DK2529622T3 - INHIBITORS OF BRUTON-TYROSINKINASE - Google Patents

INHIBITORS OF BRUTON-TYROSINKINASE Download PDF

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Publication number
DK2529622T3
DK2529622T3 DK12166302.5T DK12166302T DK2529622T3 DK 2529622 T3 DK2529622 T3 DK 2529622T3 DK 12166302 T DK12166302 T DK 12166302T DK 2529622 T3 DK2529622 T3 DK 2529622T3
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formula
compound
compounds
cases
btk
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DK12166302.5T
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Danish (da)
English (en)
Inventor
Lee Honigberg
Erik Verner
Zhengying Pan
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Pharmacyclics Llc
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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    • C—CHEMISTRY; METALLURGY
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    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K16/00—Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies
    • C07K16/18—Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies against material from animals or humans
    • C07K16/28—Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies against material from animals or humans against receptors, cell surface antigens or cell surface determinants
    • C07K16/2887—Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies against material from animals or humans against receptors, cell surface antigens or cell surface determinants against CD20
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    • C07K—PEPTIDES
    • C07K2317/00—Immunoglobulins specific features
    • C07K2317/20—Immunoglobulins specific features characterized by taxonomic origin
    • C07K2317/24—Immunoglobulins specific features characterized by taxonomic origin containing regions, domains or residues from different species, e.g. chimeric, humanized or veneered

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  • Health & Medical Sciences (AREA)
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  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
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  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Immunology (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Hematology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Pulmonology (AREA)
  • Neurosurgery (AREA)
  • Dermatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Obesity (AREA)
  • Oncology (AREA)
  • Reproductive Health (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Mycology (AREA)
  • Microbiology (AREA)
  • Hospice & Palliative Care (AREA)
DK12166302.5T 2006-09-22 2006-12-28 INHIBITORS OF BRUTON-TYROSINKINASE DK2529622T3 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US82672006P 2006-09-22 2006-09-22
US82859006P 2006-10-06 2006-10-06
EP06850039.6A EP2081435B1 (en) 2006-09-22 2006-12-28 Inhibitors of bruton's tyrosine kinase

Publications (1)

Publication Number Publication Date
DK2529622T3 true DK2529622T3 (en) 2018-05-07

Family

ID=39225888

Family Applications (7)

Application Number Title Priority Date Filing Date
DK12166302.5T DK2529622T3 (en) 2006-09-22 2006-12-28 INHIBITORS OF BRUTON-TYROSINKINASE
DK12166305.8T DK2526934T3 (en) 2006-09-22 2006-12-28 Inhibitors of Bruton's tyrosine kinase
DK10155834.4T DK2201840T3 (da) 2006-09-22 2006-12-28 Hæmmere af Brutons tyrosinkinase
DK12166298.5T DK2529621T3 (en) 2006-09-22 2006-12-28 Inhibitors of Bruton's tyrosine kinase
DK12166301.7T DK2526933T3 (en) 2006-09-22 2006-12-28 Inhibitors of Bruton's tyrosine kinase
DK06850039.6T DK2081435T3 (en) 2006-09-22 2006-12-28 INHIBITORS OF BRUTON'S TYROSINKINASE
DK12166300.9T DK2526771T3 (en) 2006-09-22 2006-12-28 Inhibitors of Bruton's tyrosine kinase

Family Applications After (6)

Application Number Title Priority Date Filing Date
DK12166305.8T DK2526934T3 (en) 2006-09-22 2006-12-28 Inhibitors of Bruton's tyrosine kinase
DK10155834.4T DK2201840T3 (da) 2006-09-22 2006-12-28 Hæmmere af Brutons tyrosinkinase
DK12166298.5T DK2529621T3 (en) 2006-09-22 2006-12-28 Inhibitors of Bruton's tyrosine kinase
DK12166301.7T DK2526933T3 (en) 2006-09-22 2006-12-28 Inhibitors of Bruton's tyrosine kinase
DK06850039.6T DK2081435T3 (en) 2006-09-22 2006-12-28 INHIBITORS OF BRUTON'S TYROSINKINASE
DK12166300.9T DK2526771T3 (en) 2006-09-22 2006-12-28 Inhibitors of Bruton's tyrosine kinase

Country Status (28)

Country Link
US (49) US7514444B2 (enExample)
EP (11) EP2443929A1 (enExample)
JP (4) JP4934197B2 (enExample)
KR (4) KR20100051863A (enExample)
CN (4) CN101805341B (enExample)
AT (1) ATE531263T1 (enExample)
AU (2) AU2006348662B8 (enExample)
BE (1) BE2015C016I2 (enExample)
BR (2) BRPI0622054B8 (enExample)
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