AR088570A1 - Metodos para tratar una enfermedad o trastorno relacionado con la tirosina quinasa de bruton - Google Patents

Metodos para tratar una enfermedad o trastorno relacionado con la tirosina quinasa de bruton

Info

Publication number
AR088570A1
AR088570A1 ARP120104042A ARP120104042A AR088570A1 AR 088570 A1 AR088570 A1 AR 088570A1 AR P120104042 A ARP120104042 A AR P120104042A AR P120104042 A ARP120104042 A AR P120104042A AR 088570 A1 AR088570 A1 AR 088570A1
Authority
AR
Argentina
Prior art keywords
illness
treat
methods
tyrosine kinase
disorder related
Prior art date
Application number
ARP120104042A
Other languages
English (en)
Original Assignee
Celgene Avilomics Res Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Celgene Avilomics Res Inc filed Critical Celgene Avilomics Res Inc
Publication of AR088570A1 publication Critical patent/AR088570A1/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841—Filling excipients; Inactive ingredients
    • A61K9/4866—Organic macromolecular compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)

Abstract

Reivindicación 1: Un método para tratar, estabilizar o disminuir la gravedad o progresión de una enfermedad o trastorno perteneciente al grupo integrado por linfoma no Hodgkin de células B, leucemia linfocitica crónica y macroglobulinemia de Waldenstrom, el método comprende la administración a un paciente que lo necesita, de una composición farmacéuticamente aceptable que comprende N-(3-(5-fluoro-2-(4-(2-metoxietoxi)fenilamino)pirimidin-4-ilamino)fenil)acrilamida de fórmula (1).
ARP120104042A 2011-10-28 2012-10-26 Metodos para tratar una enfermedad o trastorno relacionado con la tirosina quinasa de bruton AR088570A1 (es)

Applications Claiming Priority (8)

Application Number Priority Date Filing Date Title
US201161552936P 2011-10-28 2011-10-28
US201161569475P 2011-12-12 2011-12-12
US201261592351P 2012-01-30 2012-01-30
US201261593056P 2012-01-31 2012-01-31
US201261604780P 2012-02-29 2012-02-29
US201261618347P 2012-03-30 2012-03-30
US201261649450P 2012-05-21 2012-05-21
US201261660319P 2012-06-15 2012-06-15

Publications (1)

Publication Number Publication Date
AR088570A1 true AR088570A1 (es) 2014-06-18

Family

ID=48168552

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP120104042A AR088570A1 (es) 2011-10-28 2012-10-26 Metodos para tratar una enfermedad o trastorno relacionado con la tirosina quinasa de bruton

Country Status (7)

Country Link
US (2) US9364476B2 (es)
EP (1) EP2770830A4 (es)
JP (1) JP2014532658A (es)
AR (1) AR088570A1 (es)
CA (1) CA2853498A1 (es)
TW (1) TW201325593A (es)
WO (1) WO2013063401A1 (es)

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US20140142129A1 (en) * 2012-11-20 2014-05-22 Celgene Avilomics Research, Inc, Methods of treating a disease or disorder associated with bruton's tyrosine kinase
WO2014081712A2 (en) * 2012-11-20 2014-05-30 Celgene Avilomics Research, Inc. Methods of treating a disease or disorder associated with bruton's tyrosine kinase
US20140140991A1 (en) * 2012-11-20 2014-05-22 Celgene Avilomics Research, Inc. Methods of treating a disease or disorder associated with bruton's tyrosine kinase
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US20160287588A1 (en) 2016-10-06
EP2770830A4 (en) 2015-05-27
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