacyclics Inc filed Critical Pharmacyclics Inc
Publication of LU92692I2 publication Critical patent/LU92692I2/fr

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    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
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    • C07KPEPTIDES
    • C07K16/00Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies
    • C07K16/18Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies against material from animals or humans
    • C07K16/28Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies against material from animals or humans against receptors, cell surface antigens or cell surface determinants
    • C07K16/2887Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies against material from animals or humans against receptors, cell surface antigens or cell surface determinants against CD20
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    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/20Immunoglobulins specific features characterized by taxonomic origin
    • C07K2317/24Immunoglobulins specific features characterized by taxonomic origin containing regions, domains or residues from different species, e.g. chimeric, humanized or veneered

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  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
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  • Endocrinology (AREA)
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  • Physical Education & Sports Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Neurology (AREA)
  • Pulmonology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Rheumatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Obesity (AREA)
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  • Genetics & Genomics (AREA)
  • Microbiology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
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LU92662C 2006-09-22 2015-04-07 Ibrutinib, ou un sel pharmaceutiquement acceptablede celui-ci LU92692I2 (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US82672006P 2006-09-22 2006-09-22
US82859006P 2006-10-06 2006-10-06
EP06850039.6A EP2081435B1 (fr) 2006-09-22 2006-12-28 Inhibiteurs de la tyrosine kinase de bruton

Publications (1)

Publication Number Publication Date
LU92692I2 true LU92692I2 (fr) 2015-11-24

Family

ID=39225888

Family Applications (3)

Application Number Title Priority Date Filing Date
LU92662C LU92692I2 (fr) 2006-09-22 2015-04-07 Ibrutinib, ou un sel pharmaceutiquement acceptablede celui-ci
LU93321C LU93321I2 (fr) 2006-09-22 2016-11-23 Ibrutinib, ou un sel pharmaceutiquement acceptable de celui-ci
LU00011C LUC00011I2 (fr) 2006-09-22 2017-03-30

Family Applications After (2)

Application Number Title Priority Date Filing Date
LU93321C LU93321I2 (fr) 2006-09-22 2016-11-23 Ibrutinib, ou un sel pharmaceutiquement acceptable de celui-ci
LU00011C LUC00011I2 (fr) 2006-09-22 2017-03-30

Country Status (28)

Country Link
US (48) US7514444B2 (fr)
EP (11) EP2201840B1 (fr)
JP (4) JP4934197B2 (fr)
KR (4) KR20100051863A (fr)
CN (4) CN102746305B (fr)
AT (1) ATE531263T1 (fr)
AU (2) AU2006348662B8 (fr)
BR (2) BRPI0622277A2 (fr)
CA (3) CA3180977A1 (fr)
CY (11) CY1112513T1 (fr)
DK (7) DK2526934T3 (fr)
EA (3) EA020001B1 (fr)
ES (8) ES2564647T3 (fr)
FR (1) FR15C0029I2 (fr)
HK (3) HK1129274A1 (fr)
HU (10) HUE033182T2 (fr)
IL (1) IL197550A0 (fr)
LT (7) LT2529622T (fr)
LU (3) LU92692I2 (fr)
MX (3) MX2009003122A (fr)
NL (1) NL300728I1 (fr)
NZ (3) NZ575650A (fr)
PL (8) PL2526934T4 (fr)
PT (7) PT2081435T (fr)
SG (2) SG166093A1 (fr)
SI (8) SI2526771T1 (fr)
WO (1) WO2008039218A2 (fr)
ZA (4) ZA200901784B (fr)

Families Citing this family (524)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK1740591T3 (da) * 2004-04-02 2009-10-26 Osi Pharm Inc Heterobicykliske proteinkinaseinhibitorer substitueret med en 6,6-biocyclisk ring
EP1906950A4 (fr) * 2005-06-21 2008-09-24 Infinity Discovery Inc Formulations d'ansamycine et leurs procedes d'utilisation
EP2865381A1 (fr) * 2006-05-18 2015-04-29 Pharmacyclics, Inc. Inhibiteurs de ITK pour le traitement des cancers des cellules sanguines
CA2660086C (fr) * 2006-08-16 2014-09-16 Novartis Ag Methode de fabrication de dispersions solides de composes therapeutiquesde cristallinite elevee
EP2201840B1 (fr) 2006-09-22 2011-11-02 Pharmacyclics, Inc. Inhibiteurs de la tyrosine kinase de Bruton
CA2668286C (fr) * 2006-11-03 2014-09-16 Pharmacyclics, Inc. Sonde d'activite de la tyrosine kinase de bruton et son procede d'utilisation
EP2954900A1 (fr) * 2007-03-28 2015-12-16 Pharmacyclics, Inc. Inhibiteurs de la tyrosine-kinase de bruton
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