CY2016041I2 - Αναστολεις κινασης τυροσινης bruton - Google Patents

Αναστολεις κινασης τυροσινης bruton

Info

Publication number
CY2016041I2
CY2016041I2 CY2016041C CY2016041C CY2016041I2 CY 2016041 I2 CY2016041 I2 CY 2016041I2 CY 2016041 C CY2016041 C CY 2016041C CY 2016041 C CY2016041 C CY 2016041C CY 2016041 I2 CY2016041 I2 CY 2016041I2
Authority
CY
Cyprus
Prior art keywords
tyrosine kinase
kinase inhibitors
bruton tyrosine
bruton
inhibitors
Prior art date
Application number
CY2016041C
Other languages
English (en)
Other versions
CY2016041I1 (el
Original Assignee
Pharmacyclics Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39225888&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CY2016041(I2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pharmacyclics Llc filed Critical Pharmacyclics Llc
Publication of CY2016041I1 publication Critical patent/CY2016041I1/el
Publication of CY2016041I2 publication Critical patent/CY2016041I2/el

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52Purines, e.g. adenine
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    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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    • A61K39/39533Antibodies; Immunoglobulins; Immune serum, e.g. antilymphocytic serum against materials from animals
    • A61K39/3955Antibodies; Immunoglobulins; Immune serum, e.g. antilymphocytic serum against materials from animals against proteinaceous materials, e.g. enzymes, hormones, lymphokines
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    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K16/00Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies
    • C07K16/18Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies against material from animals or humans
    • C07K16/28Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies against material from animals or humans against receptors, cell surface antigens or cell surface determinants
    • C07K16/2887Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies against material from animals or humans against receptors, cell surface antigens or cell surface determinants against CD20
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    • CCHEMISTRY; METALLURGY
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    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/20Immunoglobulins specific features characterized by taxonomic origin
    • C07K2317/24Immunoglobulins specific features characterized by taxonomic origin containing regions, domains or residues from different species, e.g. chimeric, humanized or veneered

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  • Health & Medical Sciences (AREA)
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  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Immunology (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Hematology (AREA)
  • Urology & Nephrology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pulmonology (AREA)
  • Biomedical Technology (AREA)
  • Rheumatology (AREA)
  • Obesity (AREA)
  • Dermatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Oncology (AREA)
  • Reproductive Health (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biochemistry (AREA)
  • Mycology (AREA)
  • Microbiology (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Ophthalmology & Optometry (AREA)
CY2016041C 2006-09-22 2016-11-15 Αναστολεις κινασης τυροσινης bruton CY2016041I2 (el)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US82672006P 2006-09-22 2006-09-22
US82859006P 2006-10-06 2006-10-06
EP06850039.6A EP2081435B1 (en) 2006-09-22 2006-12-28 Inhibitors of bruton's tyrosine kinase

Publications (2)

Publication Number Publication Date
CY2016041I1 CY2016041I1 (el) 2017-03-15
CY2016041I2 true CY2016041I2 (el) 2017-03-15

Family

ID=39225888

Family Applications (11)

Application Number Title Priority Date Filing Date
CY20121100100T CY1112513T1 (el) 2006-09-22 2012-01-27 Αναστολεις της κινασης τυροσινης του bruton
CY2015016C CY2015016I2 (el) 2006-09-22 2015-04-03 Αναστολεις της κινασης τυροσινης του bruton
CY20151100453T CY1116295T1 (el) 2006-09-22 2015-05-20 Αναστολεις της κινασης τυροσινης toy bruton
CY20161100196T CY1117587T1 (el) 2006-09-22 2016-03-07 Αναστολεις κινασης τυροσινης bruton
CY20161100734T CY1117840T1 (el) 2006-09-22 2016-07-26 Αναστολεις κινασης τυροσινης bruton
CY20161100765T CY1117897T1 (el) 2006-09-22 2016-08-03 Αναστολεις κινασης τυροσινης bruton
CY2016041C CY2016041I2 (el) 2006-09-22 2016-11-15 Αναστολεις κινασης τυροσινης bruton
CY20161101348T CY1119209T1 (el) 2006-09-22 2016-12-27 Αναστολεις κινασης τυροσινης bruton
CY20171100248T CY1118666T1 (el) 2006-09-22 2017-02-22 Αναστολεις κινασης τυροσινης bruton
CY2017012C CY2017012I2 (el) 2006-09-22 2017-03-31 Αναστολεις κινασης τυροσινης bruton
CY20181100404T CY1120135T1 (el) 2006-09-22 2018-04-17 Αναστολεις κινασης τυροσινης bruton

Family Applications Before (6)

Application Number Title Priority Date Filing Date
CY20121100100T CY1112513T1 (el) 2006-09-22 2012-01-27 Αναστολεις της κινασης τυροσινης του bruton
CY2015016C CY2015016I2 (el) 2006-09-22 2015-04-03 Αναστολεις της κινασης τυροσινης του bruton
CY20151100453T CY1116295T1 (el) 2006-09-22 2015-05-20 Αναστολεις της κινασης τυροσινης toy bruton
CY20161100196T CY1117587T1 (el) 2006-09-22 2016-03-07 Αναστολεις κινασης τυροσινης bruton
CY20161100734T CY1117840T1 (el) 2006-09-22 2016-07-26 Αναστολεις κινασης τυροσινης bruton
CY20161100765T CY1117897T1 (el) 2006-09-22 2016-08-03 Αναστολεις κινασης τυροσινης bruton

Family Applications After (4)

Application Number Title Priority Date Filing Date
CY20161101348T CY1119209T1 (el) 2006-09-22 2016-12-27 Αναστολεις κινασης τυροσινης bruton
CY20171100248T CY1118666T1 (el) 2006-09-22 2017-02-22 Αναστολεις κινασης τυροσινης bruton
CY2017012C CY2017012I2 (el) 2006-09-22 2017-03-31 Αναστολεις κινασης τυροσινης bruton
CY20181100404T CY1120135T1 (el) 2006-09-22 2018-04-17 Αναστολεις κινασης τυροσινης bruton

Country Status (27)

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