EA200600317A1 - Производные омега-карбоксиарилдифенилмочевины (варианты), фармацевтическая композиция (варианты) и способ лечения и предупреждения заболеваний и состояний с их использованием (варианты) - Google Patents

Производные омега-карбоксиарилдифенилмочевины (варианты), фармацевтическая композиция (варианты) и способ лечения и предупреждения заболеваний и состояний с их использованием (варианты)

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Publication number
EA200600317A1
EA200600317A1 EA200600317A EA200600317A EA200600317A1 EA 200600317 A1 EA200600317 A1 EA 200600317A1 EA 200600317 A EA200600317 A EA 200600317A EA 200600317 A EA200600317 A EA 200600317A EA 200600317 A1 EA200600317 A1 EA 200600317A1
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EA
Eurasian Patent Office
Prior art keywords
options
carboxyaryldiphenylmoleum
omega
diseases
prevention
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EA200600317A
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English (en)
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EA010485B1 (ru
Inventor
Стивен Бойер
Жак Дюма
Бернд Ридль
Скотт Уилхелм
Original Assignee
Байер Фамэсьютиклс Копэрейшн
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34107784&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EA200600317(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Байер Фамэсьютиклс Копэрейшн filed Critical Байер Фамэсьютиклс Копэрейшн
Publication of EA200600317A1 publication Critical patent/EA200600317A1/ru
Publication of EA010485B1 publication Critical patent/EA010485B1/ru

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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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Abstract

Предложено соединение формулы (I), его соли, его пролекарственные формы, его метаболиты, фармацевтические композиции, содержащие данное соединение, и применение данного соединения и композиций для лечения заболеваний, опосредованных raf, VEGFR, PDGFR, р38 и flt-3.
EA200600317A 2003-07-23 2004-07-22 Производное n,n'-дифенилмочевины, фармацевтическая композиция (варианты) и способ лечения и предупреждения заболеваний и состояний с его использованием (варианты) EA010485B1 (ru)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US48910203P 2003-07-23 2003-07-23
US54032604P 2004-02-02 2004-02-02
PCT/US2004/023500 WO2005009961A2 (en) 2003-07-23 2004-07-22 Fluoro substituted omega-carboxyaryl diphenyl urea for the treatment and prevention of diseases and conditions

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