KR101520086B1 - 1´,3´-이치환된-4-페닐-3,4,5,6-테트라히드로-2h,1´h-[1,4´]비피리디닐-2´-온 - Google Patents
1´,3´-이치환된-4-페닐-3,4,5,6-테트라히드로-2h,1´h-[1,4´]비피리디닐-2´-온 Download PDFInfo
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- KR101520086B1 KR101520086B1 KR1020147000745A KR20147000745A KR101520086B1 KR 101520086 B1 KR101520086 B1 KR 101520086B1 KR 1020147000745 A KR1020147000745 A KR 1020147000745A KR 20147000745 A KR20147000745 A KR 20147000745A KR 101520086 B1 KR101520086 B1 KR 101520086B1
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
- A61K31/4545—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/444—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
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- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
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- C07D491/107—Spiro-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP07116390 | 2007-09-14 | ||
| EP07116390.1 | 2007-09-14 | ||
| PCT/EP2008/007551 WO2009033704A1 (en) | 2007-09-14 | 2008-09-12 | 1',3'-disubstituted-4-phenyl-3,4,5,6-tetrahydro-2h, 1'h-[1, 4'] bipyridinyl-2'-ones |
Related Parent Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1020107008034A Division KR101533440B1 (ko) | 2007-09-14 | 2008-09-12 | 1´,3´-이치환된-4-페닐-3,4,5,6-테트라히드로-2h,1´h-[1,4´]비피리디닐-2´-온 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| KR20140034904A KR20140034904A (ko) | 2014-03-20 |
| KR101520086B1 true KR101520086B1 (ko) | 2015-05-14 |
Family
ID=39930548
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1020107008034A Active KR101533440B1 (ko) | 2007-09-14 | 2008-09-12 | 1´,3´-이치환된-4-페닐-3,4,5,6-테트라히드로-2h,1´h-[1,4´]비피리디닐-2´-온 |
| KR1020147000745A Active KR101520086B1 (ko) | 2007-09-14 | 2008-09-12 | 1´,3´-이치환된-4-페닐-3,4,5,6-테트라히드로-2h,1´h-[1,4´]비피리디닐-2´-온 |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1020107008034A Active KR101533440B1 (ko) | 2007-09-14 | 2008-09-12 | 1´,3´-이치환된-4-페닐-3,4,5,6-테트라히드로-2h,1´h-[1,4´]비피리디닐-2´-온 |
Country Status (29)
| Country | Link |
|---|---|
| US (6) | US9114138B2 (enExample) |
| EP (1) | EP2203439B1 (enExample) |
| JP (1) | JP5133416B2 (enExample) |
| KR (2) | KR101533440B1 (enExample) |
| CN (2) | CN103342695B (enExample) |
| AR (1) | AR068511A1 (enExample) |
| AT (1) | ATE496906T1 (enExample) |
| AU (1) | AU2008297878B2 (enExample) |
| BR (1) | BRPI0816767B8 (enExample) |
| CA (1) | CA2696948C (enExample) |
| CL (1) | CL2008002745A1 (enExample) |
| CY (1) | CY1111219T1 (enExample) |
| DE (1) | DE602008004794D1 (enExample) |
| DK (1) | DK2203439T3 (enExample) |
| EA (1) | EA017648B1 (enExample) |
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| IL (2) | IL204032A (enExample) |
| MX (1) | MX2010002536A (enExample) |
| MY (1) | MY152078A (enExample) |
| NZ (1) | NZ584145A (enExample) |
| PL (1) | PL2203439T3 (enExample) |
| PT (1) | PT2203439E (enExample) |
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| WO (1) | WO2009033704A1 (enExample) |
| ZA (1) | ZA201001151B (enExample) |
Families Citing this family (27)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0420722D0 (en) | 2004-09-17 | 2004-10-20 | Addex Pharmaceuticals Sa | Novel allosteric modulators |
| TWI417095B (zh) | 2006-03-15 | 2013-12-01 | Janssen Pharmaceuticals Inc | 1,4-二取代之3-氰基-吡啶酮衍生物及其作為mGluR2-受體之正向異位性調節劑之用途 |
| TW200845978A (en) | 2007-03-07 | 2008-12-01 | Janssen Pharmaceutica Nv | 3-cyano-4-(4-tetrahydropyran-phenyl)-pyridin-2-one derivatives |
| TW200900065A (en) | 2007-03-07 | 2009-01-01 | Janssen Pharmaceutica Nv | 3-cyano-4-(4-pyridinyloxy-phenyl)-pyridin-2-one derivatives |
| JP5433579B2 (ja) | 2007-09-14 | 2014-03-05 | ジャンセン ファーマシューティカルズ, インコーポレイテッド. | 1,3−二置換−4−フェニル−1h−ピリジン−2−オン |
| ATE516272T1 (de) | 2007-09-14 | 2011-07-15 | Ortho Mcneil Janssen Pharm | 1,3-disubstituierte 4-(aryl-x-phenyl)-1h-pyridin- 2-one |
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