PL214988B1 - Zwiazek 2,4-pirymidynodiaminy, kompozycja zawierajaca ten zwiazek oraz zastosowanie tego zwiazku - Google Patents

Zwiazek 2,4-pirymidynodiaminy, kompozycja zawierajaca ten zwiazek oraz zastosowanie tego zwiazku

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Publication number
PL214988B1
PL214988B1 PL373530A PL37353003A PL214988B1 PL 214988 B1 PL214988 B1 PL 214988B1 PL 373530 A PL373530 A PL 373530A PL 37353003 A PL37353003 A PL 37353003A PL 214988 B1 PL214988 B1 PL 214988B1
Authority
PL
Poland
Prior art keywords
compound
fluoro
chloro
group
pyrimidinamine
Prior art date
Application number
PL373530A
Other languages
English (en)
Polish (pl)
Other versions
PL373530A1 (en
Inventor
Rajinder Singh
Ankush Argade
Donald G. Payan
Susan Molineaux
Sacha J. Holland
Jeffrey Clough
Holger Keim
Somasekhar Bhamidipati
Catherine Sylvain
Weigun Li
Alexander B. Rossi
Original Assignee
Rigel Pharmaceuticals
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=32996332&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PL214988(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Rigel Pharmaceuticals filed Critical Rigel Pharmaceuticals
Publication of PL373530A1 publication Critical patent/PL373530A1/xx
Publication of PL214988B1 publication Critical patent/PL214988B1/pl

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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A—HUMAN NECESSITIES
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    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
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