JP4934197B2 - ブルートンチロシンキナーゼ阻害剤 - Google Patents

ブルートンチロシンキナーゼ阻害剤 Download PDF

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JP4934197B2
JP4934197B2 JP2009529166A JP2009529166A JP4934197B2 JP 4934197 B2 JP4934197 B2 JP 4934197B2 JP 2009529166 A JP2009529166 A JP 2009529166A JP 2009529166 A JP2009529166 A JP 2009529166A JP 4934197 B2 JP4934197 B2 JP 4934197B2
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compound
formula
substituted
tyrosine kinase
alkyl
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JP2010504324A5 (OSRAM
JP2010504324A (ja
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リー・ホニグバーグ
エリック・バーナー
パン・ジェンイン
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Pharmacyclics LLC
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Pharmacyclics LLC
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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  • Immunology (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Hematology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Pulmonology (AREA)
  • Neurosurgery (AREA)
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  • Ophthalmology & Optometry (AREA)
JP2009529166A 2006-09-22 2006-12-28 ブルートンチロシンキナーゼ阻害剤 Active JP4934197B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US82672006P 2006-09-22 2006-09-22
US60/826,720 2006-09-22
US82859006P 2006-10-06 2006-10-06
US60/828,590 2006-10-06
PCT/US2006/049626 WO2008039218A2 (en) 2006-09-22 2006-12-28 Inhibitors of bruton's tyrosine kinase

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JP2010155965A Division JP5193256B2 (ja) 2006-09-22 2010-07-08 ブルートンチロシンキナーゼ阻害剤

Publications (3)

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JP2010504324A JP2010504324A (ja) 2010-02-12
JP2010504324A5 JP2010504324A5 (OSRAM) 2010-08-26
JP4934197B2 true JP4934197B2 (ja) 2012-05-16

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JP2009529166A Active JP4934197B2 (ja) 2006-09-22 2006-12-28 ブルートンチロシンキナーゼ阻害剤
JP2010155965A Active JP5193256B2 (ja) 2006-09-22 2010-07-08 ブルートンチロシンキナーゼ阻害剤
JP2012049524A Active JP5635544B2 (ja) 2006-09-22 2012-03-06 ブルートンチロシンキナーゼ阻害剤
JP2012286719A Active JP5718890B2 (ja) 2006-09-22 2012-12-28 ブルートンチロシンキナーゼ阻害剤

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JP2012049524A Active JP5635544B2 (ja) 2006-09-22 2012-03-06 ブルートンチロシンキナーゼ阻害剤
JP2012286719A Active JP5718890B2 (ja) 2006-09-22 2012-12-28 ブルートンチロシンキナーゼ阻害剤

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HK1140107A1 (en) 2010-10-08
JP2010504324A (ja) 2010-02-12
CA2663116C (en) 2014-06-10
PL2530083T3 (pl) 2016-11-30
US9266893B2 (en) 2016-02-23
US8236812B2 (en) 2012-08-07
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US20120214826A1 (en) 2012-08-23
CY1112513T1 (el) 2015-12-09
US8088781B2 (en) 2012-01-03
US8563563B2 (en) 2013-10-22
PL2526933T3 (pl) 2015-08-31
KR20090091115A (ko) 2009-08-26
US20110184001A1 (en) 2011-07-28
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US20140135347A1 (en) 2014-05-15
EP2532234A1 (en) 2012-12-12
US20110008257A1 (en) 2011-01-13
US20120122894A1 (en) 2012-05-17
EP2529621B1 (en) 2016-10-05
CY1117897T1 (el) 2017-05-17
US8735404B2 (en) 2014-05-27
BE2015C016I2 (OSRAM) 2025-12-10
HUE033182T2 (en) 2017-11-28
LU92692I2 (fr) 2015-11-24
PL2529622T3 (pl) 2018-07-31
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US9212185B2 (en) 2015-12-15
US8957079B2 (en) 2015-02-17
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HUE028086T2 (en) 2016-11-28
US20120095026A1 (en) 2012-04-19
US8952015B2 (en) 2015-02-10
DK2201840T3 (da) 2012-02-20
HUS1600049I1 (hu) 2017-01-30
LT2526771T (lt) 2017-06-12
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US8008309B2 (en) 2011-08-30
US9133201B2 (en) 2015-09-15
US8754091B2 (en) 2014-06-17
AU2010201052B2 (en) 2012-03-15
ATE531263T1 (de) 2011-11-15
CY2016041I1 (el) 2017-03-15
LTPA2016034I1 (lt) 2016-12-27
LT2529622T (lt) 2018-05-10
US8748439B2 (en) 2014-06-10
EA200900351A1 (ru) 2009-10-30
US8497277B2 (en) 2013-07-30
US8501751B2 (en) 2013-08-06
US20120108612A1 (en) 2012-05-03
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