AP2003002762A0 - Pyrazole compounds useful as protein kinase inhibitors - Google Patents

Pyrazole compounds useful as protein kinase inhibitors

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Publication number
AP2003002762A0
AP2003002762A0 APAP/P/2003/002762A AP2003002762A AP2003002762A0 AP 2003002762 A0 AP2003002762 A0 AP 2003002762A0 AP 2003002762 A AP2003002762 A AP 2003002762A AP 2003002762 A0 AP2003002762 A0 AP 2003002762A0
Authority
AP
ARIPO
Prior art keywords
ring
protein kinase
kinase inhibitors
pyrazole compounds
compounds useful
Prior art date
Application number
APAP/P/2003/002762A
Other languages
English (en)
Inventor
Robert Davies
David Bebbington
Ronald Knegtel
Marion Woods Wannamaker
Pan Li
Cornelia Forster
Albert Pierce
David Kay
Original Assignee
Vertex Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27398347&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AP2003002762(A0) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Vertex Pharma filed Critical Vertex Pharma
Publication of AP2003002762A0 publication Critical patent/AP2003002762A0/en

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    • C07D513/04—Ortho-condensed systems

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  • Diabetes (AREA)
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  • Neurology (AREA)
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APAP/P/2003/002762A 2000-09-15 2001-09-14 Pyrazole compounds useful as protein kinase inhibitors AP2003002762A0 (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US23279500P 2000-09-15 2000-09-15
US25788700P 2000-12-21 2000-12-21
US28694901P 2001-04-27 2001-04-27
PCT/US2001/028940 WO2002022607A1 (en) 2000-09-15 2001-09-14 Pyrazole compounds useful as protein kinase inhibitors

Publications (1)

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AP2003002762A0 true AP2003002762A0 (en) 2003-03-31

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APAP/P/2003/002762A AP2003002762A0 (en) 2000-09-15 2001-09-14 Pyrazole compounds useful as protein kinase inhibitors

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US (7) US6638926B2 (enExample)
EP (8) EP1317444B1 (enExample)
JP (9) JP2004509115A (enExample)
KR (4) KR100896664B1 (enExample)
CN (3) CN1469875A (enExample)
AP (1) AP2003002762A0 (enExample)
AT (8) ATE346064T1 (enExample)
AU (9) AU2001292670A1 (enExample)
BR (1) BR0114088A (enExample)
CA (8) CA2422380C (enExample)
DE (8) DE60128709T2 (enExample)
DK (1) DK1318997T3 (enExample)
ES (3) ES2266259T3 (enExample)
HU (4) HUP0302172A2 (enExample)
IL (6) IL154784A0 (enExample)
MX (8) MXPA03002293A (enExample)
NO (4) NO20031190L (enExample)
NZ (4) NZ525014A (enExample)
PE (1) PE20020451A1 (enExample)
PL (1) PL361676A1 (enExample)
PT (2) PT1318997E (enExample)
TW (1) TWI303636B (enExample)
WO (8) WO2002022602A2 (enExample)

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US6184226B1 (en) * 1998-08-28 2001-02-06 Scios Inc. Quinazoline derivatives as inhibitors of P-38 α
US6982260B1 (en) 1999-11-22 2006-01-03 Warner-Lambert Company Quinazolines and their use for inhibiting cyclin-dependent kinase enzymes
WO2001047922A2 (en) 1999-12-24 2001-07-05 Aventis Pharma Limited Azaindoles
US6638926B2 (en) 2000-09-15 2003-10-28 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
US7473691B2 (en) * 2000-09-15 2009-01-06 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
US6660731B2 (en) * 2000-09-15 2003-12-09 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
WO2002050073A1 (en) * 2000-12-19 2002-06-27 Smithkline Beecham P.L.C. Pyrazolo[3,4-c]pyridines as gsk-3 inhibitors
KR100847169B1 (ko) 2000-12-21 2008-07-17 글락소 그룹 리미티드 혈관형성 조절제로서의 피리미딘아민
CA2432799C (en) * 2000-12-21 2008-08-19 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
WO2002079163A1 (en) * 2001-03-30 2002-10-10 Smithkline Beecham Corporation Aminopyridine derivatives as estrogen receptor modulators
US6884804B2 (en) 2001-05-16 2005-04-26 Vertex Pharmaceuticals Incorporated Inhibitors of Src and other protein kinases
GB0115109D0 (en) 2001-06-21 2001-08-15 Aventis Pharma Ltd Chemical compounds
US6939874B2 (en) 2001-08-22 2005-09-06 Amgen Inc. Substituted pyrimidinyl derivatives and methods of use
US7115617B2 (en) 2001-08-22 2006-10-03 Amgen Inc. Amino-substituted pyrimidinyl derivatives and methods of use
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