DK1663978T3 - Fluorsubstitueret omega-carboxyaryl-diphenylurinstof til behandling og forebyggelse af sygdomme og lidelser - Google Patents

Fluorsubstitueret omega-carboxyaryl-diphenylurinstof til behandling og forebyggelse af sygdomme og lidelser

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Publication number
DK1663978T3
DK1663978T3 DK04786091T DK04786091T DK1663978T3 DK 1663978 T3 DK1663978 T3 DK 1663978T3 DK 04786091 T DK04786091 T DK 04786091T DK 04786091 T DK04786091 T DK 04786091T DK 1663978 T3 DK1663978 T3 DK 1663978T3
Authority
DK
Denmark
Prior art keywords
carboxyaryl
diphenylurea
fluoro
disorders
diseases
Prior art date
Application number
DK04786091T
Other languages
English (en)
Inventor
Jacques Dumas
Stephen Boyer
Bernd Riedl
Scott Wilhelm
Original Assignee
Bayer Pharmaceuticals Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Family has litigation
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Application filed by Bayer Pharmaceuticals Corp filed Critical Bayer Pharmaceuticals Corp
Application granted granted Critical
Publication of DK1663978T3 publication Critical patent/DK1663978T3/da

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
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    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/62—Oxygen or sulfur atoms
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4412—Non condensed pyridines; Hydrogenated derivatives thereof having oxo groups directly attached to the heterocyclic ring
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    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
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DK04786091T 2003-07-23 2004-07-22 Fluorsubstitueret omega-carboxyaryl-diphenylurinstof til behandling og forebyggelse af sygdomme og lidelser DK1663978T3 (da)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US48910203P 2003-07-23 2003-07-23
US54032604P 2004-02-02 2004-02-02
PCT/US2004/023500 WO2005009961A2 (en) 2003-07-23 2004-07-22 Fluoro substituted omega-carboxyaryl diphenyl urea for the treatment and prevention of diseases and conditions

Publications (1)

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DK1663978T3 true DK1663978T3 (da) 2008-04-07

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US (3) US8637553B2 (da)
EP (1) EP1663978B1 (da)
JP (2) JP4777887B2 (da)
KR (1) KR101139557B1 (da)
CN (2) CN102816113B (da)
AR (3) AR048741A1 (da)
AU (2) AU2004259760B9 (da)
BE (1) BE2013C067I2 (da)
BR (2) BR122016015715B8 (da)
CA (1) CA2532865C (da)
CL (1) CL2004001834A1 (da)
CR (1) CR10193A (da)
CY (2) CY1107094T1 (da)
DE (1) DE602004010407T2 (da)
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