NZ595230A - Pyrimidinopyrazole derivatives as inhibitors of Bruton's tyrosine kinase - Google Patents
Pyrimidinopyrazole derivatives as inhibitors of Bruton's tyrosine kinaseInfo
- Publication number
- NZ595230A NZ595230A NZ595230A NZ59523006A NZ595230A NZ 595230 A NZ595230 A NZ 595230A NZ 595230 A NZ595230 A NZ 595230A NZ 59523006 A NZ59523006 A NZ 59523006A NZ 595230 A NZ595230 A NZ 595230A
- Authority
- NZ
- New Zealand
- Prior art keywords
- inhibitors
- conditions
- btk
- bruton
- tyrosine kinase
- Prior art date
Links
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
- A61K31/52—Purines, e.g. adenine
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
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- C07D487/04—Ortho-condensed systems
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K16/00—Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies
- C07K16/18—Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies against material from animals or humans
- C07K16/28—Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies against material from animals or humans against receptors, cell surface antigens or cell surface determinants
- C07K16/2887—Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies against material from animals or humans against receptors, cell surface antigens or cell surface determinants against CD20
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- C07K—PEPTIDES
- C07K2317/00—Immunoglobulins specific features
- C07K2317/20—Immunoglobulins specific features characterized by taxonomic origin
- C07K2317/24—Immunoglobulins specific features characterized by taxonomic origin containing regions, domains or residues from different species, e.g. chimeric, humanized or veneered
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Epidemiology (AREA)
- Immunology (AREA)
- Diabetes (AREA)
- Endocrinology (AREA)
- Hematology (AREA)
- Neurology (AREA)
- Urology & Nephrology (AREA)
- Physical Education & Sports Medicine (AREA)
- Neurosurgery (AREA)
- Pulmonology (AREA)
- Biomedical Technology (AREA)
- Rheumatology (AREA)
- Dermatology (AREA)
- Obesity (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Oncology (AREA)
- Reproductive Health (AREA)
- Genetics & Genomics (AREA)
- Microbiology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Molecular Biology (AREA)
- Biophysics (AREA)
- Biochemistry (AREA)
- Mycology (AREA)
- Emergency Medicine (AREA)
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| NZ601278A NZ601278A (en) | 2006-09-22 | 2006-12-28 | Inhibitors of Bruton's tyrosine kinase |
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US82672006P | 2006-09-22 | 2006-09-22 | |
| US82859006P | 2006-10-06 | 2006-10-06 | |
| PCT/US2006/049626 WO2008039218A2 (en) | 2006-09-22 | 2006-12-28 | Inhibitors of bruton's tyrosine kinase |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| NZ595230A true NZ595230A (en) | 2013-02-22 |
Family
ID=39225888
Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NZ595230A NZ595230A (en) | 2006-09-22 | 2006-12-28 | Pyrimidinopyrazole derivatives as inhibitors of Bruton's tyrosine kinase |
| NZ601278A NZ601278A (en) | 2006-09-22 | 2006-12-28 | Inhibitors of Bruton's tyrosine kinase |
| NZ575650A NZ575650A (en) | 2006-09-22 | 2006-12-28 | Pyrimidinopyrazole derivatives as inhibitors of Bruton's tyrosine kinase |
Family Applications After (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NZ601278A NZ601278A (en) | 2006-09-22 | 2006-12-28 | Inhibitors of Bruton's tyrosine kinase |
| NZ575650A NZ575650A (en) | 2006-09-22 | 2006-12-28 | Pyrimidinopyrazole derivatives as inhibitors of Bruton's tyrosine kinase |
Country Status (28)
| Country | Link |
|---|---|
| US (49) | US7514444B2 (OSRAM) |
| EP (11) | EP2529622B1 (OSRAM) |
| JP (4) | JP4934197B2 (OSRAM) |
| KR (4) | KR101464424B1 (OSRAM) |
| CN (4) | CN101805341B (OSRAM) |
| AT (1) | ATE531263T1 (OSRAM) |
| AU (2) | AU2006348662B8 (OSRAM) |
| BE (1) | BE2015C016I2 (OSRAM) |
| BR (2) | BRPI0622054B8 (OSRAM) |
| CA (3) | CA3180977A1 (OSRAM) |
| CY (11) | CY1112513T1 (OSRAM) |
| DK (7) | DK2526934T3 (OSRAM) |
| EA (3) | EA020001B1 (OSRAM) |
| ES (8) | ES2585902T3 (OSRAM) |
| FR (1) | FR15C0029I2 (OSRAM) |
| HU (10) | HUE031334T2 (OSRAM) |
| IL (1) | IL197550A0 (OSRAM) |
| LT (7) | LT2530083T (OSRAM) |
| LU (3) | LU92692I2 (OSRAM) |
| MX (3) | MX2009003122A (OSRAM) |
| NL (1) | NL300728I2 (OSRAM) |
| NZ (3) | NZ595230A (OSRAM) |
| PL (8) | PL2201840T3 (OSRAM) |
| PT (7) | PT2529622T (OSRAM) |
| SG (2) | SG166093A1 (OSRAM) |
| SI (8) | SI2530083T1 (OSRAM) |
| WO (1) | WO2008039218A2 (OSRAM) |
| ZA (4) | ZA200901784B (OSRAM) |
Families Citing this family (559)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2308879A1 (en) | 2004-04-02 | 2011-04-13 | OSI Pharmaceuticals, Inc. | 6,6-bicyclic ring substituted heterobicyclic protein kinase inhibitors |
| WO2007002093A2 (en) * | 2005-06-21 | 2007-01-04 | Infinity Discovery, Inc. | Ansamycin formulations and methods of use thereof |
| AU2007254179B2 (en) * | 2006-05-18 | 2013-03-21 | Pharmacyclics Llc | Intracellular kinase inhibitors |
| CA2660086C (en) * | 2006-08-16 | 2014-09-16 | Novartis Ag | Method of making solid dispersions of highly crystalline therapeutic compounds |
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