LU92300I2 - Regorafenib et ses sels pharmaceutiquement acceptables (STIVARGA) - Google Patents

Regorafenib et ses sels pharmaceutiquement acceptables (STIVARGA)

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Publication number
LU92300I2
LU92300I2 LU92300C LU92300C LU92300I2 LU 92300 I2 LU92300 I2 LU 92300I2 LU 92300 C LU92300 C LU 92300C LU 92300 C LU92300 C LU 92300C LU 92300 I2 LU92300 I2 LU 92300I2
Authority
LU
Luxembourg
Prior art keywords
stivarga
regorafenib
pharmaceutically acceptable
acceptable salts
compound
Prior art date
Application number
LU92300C
Other languages
English (en)
Other versions
LU92300I9 (fr
Original Assignee
Bayer Healthcare Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34107784&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=LU92300(I2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bayer Healthcare Llc filed Critical Bayer Healthcare Llc
Publication of LU92300I2 publication Critical patent/LU92300I2/fr
Publication of LU92300I9 publication Critical patent/LU92300I9/fr

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
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    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/62—Oxygen or sulfur atoms
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4412—Non condensed pyridines; Hydrogenated derivatives thereof having oxo groups directly attached to the heterocyclic ring
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    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/81—Amides; Imides

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LU92300C 2003-07-23 2013-10-30 Regorafenib et ses sels pharmaceutiquement acceptables (STIVARGA) LU92300I2 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US48910203P 2003-07-23 2003-07-23
US54032604P 2004-02-02 2004-02-02

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