JP4934197B2 - ブルートンチロシンキナーゼ阻害剤 - Google Patents

ブルートンチロシンキナーゼ阻害剤 Download PDF

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JP4934197B2
JP4934197B2 JP2009529166A JP2009529166A JP4934197B2 JP 4934197 B2 JP4934197 B2 JP 4934197B2 JP 2009529166 A JP2009529166 A JP 2009529166A JP 2009529166 A JP2009529166 A JP 2009529166A JP 4934197 B2 JP4934197 B2 JP 4934197B2
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compound
formula
substituted
tyrosine kinase
alkyl
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JP2010504324A (ja
JP2010504324A5 (Direct
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リー・ホニグバーグ
エリック・バーナー
パン・ジェンイン
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Pharmacyclics LLC
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Pharmacyclics LLC
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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  • Urology & Nephrology (AREA)
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  • Neurology (AREA)
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JP2009529166A 2006-09-22 2006-12-28 ブルートンチロシンキナーゼ阻害剤 Active JP4934197B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US82672006P 2006-09-22 2006-09-22
US60/826,720 2006-09-22
US82859006P 2006-10-06 2006-10-06
US60/828,590 2006-10-06
PCT/US2006/049626 WO2008039218A2 (en) 2006-09-22 2006-12-28 Inhibitors of bruton's tyrosine kinase

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JP2010155965A Division JP5193256B2 (ja) 2006-09-22 2010-07-08 ブルートンチロシンキナーゼ阻害剤

Publications (3)

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JP2010504324A JP2010504324A (ja) 2010-02-12
JP2010504324A5 JP2010504324A5 (Direct) 2010-08-26
JP4934197B2 true JP4934197B2 (ja) 2012-05-16

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JP2010155965A Active JP5193256B2 (ja) 2006-09-22 2010-07-08 ブルートンチロシンキナーゼ阻害剤
JP2012049524A Active JP5635544B2 (ja) 2006-09-22 2012-03-06 ブルートンチロシンキナーゼ阻害剤
JP2012286719A Active JP5718890B2 (ja) 2006-09-22 2012-12-28 ブルートンチロシンキナーゼ阻害剤

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JP2012286719A Active JP5718890B2 (ja) 2006-09-22 2012-12-28 ブルートンチロシンキナーゼ阻害剤

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WO2008039218A2 (en) 2008-04-03
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PL2081435T3 (pl) 2016-11-30
US7514444B2 (en) 2009-04-07
US20110257203A1 (en) 2011-10-20
CN102887900B (zh) 2015-04-29
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PT2526933E (pt) 2015-06-23
EP2081435A2 (en) 2009-07-29
LTPA2016034I1 (lt) 2016-12-27
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EP2529622B1 (en) 2018-01-17
ES2616789T3 (es) 2017-06-14
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EP2526771B1 (en) 2016-11-30
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EP2526934A2 (en) 2012-11-28
EP2526933A2 (en) 2012-11-28
AU2006348662B8 (en) 2014-05-29
PT2529621T (pt) 2016-12-23
PT2530083T (pt) 2016-08-01
PL2526771T3 (pl) 2017-06-30
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EP2081435B1 (en) 2016-05-04
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CN102746305B (zh) 2015-02-11
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US20120108612A1 (en) 2012-05-03
US20120095026A1 (en) 2012-04-19
CA2663116A1 (en) 2008-04-03
PL2529621T3 (pl) 2017-06-30
BE2015C016I2 (Direct) 2025-12-10
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LT2529621T (lt) 2017-01-10
US8883435B2 (en) 2014-11-11
NL300728I1 (Direct) 2016-01-26
SI2526933T1 (sl) 2015-07-31
DK2201840T3 (da) 2012-02-20
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