ATE531263T1 - Hemmer der bruton-tyrosinkinase - Google Patents

Hemmer der bruton-tyrosinkinase

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Publication number
ATE531263T1
ATE531263T1 AT10155834T AT10155834T ATE531263T1 AT E531263 T1 ATE531263 T1 AT E531263T1 AT 10155834 T AT10155834 T AT 10155834T AT 10155834 T AT10155834 T AT 10155834T AT E531263 T1 ATE531263 T1 AT E531263T1
Authority
AT
Austria
Prior art keywords
disclosed
tyrosine kinase
compounds
conditions
btk
Prior art date
Application number
AT10155834T
Other languages
English (en)
Inventor
Lee Honigberg
Erik Verner
Zhengying Pan
Original Assignee
Pharmacyclics Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39225888&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ATE531263(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pharmacyclics Inc filed Critical Pharmacyclics Inc
Application granted granted Critical
Publication of ATE531263T1 publication Critical patent/ATE531263T1/de

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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    • A61K39/39533—Antibodies; Immunoglobulins; Immune serum, e.g. antilymphocytic serum against materials from animals
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K16/00—Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies
    • C07K16/18—Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies against material from animals or humans
    • C07K16/28—Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies against material from animals or humans against receptors, cell surface antigens or cell surface determinants
    • C07K16/2887—Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies against material from animals or humans against receptors, cell surface antigens or cell surface determinants against CD20
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    • C07K2317/24—Immunoglobulins specific features characterized by taxonomic origin containing regions, domains or residues from different species, e.g. chimeric, humanized or veneered

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  • Organic Chemistry (AREA)
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  • Animal Behavior & Ethology (AREA)
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  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Diabetes (AREA)
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  • Urology & Nephrology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Pulmonology (AREA)
  • Rheumatology (AREA)
  • Obesity (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Dermatology (AREA)
  • Oncology (AREA)
  • Reproductive Health (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biochemistry (AREA)
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  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
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AT10155834T 2006-09-22 2006-12-28 Hemmer der bruton-tyrosinkinase ATE531263T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US82672006P 2006-09-22 2006-09-22
US82859006P 2006-10-06 2006-10-06

Publications (1)

Publication Number Publication Date
ATE531263T1 true ATE531263T1 (de) 2011-11-15

Family

ID=39225888

Family Applications (1)

Application Number Title Priority Date Filing Date
AT10155834T ATE531263T1 (de) 2006-09-22 2006-12-28 Hemmer der bruton-tyrosinkinase

Country Status (27)

Country Link
US (49) US7514444B2 (de)
EP (11) EP2530083B1 (de)
JP (4) JP4934197B2 (de)
KR (4) KR20100051863A (de)
CN (4) CN102887900B (de)
AT (1) ATE531263T1 (de)
AU (2) AU2006348662B8 (de)
BR (2) BRPI0622054B8 (de)
CA (3) CA2663116C (de)
CY (11) CY1112513T1 (de)
DK (7) DK2529622T3 (de)
EA (3) EA024255B1 (de)
ES (8) ES2564647T3 (de)
FR (1) FR15C0029I2 (de)
HU (10) HUE028086T2 (de)
IL (1) IL197550A0 (de)
LT (7) LT2526771T (de)
LU (3) LU92692I2 (de)
MX (3) MX2009003122A (de)
NL (1) NL300728I1 (de)
NZ (3) NZ575650A (de)
PL (8) PL2526934T4 (de)
PT (7) PT2201840E (de)
SG (2) SG10201503235VA (de)
SI (8) SI2529621T1 (de)
WO (1) WO2008039218A2 (de)
ZA (4) ZA200901784B (de)

Families Citing this family (556)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR048518A1 (es) 2004-04-02 2006-05-03 Osi Pharm Inc Inhibidores heterobiciclicos de proteina quinasas sustituidos con anillos 6,6 -biciclicos
EP1906950A4 (de) * 2005-06-21 2008-09-24 Infinity Discovery Inc Ansamycin-formulierungen und anwendungsverfahren dafür
US8604031B2 (en) * 2006-05-18 2013-12-10 Mannkind Corporation Intracellular kinase inhibitors
WO2008021347A2 (en) * 2006-08-16 2008-02-21 Novartis Ag Method for making solid dispersions of highly crystalline therapeutic compounds
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