NO20053644L - (2S)-2-[(4S)-4-(2,2-difluorvinyl)-2-oksopyrrolidinyl ]butanamid og farmasoytisk preparat - Google Patents
(2S)-2-[(4S)-4-(2,2-difluorvinyl)-2-oksopyrrolidinyl ]butanamid og farmasoytisk preparatInfo
- Publication number
- NO20053644L NO20053644L NO20053644A NO20053644A NO20053644L NO 20053644 L NO20053644 L NO 20053644L NO 20053644 A NO20053644 A NO 20053644A NO 20053644 A NO20053644 A NO 20053644A NO 20053644 L NO20053644 L NO 20053644L
- Authority
- NO
- Norway
- Prior art keywords
- difluorovinyl
- oxopyrrolidinyl
- butanamide
- pharmaceutical preparation
- epilepsy
- Prior art date
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- C07D207/18—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
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- A61K31/4015—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil having oxo groups directly attached to the heterocyclic ring, e.g. piracetam, ethosuximide
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Abstract
Oppfinnelsen angår 2-okso-l-pyrrolidinderivater av formel I hvori substituentene er som definert i beskrivelsen, så vel som deres anvendelse som farmas0ytiske midler. Forbindelsene ifølge oppfinnelsen er særlig egnet for behand-ling av nevrologiske sykdommer slik som epilepsi.
Applications Claiming Priority (2)
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NO20053644A NO20053644L (no) | 2000-02-23 | 2005-07-27 | (2S)-2-[(4S)-4-(2,2-difluorvinyl)-2-oksopyrrolidinyl ]butanamid og farmasoytisk preparat |
NO20053645A NO20053645L (no) | 2000-02-23 | 2005-07-27 | (4R)- og (4S)-diastereoisomerer av (2S)-2-[ 2-oksy-4-propylpyrrolidinyl]butanamid og farmasoytisk preparat inneholdende disse |
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