KR100229294B1 - 퀴나졸린 유도체 - Google Patents

퀴나졸린 유도체 Download PDF

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Publication number
KR100229294B1
KR100229294B1 KR1019930000645A KR930000645A KR100229294B1 KR 100229294 B1 KR100229294 B1 KR 100229294B1 KR 1019930000645 A KR1019930000645 A KR 1019930000645A KR 930000645 A KR930000645 A KR 930000645A KR 100229294 B1 KR100229294 B1 KR 100229294B1
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KR
South Korea
Prior art keywords
alkyl
alkoxy
amino
alkylamino
hydroxy
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
KR1019930000645A
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English (en)
Korean (ko)
Other versions
KR930016407A (ko
Inventor
바커앤드류존
Original Assignee
사라 엔 람베쓰
제네카 리미티드
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB929201095A external-priority patent/GB9201095D0/en
Priority claimed from GB929213572A external-priority patent/GB9213572D0/en
Priority claimed from GB929223735A external-priority patent/GB9223735D0/en
Application filed by 사라 엔 람베쓰, 제네카 리미티드 filed Critical 사라 엔 람베쓰
Publication of KR930016407A publication Critical patent/KR930016407A/ko
Application granted granted Critical
Publication of KR100229294B1 publication Critical patent/KR100229294B1/ko
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/94—Nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04—Ortho-condensed systems

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Treatments For Attaching Organic Compounds To Fibrous Goods (AREA)
  • Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
  • Cosmetics (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
KR1019930000645A 1992-01-20 1993-01-20 퀴나졸린 유도체 Expired - Lifetime KR100229294B1 (ko)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
GB9201095.8 1992-01-20
GB929201095A GB9201095D0 (en) 1992-01-20 1992-01-20 Quinazoline derivatives
GB929213572A GB9213572D0 (en) 1992-06-26 1992-06-26 Quinazoline derivatives
GB9213572.2 1992-11-12
GB929223735A GB9223735D0 (en) 1992-11-12 1992-11-12 Quinazoline derivatives
GB9223735.3 1992-11-12

Publications (2)

Publication Number Publication Date
KR930016407A KR930016407A (ko) 1993-08-26
KR100229294B1 true KR100229294B1 (ko) 1999-11-01

Family

ID=27266013

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019930000645A Expired - Lifetime KR100229294B1 (ko) 1992-01-20 1993-01-20 퀴나졸린 유도체

Country Status (22)

Country Link
US (2) US5457105A (enExample)
EP (1) EP0566226B1 (enExample)
KR (1) KR100229294B1 (enExample)
AT (1) ATE130000T1 (enExample)
AU (1) AU661533B2 (enExample)
CA (1) CA2086968C (enExample)
CZ (1) CZ282038B6 (enExample)
DE (1) DE69300754T2 (enExample)
DK (1) DK0566226T3 (enExample)
ES (1) ES2078798T3 (enExample)
FI (1) FI111631B (enExample)
GB (1) GB9300059D0 (enExample)
GR (1) GR3018143T3 (enExample)
HK (1) HK36497A (enExample)
HU (2) HU221622B1 (enExample)
IL (1) IL104479A (enExample)
NO (1) NO301541B1 (enExample)
NZ (1) NZ245662A (enExample)
RU (1) RU2127263C1 (enExample)
SK (1) SK281551B6 (enExample)
TW (1) TW283146B (enExample)
UA (1) UA34426C2 (enExample)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR100753385B1 (ko) 2003-06-10 2007-08-30 에프. 호프만-라 로슈 아게 1,3,4-트리아자-페날린 및 1,3,4,6-테트라아자페날린유도체

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