SG11201500883YA - 5-(1H-PYRAZOL-4-YL)-1H-PYRROLO[2,3-b]PYRIDINE DERIVATIVES AS KINASE INHIBITORS - Google Patents

5-(1H-PYRAZOL-4-YL)-1H-PYRROLO[2,3-b]PYRIDINE DERIVATIVES AS KINASE INHIBITORS

Info

Publication number
SG11201500883YA
SG11201500883YA SG11201500883YA SG11201500883YA SG11201500883YA SG 11201500883Y A SG11201500883Y A SG 11201500883YA SG 11201500883Y A SG11201500883Y A SG 11201500883YA SG 11201500883Y A SG11201500883Y A SG 11201500883YA SG 11201500883Y A SG11201500883Y A SG 11201500883YA
Authority
SG
Singapore
Prior art keywords
pyrrolo
pyrazol
kinase inhibitors
pyridine derivatives
pyridine
Prior art date
Application number
SG11201500883YA
Inventor
Venkateshwar Rao Gummadi
Subramanya Hosahalli
Srinivas Nanduri
Renukappa Girish Aggunda
Original Assignee
Aurigene Discovery Tech Ltd
Um Pharmauji Sdn Bhd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aurigene Discovery Tech Ltd, Um Pharmauji Sdn Bhd filed Critical Aurigene Discovery Tech Ltd
Publication of SG11201500883YA publication Critical patent/SG11201500883YA/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
SG11201500883YA 2012-08-07 2013-07-25 5-(1H-PYRAZOL-4-YL)-1H-PYRROLO[2,3-b]PYRIDINE DERIVATIVES AS KINASE INHIBITORS SG11201500883YA (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IN3217CH2012 2012-08-07
PCT/IB2013/056105 WO2014024077A1 (en) 2012-08-07 2013-07-25 5-(1H-PYRAZOL-4-YL)-1H-PYRROLO[2,3-b]PYRIDINE DERIVATIVES AS KINASE INHIBITORS

Publications (1)

Publication Number Publication Date
SG11201500883YA true SG11201500883YA (en) 2015-04-29

Family

ID=50067477

Family Applications (1)

Application Number Title Priority Date Filing Date
SG11201500883YA SG11201500883YA (en) 2012-08-07 2013-07-25 5-(1H-PYRAZOL-4-YL)-1H-PYRROLO[2,3-b]PYRIDINE DERIVATIVES AS KINASE INHIBITORS

Country Status (4)

Country Link
US (1) US20150183781A1 (en)
EP (1) EP2882748A1 (en)
SG (1) SG11201500883YA (en)
WO (1) WO2014024077A1 (en)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP6839715B2 (en) * 2015-09-29 2021-03-10 ノバルティス アーゲー Method for preparing 1- (4-methanesulfonyl-2-trifluoromethyl-benzyl) -2-methyl-1H-pyrrolo [2,3-b] pyridine-3-yl-acetic acid
EP3883573A4 (en) * 2018-11-19 2022-08-17 Dana-Farber Cancer Institute, Inc. Macrocyclic inhibitors of dyrk1a

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2005539000A (en) * 2002-07-31 2005-12-22 スミスクライン・ビーチャム・コーポレイション 2-Phenylpyridin-4-yl derivatives as ALK5 inhibitors
US20090149504A1 (en) * 2005-06-17 2009-06-11 Aurigene Discovery Technologies Limited Novel 5-Substituted Indole Derivatives As Dipeptidyl Peptidase IV (DPP-IV) Inhibitors
TWI522337B (en) * 2005-06-22 2016-02-21 普雷辛肯公司 Compounds and methods for kinase modulation, and indications therefor
EP2265270A1 (en) * 2008-02-04 2010-12-29 OSI Pharmaceuticals, Inc. 2-aminopyridine kinase inhibitors
WO2014004863A2 (en) * 2012-06-27 2014-01-03 Alzheimer's Institute Of America, Inc. Compounds, compositions, and therapeutic uses thereof

Also Published As

Publication number Publication date
EP2882748A4 (en) 2015-06-17
EP2882748A1 (en) 2015-06-17
WO2014024077A9 (en) 2014-04-03
WO2014024077A1 (en) 2014-02-13
US20150183781A1 (en) 2015-07-02

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