SG10201605472WA - Certain Chemical Entities, Compositions And Methods - Google Patents

Certain Chemical Entities, Compositions And Methods

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Publication number
SG10201605472WA
SG10201605472WA SG10201605472WA SG10201605472WA SG10201605472WA SG 10201605472W A SG10201605472W A SG 10201605472WA SG 10201605472W A SG10201605472W A SG 10201605472WA SG 10201605472W A SG10201605472W A SG 10201605472WA SG 10201605472W A SG10201605472W A SG 10201605472WA
Authority
SG
Singapore
Prior art keywords
compositions
methods
chemical entities
certain chemical
certain
Prior art date
Application number
SG10201605472WA
Other languages
English (en)
Inventor
Pingda Ren
Yi Liu
Troy Edward Wilson
Liansheng Li
Katrina Chan
Christian Rommel
Original Assignee
Intellikine Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Intellikine Llc filed Critical Intellikine Llc
Publication of SG10201605472WA publication Critical patent/SG10201605472WA/en

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    • C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/04—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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