BRPI0611863B1 - Composto, bem como composição e kit compreendendo o mesmo, composto intermediário na preparação do mesmo, método para tratamento e uso do mesmo - Google Patents

Composto, bem como composição e kit compreendendo o mesmo, composto intermediário na preparação do mesmo, método para tratamento e uso do mesmo Download PDF

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Publication number
BRPI0611863B1
BRPI0611863B1 BRPI0611863-1A BRPI0611863A BRPI0611863B1 BR PI0611863 B1 BRPI0611863 B1 BR PI0611863B1 BR PI0611863 A BRPI0611863 A BR PI0611863A BR PI0611863 B1 BRPI0611863 B1 BR PI0611863B1
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BR
Brazil
Prior art keywords
optionally substituted
fluorine
nhc
nrr
group
Prior art date
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BRPI0611863-1A
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English (en)
Portuguese (pt)
Inventor
Prabha N. Ibrahim
Dean R. Artis
Ryan Bremer
Shumeye Mamo
Marika Nespi
Chao Zhang
Jiazhong Zhang
Yong-Liang Zhu
James Tsai
Klaus-Peter Hirth
Gideon Bollag
Wayne Spevak
Hanna Cho
Samuel J. Gillette
Guoxiam Wu
Hongyao Zhu
Shenghua Shi
Original Assignee
Plexxikon, Inc
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Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=37033831&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BRPI0611863(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Plexxikon, Inc filed Critical Plexxikon, Inc
Publication of BRPI0611863A2 publication Critical patent/BRPI0611863A2/pt
Publication of BRPI0611863B1 publication Critical patent/BRPI0611863B1/pt

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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
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