TWI303636B - Pyrazole compositions useful as protein kinase inhibitors - Google Patents

Pyrazole compositions useful as protein kinase inhibitors Download PDF

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Publication number
TWI303636B
TWI303636B TW090122889A TW90122889A TWI303636B TW I303636 B TWI303636 B TW I303636B TW 090122889 A TW090122889 A TW 090122889A TW 90122889 A TW90122889 A TW 90122889A TW I303636 B TWI303636 B TW I303636B
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group
ring
aliphatic group
alkyl
aliphatic
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TW090122889A
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Chinese (zh)
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Davies Robert
Bebbington Daivd
Knegtel Ronald
Wannamaker Marion
Li Pan
J Forester Cornelia
Lauffer David
Pierce Albert
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Vertex Pharma
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TW090122889A 2000-09-15 2001-09-14 Pyrazole compositions useful as protein kinase inhibitors TWI303636B (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US23279500P 2000-09-15 2000-09-15
US25788700P 2000-12-21 2000-12-21
US28694901P 2001-04-27 2001-04-27

Publications (1)

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TWI303636B true TWI303636B (en) 2008-12-01

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ID=27398347

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TW090122889A TWI303636B (en) 2000-09-15 2001-09-14 Pyrazole compositions useful as protein kinase inhibitors

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US (7) US6638926B2 (enExample)
EP (8) EP1317452B1 (enExample)
JP (9) JP4922539B2 (enExample)
KR (4) KR100876069B1 (enExample)
CN (3) CN100355750C (enExample)
AP (1) AP2003002762A0 (enExample)
AT (8) ATE363284T1 (enExample)
AU (9) AU2001294558A1 (enExample)
BR (1) BR0114088A (enExample)
CA (8) CA2422378C (enExample)
DE (8) DE60124744T2 (enExample)
DK (1) DK1318997T3 (enExample)
ES (3) ES2266259T3 (enExample)
HU (4) HUP0302173A2 (enExample)
IL (6) IL154786A0 (enExample)
MX (8) MXPA03002299A (enExample)
NO (4) NO327708B1 (enExample)
NZ (4) NZ525008A (enExample)
PE (1) PE20020451A1 (enExample)
PL (1) PL361676A1 (enExample)
PT (2) PT1317448E (enExample)
TW (1) TWI303636B (enExample)
WO (8) WO2002022603A1 (enExample)

Cited By (1)

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TWI476192B (zh) * 2009-02-27 2015-03-11 Ambit Biosciences Corp Ｊａｋ激酶調節化合物及其使用方法

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US6982260B1 (en) 1999-11-22 2006-01-03 Warner-Lambert Company Quinazolines and their use for inhibiting cyclin-dependent kinase enzymes
WO2001047922A2 (en) 1999-12-24 2001-07-05 Aventis Pharma Limited Azaindoles
DK1318997T3 (da) * 2000-09-15 2006-09-25 Vertex Pharma Pyrazolforbindelser der er nyttige som proteinkinase-inhibitorer
US6660731B2 (en) * 2000-09-15 2003-12-09 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
US7473691B2 (en) * 2000-09-15 2009-01-06 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
US7105532B2 (en) * 2000-12-19 2006-09-12 Smithkline Beecham Corporation Pyrazolo[3,4-c]pyridines as gsk-3 inhibitors
ATE430742T1 (de) * 2000-12-21 2009-05-15 Smithkline Beecham Corp Pyrimidinamine als angiogenesemodulatoren
HUP0400639A3 (en) 2000-12-21 2010-03-29 Vertex Pharma Pyrazole compounds useful as protein kinase inhibitors and pharmaceutical compositions containing them
US7276523B2 (en) 2001-03-30 2007-10-02 Smithkline Beecham Corporation Aminopyridine derivatives as estrogen receptor modulators
JP4316893B2 (ja) 2001-05-16 2009-08-19 バーテックス ファーマシューティカルズ インコーポレイテッド Ｓｒｃおよび他のプロテインキナーゼのインヒビター
GB0115109D0 (en) 2001-06-21 2001-08-15 Aventis Pharma Ltd Chemical compounds
US6939874B2 (en) 2001-08-22 2005-09-06 Amgen Inc. Substituted pyrimidinyl derivatives and methods of use
US7115617B2 (en) 2001-08-22 2006-10-03 Amgen Inc. Amino-substituted pyrimidinyl derivatives and methods of use
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