TWI303636B - Pyrazole compositions useful as protein kinase inhibitors - Google Patents

Pyrazole compositions useful as protein kinase inhibitors Download PDF

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Publication number
TWI303636B
TWI303636B TW090122889A TW90122889A TWI303636B TW I303636 B TWI303636 B TW I303636B TW 090122889 A TW090122889 A TW 090122889A TW 90122889 A TW90122889 A TW 90122889A TW I303636 B TWI303636 B TW I303636B
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group
ring
aliphatic group
alkyl
aliphatic
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TW090122889A
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Chinese (zh)
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Davies Robert
Bebbington Daivd
Knegtel Ronald
Wannamaker Marion
Li Pan
J Forester Cornelia
Lauffer David
Pierce Albert
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Vertex Pharma
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TW090122889A 2000-09-15 2001-09-14 Pyrazole compositions useful as protein kinase inhibitors TWI303636B (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US23279500P 2000-09-15 2000-09-15
US25788700P 2000-12-21 2000-12-21
US28694901P 2001-04-27 2001-04-27

Publications (1)

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TWI303636B true TWI303636B (en) 2008-12-01

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TW090122889A TWI303636B (en) 2000-09-15 2001-09-14 Pyrazole compositions useful as protein kinase inhibitors

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US (7) US6638926B2 (enExample)
EP (8) EP1317444B1 (enExample)
JP (9) JP2004509115A (enExample)
KR (4) KR100896664B1 (enExample)
CN (3) CN1469875A (enExample)
AP (1) AP2003002762A0 (enExample)
AT (8) ATE346064T1 (enExample)
AU (9) AU2001292670A1 (enExample)
BR (1) BR0114088A (enExample)
CA (8) CA2422380C (enExample)
DE (8) DE60128709T2 (enExample)
DK (1) DK1318997T3 (enExample)
ES (3) ES2266259T3 (enExample)
HU (4) HUP0302172A2 (enExample)
IL (6) IL154784A0 (enExample)
MX (8) MXPA03002293A (enExample)
NO (4) NO20031190L (enExample)
NZ (4) NZ525014A (enExample)
PE (1) PE20020451A1 (enExample)
PL (1) PL361676A1 (enExample)
PT (2) PT1318997E (enExample)
TW (1) TWI303636B (enExample)
WO (8) WO2002022602A2 (enExample)

Cited By (1)

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Publication number Priority date Publication date Assignee Title
TWI476192B (zh) * 2009-02-27 2015-03-11 Ambit Biosciences Corp Ｊａｋ激酶調節化合物及其使用方法

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US6184226B1 (en) * 1998-08-28 2001-02-06 Scios Inc. Quinazoline derivatives as inhibitors of P-38 α
US6982260B1 (en) 1999-11-22 2006-01-03 Warner-Lambert Company Quinazolines and their use for inhibiting cyclin-dependent kinase enzymes
WO2001047922A2 (en) 1999-12-24 2001-07-05 Aventis Pharma Limited Azaindoles
US6638926B2 (en) 2000-09-15 2003-10-28 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
US7473691B2 (en) * 2000-09-15 2009-01-06 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
US6660731B2 (en) * 2000-09-15 2003-12-09 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
WO2002050073A1 (en) * 2000-12-19 2002-06-27 Smithkline Beecham P.L.C. Pyrazolo[3,4-c]pyridines as gsk-3 inhibitors
KR100847169B1 (ko) 2000-12-21 2008-07-17 글락소 그룹 리미티드 혈관형성 조절제로서의 피리미딘아민
CA2432799C (en) * 2000-12-21 2008-08-19 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
WO2002079163A1 (en) * 2001-03-30 2002-10-10 Smithkline Beecham Corporation Aminopyridine derivatives as estrogen receptor modulators
US6884804B2 (en) 2001-05-16 2005-04-26 Vertex Pharmaceuticals Incorporated Inhibitors of Src and other protein kinases
GB0115109D0 (en) 2001-06-21 2001-08-15 Aventis Pharma Ltd Chemical compounds
US6939874B2 (en) 2001-08-22 2005-09-06 Amgen Inc. Substituted pyrimidinyl derivatives and methods of use
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