ATE321770T1 - Pseudoerythromycin-derivate - Google Patents

Pseudoerythromycin-derivate

Info

Publication number
ATE321770T1
ATE321770T1 AT00953461T AT00953461T ATE321770T1 AT E321770 T1 ATE321770 T1 AT E321770T1 AT 00953461 T AT00953461 T AT 00953461T AT 00953461 T AT00953461 T AT 00953461T AT E321770 T1 ATE321770 T1 AT E321770T1
Authority
AT
Austria
Prior art keywords
derivatives
pseudoerythromycin
psedoerythromycin
sulfonyl
alkynyl
Prior art date
Application number
AT00953461T
Other languages
English (en)
Inventor
Satoshi Omura
Yuzuru Iwai
Toshiaki Sunazuka
Tohru Nagamitsu
Original Assignee
Kitasato Inst
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Kitasato Inst filed Critical Kitasato Inst
Application granted granted Critical
Publication of ATE321770T1 publication Critical patent/ATE321770T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pulmonology (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AT00953461T 2000-08-17 2000-08-17 Pseudoerythromycin-derivate ATE321770T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
PCT/JP2000/005503 WO2002014338A1 (fr) 2000-08-17 2000-08-17 Nouveaux derives de pseudoerythromycine
EP00953461A EP1256587B1 (de) 2000-08-17 2000-08-17 Pseudoerythromycin-derivate

Publications (1)

Publication Number Publication Date
ATE321770T1 true ATE321770T1 (de) 2006-04-15

Family

ID=11736361

Family Applications (2)

Application Number Title Priority Date Filing Date
AT00953461T ATE321770T1 (de) 2000-08-17 2000-08-17 Pseudoerythromycin-derivate
AT04022619T ATE316977T1 (de) 2000-08-17 2000-08-17 Neue pseudoerythromycin derivate

Family Applications After (1)

Application Number Title Priority Date Filing Date
AT04022619T ATE316977T1 (de) 2000-08-17 2000-08-17 Neue pseudoerythromycin derivate

Country Status (11)

Country Link
US (1) US6734292B1 (de)
EP (2) EP1489090B1 (de)
KR (6) KR20040066184A (de)
AT (2) ATE321770T1 (de)
AU (1) AU2000265939A1 (de)
CA (1) CA2386828C (de)
DE (2) DE60027015T2 (de)
DK (1) DK1489090T3 (de)
ES (2) ES2257720T3 (de)
PT (1) PT1489090E (de)
WO (1) WO2002014338A1 (de)

Families Citing this family (30)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2319693C9 (ru) 1999-01-13 2008-08-20 Байер Копэрейшн Производные мочевины (варианты), фармацевтическая композиция (варианты) и способ лечения заболевания, связанного с ростом раковых клеток (варианты)
ATE538794T1 (de) 1999-01-13 2012-01-15 Bayer Healthcare Llc Gamma carboxyarylsubstituierte diphenylharnstoffverbindungen als p38 kinasehemmer
US8124630B2 (en) 1999-01-13 2012-02-28 Bayer Healthcare Llc ω-carboxyaryl substituted diphenyl ureas as raf kinase inhibitors
US7838541B2 (en) 2002-02-11 2010-11-23 Bayer Healthcare, Llc Aryl ureas with angiogenesis inhibiting activity
US20030216396A1 (en) 2002-02-11 2003-11-20 Bayer Corporation Pyridine, quinoline, and isoquinoline N-oxides as kinase inhibitors
JP2003327536A (ja) * 2002-03-07 2003-11-19 Kitasato Inst:The ヒト免疫不全症候群ウイルスの感染、増殖抑制剤
US20040067896A1 (en) * 2002-07-25 2004-04-08 The Kitasato Institute Novel pseudoerythromycin derivatives
UY28213A1 (es) 2003-02-28 2004-09-30 Bayer Pharmaceuticals Corp Nuevos derivados de cianopiridina útiles en el tratamiento de cáncer y otros trastornos.
WO2004113274A2 (en) 2003-05-20 2004-12-29 Bayer Pharmaceuticals Corporation Diaryl ureas with kinase inhibiting activity
RS52625B (sr) 2003-07-23 2013-06-28 Bayer Healthcare Llc Fluoro supstituisana omega-karboksiaril difenil urea za lečenje i prevenciju bolesti i stanja bolesti
US7419962B2 (en) * 2004-12-07 2008-09-02 Enanta Pharmaceuticals, Inc. 3,6-bicyclolides
US7229972B2 (en) * 2004-12-07 2007-06-12 Enanta Pharmaceuticals, Inc. 3,6-Bicyclolides
EP3290427A1 (de) 2005-08-24 2018-03-07 Melinta Therapeutics, Inc. Triazolverbindungen und verfahren zur herstellung und verwendung davon
CN101326192B (zh) * 2005-10-14 2012-06-20 社团法人北里研究所 新型二氢伪红霉素衍生物
US7407942B2 (en) * 2006-03-29 2008-08-05 Emata Pharmaceuticals, Inc 3,6-bridged 9,12-oxolides
US8097419B2 (en) 2006-09-12 2012-01-17 Longhorn Vaccines & Diagnostics Llc Compositions and method for rapid, real-time detection of influenza A virus (H1N1) swine 2009
US8080645B2 (en) * 2007-10-01 2011-12-20 Longhorn Vaccines & Diagnostics Llc Biological specimen collection/transport compositions and methods
US8652782B2 (en) 2006-09-12 2014-02-18 Longhorn Vaccines & Diagnostics, Llc Compositions and methods for detecting, identifying and quantitating mycobacterial-specific nucleic acids
US20090098527A1 (en) * 2006-09-12 2009-04-16 Fischer Gerald W Biological organism identification product and methods
US9481912B2 (en) 2006-09-12 2016-11-01 Longhorn Vaccines And Diagnostics, Llc Compositions and methods for detecting and identifying nucleic acid sequences in biological samples
US9683256B2 (en) 2007-10-01 2017-06-20 Longhorn Vaccines And Diagnostics, Llc Biological specimen collection and transport system
US11041215B2 (en) 2007-08-24 2021-06-22 Longhorn Vaccines And Diagnostics, Llc PCR ready compositions and methods for detecting and identifying nucleic acid sequences
CA2976814C (en) 2007-08-27 2022-12-13 Longhorn Vaccines & Diagnostics, Llc Immunogenic compositions and methods for treating influenza
US10004799B2 (en) 2007-08-27 2018-06-26 Longhorn Vaccines And Diagnostics, Llc Composite antigenic sequences and vaccines
US11041216B2 (en) 2007-10-01 2021-06-22 Longhorn Vaccines And Diagnostics, Llc Compositions and methods for detecting and quantifying nucleic acid sequences in blood samples
EP2195466B1 (de) 2007-10-01 2012-10-10 Longhorn Vaccines & Diagnostics, LLC Verfahren zum aufbewahren biologischer proben
JP5733601B2 (ja) * 2010-07-13 2015-06-10 国立大学法人 千葉大学 劇症型炎症の予防および/または治療剤
EP2806890A4 (de) 2012-01-26 2015-09-02 Longhorn Vaccines & Diagnostics Llc Zusammengesetzte antigensequenzen und impfstoffe
CA2985652C (en) 2015-05-14 2020-03-10 Gerald W. FISHER Rapid methods for the extraction of nucleic acids from biological samples
CN118139870A (zh) * 2021-09-07 2024-06-04 硕腾服务有限责任公司 免疫调节氮环内酯

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5106961A (en) 1987-05-26 1992-04-21 Eli Lilly And Company Erythromycin ring-contracted derivatives
CA1321581C (en) * 1987-05-26 1993-08-24 Herbert A. Kirst Ring-contracted macrolides
US4920102A (en) * 1988-04-18 1990-04-24 Eli Lilly And Company Method for treating gastrointestinal disorders
AU663089B2 (en) * 1991-04-09 1995-09-28 Abbott Laboratories Macrocyclic lactam prokinetic agents
US5554605A (en) 1991-04-09 1996-09-10 Abbott Laboratories Macrocyclic lactam prokinetic agents
DE4200145A1 (de) * 1992-01-07 1993-07-08 Kali Chemie Pharma Gmbh 7,10-epoxy-oxacyclododecan-derivate, verfahren und zwischenprodukte zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
DE19644195A1 (de) 1996-10-24 1998-04-30 Solvay Pharm Gmbh 10,13,15-Trioxatricyclo[9.2.1.1.·9·.·6·]-pentadecanon-Derivate, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende Arzneimittel
DE19805822B4 (de) * 1998-02-13 2009-02-05 Solvay Pharmaceuticals Gmbh 11-Acetyl-12,13-dioxabicyclo[8.2.1]tridecenon-Derivate, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende Arzneimittel

Also Published As

Publication number Publication date
DE60027015D1 (en) 2006-05-18
EP1256587A1 (de) 2002-11-13
CA2386828A1 (en) 2002-02-21
WO2002014338A1 (fr) 2002-02-21
KR20040066186A (ko) 2004-07-23
EP1256587A4 (de) 2004-01-28
DE60025856T2 (de) 2006-10-19
ES2261224T3 (es) 2006-11-16
ATE316977T1 (de) 2006-02-15
US6734292B1 (en) 2004-05-11
PT1489090E (pt) 2006-05-31
DK1489090T3 (da) 2006-05-22
AU2000265939A1 (en) 2002-02-25
ES2257720T3 (es) 2006-08-01
KR20040066185A (ko) 2004-07-23
KR20040066187A (ko) 2004-07-23
DE60025856D1 (de) 2006-04-13
EP1489090B1 (de) 2006-02-01
KR20040074096A (ko) 2004-08-21
DE60027015T2 (de) 2006-10-05
EP1489090A1 (de) 2004-12-22
CA2386828C (en) 2006-01-24
EP1256587B1 (de) 2006-03-29
KR20040066188A (ko) 2004-07-23
KR20040066184A (ko) 2004-07-23

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