BRPI0516915A - derivados de tiazol substituìdos por 5-carboxamido que interagem com canais de ìons, particularmante com canais de ìons da famìlia kv - Google Patents
derivados de tiazol substituìdos por 5-carboxamido que interagem com canais de ìons, particularmante com canais de ìons da famìlia kvInfo
- Publication number
- BRPI0516915A BRPI0516915A BRPI0516915-1A BRPI0516915A BRPI0516915A BR PI0516915 A BRPI0516915 A BR PI0516915A BR PI0516915 A BRPI0516915 A BR PI0516915A BR PI0516915 A BRPI0516915 A BR PI0516915A
- Authority
- BR
- Brazil
- Prior art keywords
- ion channels
- interact
- compounds
- family
- thiazole derivatives
- Prior art date
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- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/32—One oxygen, sulfur or nitrogen atom
- C07D239/42—One nitrogen atom
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Abstract
DERIVADOS DE TIAZOL SUBSTITUIDOS POR 5- CARBOXAMIDO QUE INTERAGEM COM CANAIS DE ìONS, PARTICULARMENTE COM CANAIS DE ìONS DA Família Kv A presente invenção refere-se a compostos que interagem com canais de íons. Particularmente, a invenção refere-se a compostos que têm a fórmula estrutural (I), (II), (III) ou (IV), seus estereoisómeros, tautómeros, racêmicos, pró-medicamentos, metabólitos, ou um sal e/ou um solvato farmaceuticamente aceitáveis dos mesmos, em que X, Y¹, Y¹, R¹, n, R³, R¬8¬, R¬9¬ R¬10¬, L¹, L², Ar¹ e Ar² são definidos na reivindicação 1. A invenção também de refere aos métodos para a preparação dos ditos compostos, às composições farmacêuticas que compreendem os ditos compostos, e ao uso dos ditos compostos nos métodos para o tratamento do corpo de seres humanos e animais.
Applications Claiming Priority (5)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US63207204P | 2004-12-01 | 2004-12-01 | |
EP04447268 | 2004-12-01 | ||
US68691205P | 2005-06-03 | 2005-06-03 | |
EP05077177 | 2005-09-22 | ||
PCT/EP2005/056390 WO2006058905A1 (en) | 2004-12-01 | 2005-12-01 | 5-CARBOXAMIDO SUBSTITUTED THIAZOLE DERIVATIVES THAT INTERACT WITH ION CHANNELS, IN PARTICULAR WITH ION CHANNELS FROM THE Kv FAMILY |
Publications (1)
Publication Number | Publication Date |
---|---|
BRPI0516915A true BRPI0516915A (pt) | 2008-03-11 |
Family
ID=36084802
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
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BRPI0516915-1A BRPI0516915A (pt) | 2004-12-01 | 2005-12-01 | derivados de tiazol substituìdos por 5-carboxamido que interagem com canais de ìons, particularmante com canais de ìons da famìlia kv |
Country Status (11)
Country | Link |
---|---|
US (1) | US20080125432A1 (pt) |
EP (1) | EP1819330A1 (pt) |
JP (1) | JP2008521862A (pt) |
KR (1) | KR20070094754A (pt) |
CN (1) | CN101098698A (pt) |
AU (1) | AU2005311251A1 (pt) |
BR (1) | BRPI0516915A (pt) |
CA (1) | CA2588517A1 (pt) |
MX (1) | MX2007006109A (pt) |
NO (1) | NO20073357L (pt) |
WO (1) | WO2006058905A1 (pt) |
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-
2005
- 2005-12-01 WO PCT/EP2005/056390 patent/WO2006058905A1/en active Application Filing
- 2005-12-01 KR KR1020077015118A patent/KR20070094754A/ko not_active Application Discontinuation
- 2005-12-01 BR BRPI0516915-1A patent/BRPI0516915A/pt not_active IP Right Cessation
- 2005-12-01 EP EP05818954A patent/EP1819330A1/en not_active Withdrawn
- 2005-12-01 JP JP2007543849A patent/JP2008521862A/ja not_active Withdrawn
- 2005-12-01 US US11/792,030 patent/US20080125432A1/en not_active Abandoned
- 2005-12-01 AU AU2005311251A patent/AU2005311251A1/en not_active Abandoned
- 2005-12-01 CA CA002588517A patent/CA2588517A1/en not_active Abandoned
- 2005-12-01 MX MX2007006109A patent/MX2007006109A/es not_active Application Discontinuation
- 2005-12-01 CN CNA2005800460095A patent/CN101098698A/zh active Pending
-
2007
- 2007-06-29 NO NO20073357A patent/NO20073357L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
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JP2008521862A (ja) | 2008-06-26 |
US20080125432A1 (en) | 2008-05-29 |
NO20073357L (no) | 2007-08-30 |
MX2007006109A (es) | 2007-10-04 |
CN101098698A (zh) | 2008-01-02 |
AU2005311251A1 (en) | 2006-06-08 |
CA2588517A1 (en) | 2006-06-08 |
KR20070094754A (ko) | 2007-09-21 |
WO2006058905A1 (en) | 2006-06-08 |
EP1819330A1 (en) | 2007-08-22 |
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