LU92692I2 - Ibrutinib, ou un sel pharmaceutiquement acceptablede celui-ci - Google Patents

Ibrutinib, ou un sel pharmaceutiquement acceptablede celui-ci Download PDF

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Publication number
LU92692I2
LU92692I2 LU92662C LU92662C LU92692I2 LU 92692 I2 LU92692 I2 LU 92692I2 LU 92662 C LU92662 C LU 92662C LU 92662 C LU92662 C LU 92662C LU 92692 I2 LU92692 I2 LU 92692I2
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LU
Luxembourg
Prior art keywords
disclosed
compounds
conditions
btk
ibrutinib
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Application number
LU92662C
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English (en)
French (fr)
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Pharmacyclics Inc
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Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39225888&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=LU92692(I2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pharmacyclics Inc filed Critical Pharmacyclics Inc
Publication of LU92692I2 publication Critical patent/LU92692I2/xx

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    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52Purines, e.g. adenine
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    • A61K31/33Heterocyclic compounds
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    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K16/00Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies
    • C07K16/18Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies against material from animals or humans
    • C07K16/28Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies against material from animals or humans against receptors, cell surface antigens or cell surface determinants
    • C07K16/2887Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies against material from animals or humans against receptors, cell surface antigens or cell surface determinants against CD20
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    • A61K2300/00Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/20Immunoglobulins specific features characterized by taxonomic origin
    • C07K2317/24Immunoglobulins specific features characterized by taxonomic origin containing regions, domains or residues from different species, e.g. chimeric, humanized or veneered
LU92662C 2006-09-22 2015-04-07 Ibrutinib, ou un sel pharmaceutiquement acceptablede celui-ci LU92692I2 (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US82672006P 2006-09-22 2006-09-22
US82859006P 2006-10-06 2006-10-06
EP06850039.6A EP2081435B1 (de) 2006-09-22 2006-12-28 Hämmer der bruton-tyrosinkinase

Publications (1)

Publication Number Publication Date
LU92692I2 true LU92692I2 (fr) 2015-11-24

Family

ID=39225888

Family Applications (3)

Application Number Title Priority Date Filing Date
LU92662C LU92692I2 (fr) 2006-09-22 2015-04-07 Ibrutinib, ou un sel pharmaceutiquement acceptablede celui-ci
LU93321C LU93321I2 (fr) 2006-09-22 2016-11-23 Ibrutinib, ou un sel pharmaceutiquement acceptable de celui-ci
LU00011C LUC00011I2 (de) 2006-09-22 2017-03-30

Family Applications After (2)

Application Number Title Priority Date Filing Date
LU93321C LU93321I2 (fr) 2006-09-22 2016-11-23 Ibrutinib, ou un sel pharmaceutiquement acceptable de celui-ci
LU00011C LUC00011I2 (de) 2006-09-22 2017-03-30

Country Status (28)

Country Link
US (48) US7514444B2 (de)
EP (11) EP2526933B1 (de)
JP (4) JP4934197B2 (de)
KR (4) KR101315610B1 (de)
CN (4) CN102746305B (de)
AT (1) ATE531263T1 (de)
AU (2) AU2006348662B8 (de)
BR (2) BRPI0622277A2 (de)
CA (3) CA2847852A1 (de)
CY (11) CY1112513T1 (de)
DK (7) DK2526934T3 (de)
EA (3) EA024255B1 (de)
ES (8) ES2564647T3 (de)
FR (1) FR15C0029I2 (de)
HK (3) HK1129274A1 (de)
HU (10) HUE033182T2 (de)
IL (1) IL197550A0 (de)
LT (7) LT2529622T (de)
LU (3) LU92692I2 (de)
MX (3) MX347525B (de)
NL (1) NL300728I2 (de)
NZ (3) NZ601278A (de)
PL (8) PL2526934T4 (de)
PT (7) PT2201840E (de)
SG (2) SG10201503235VA (de)
SI (8) SI2526934T1 (de)
WO (1) WO2008039218A2 (de)
ZA (4) ZA200901784B (de)

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AU2007254179B2 (en) * 2006-05-18 2013-03-21 Pharmacyclics Llc Intracellular kinase inhibitors
JP5546860B2 (ja) * 2006-08-16 2014-07-09 ノバルティス アーゲー 高結晶性治療化合物の固体分散体を製造するための方法
NZ601278A (en) * 2006-09-22 2013-09-27 Pharmacyclics Inc Inhibitors of Bruton's tyrosine kinase
ES2403546T3 (es) * 2006-11-03 2013-05-20 Pharmacyclics, Inc. Sonda de actividad de la tirosina-cinasa de Bruton y procedimiento de utilización
CA3143428A1 (en) * 2007-03-28 2008-10-09 Pharmacyclics Llc 8-amino-3-substituted-imidazo[1,5-a]pyrazine and use thereof as inhibitors of bruton's tyrosine kinase
US20120101114A1 (en) * 2007-03-28 2012-04-26 Pharmacyclics, Inc. Inhibitors of bruton's tyrosine kinase
CA2684211A1 (en) * 2007-04-12 2008-10-23 Infinity Discovery, Inc. Hydroquinone ansamycin formulations
US7989465B2 (en) * 2007-10-19 2011-08-02 Avila Therapeutics, Inc. 4,6-disubstituted pyrimidines useful as kinase inhibitors
US7982036B2 (en) 2007-10-19 2011-07-19 Avila Therapeutics, Inc. 4,6-disubstitued pyrimidines useful as kinase inhibitors
EP2250173A1 (de) * 2008-01-18 2010-11-17 OSI Pharmaceuticals, Inc. Imidazopyrazinolderivate zur behandlung von krebs
JP2011520970A (ja) * 2008-05-19 2011-07-21 オーエスアイ・フアーマスーテイカルズ・インコーポレーテツド 置換されたイミダゾピラジン類およびイミダゾトリアジン類
US20100101977A1 (en) * 2008-06-05 2010-04-29 United Comb & Novelty Corporation Stackable Packaging For Lipped Containers
US11351168B1 (en) 2008-06-27 2022-06-07 Celgene Car Llc 2,4-disubstituted pyrimidines useful as kinase inhibitors
US8338439B2 (en) 2008-06-27 2012-12-25 Celgene Avilomics Research, Inc. 2,4-disubstituted pyrimidines useful as kinase inhibitors
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CN106008514A (zh) 2014-01-29 2016-10-12 苏州晶云药物科技有限公司 依鲁替尼的新晶型及其制备方法

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