PE20040197A1 - Pirazolopiridinas sustituidas con carbamato - Google Patents

Pirazolopiridinas sustituidas con carbamato

Info

Publication number
PE20040197A1
PE20040197A1 PE2003000444A PE2003000444A PE20040197A1 PE 20040197 A1 PE20040197 A1 PE 20040197A1 PE 2003000444 A PE2003000444 A PE 2003000444A PE 2003000444 A PE2003000444 A PE 2003000444A PE 20040197 A1 PE20040197 A1 PE 20040197A1
Authority
PE
Peru
Prior art keywords
methyl
carbamate
pyrazolopyridines
substituted
compounds
Prior art date
Application number
PE2003000444A
Other languages
English (en)
Spanish (es)
Inventor
Cristina Alonso-Alija
Erwin Bischoff
Achim Feurer
Stefan Weigand
Elke Stahl
Johannes-Peter Stasch
Klaus Munter
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=29265155&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PE20040197(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of PE20040197A1 publication Critical patent/PE20040197A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/06—Antiglaucoma agents or miotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/02—Non-specific cardiovascular stimulants, e.g. drugs for syncope, antihypotensives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Epidemiology (AREA)
  • Reproductive Health (AREA)
  • Endocrinology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Psychiatry (AREA)
  • Rheumatology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Ophthalmology & Optometry (AREA)
  • Urology & Nephrology (AREA)
  • Pain & Pain Management (AREA)
  • Psychology (AREA)
  • Hospice & Palliative Care (AREA)
  • Vascular Medicine (AREA)
  • Pregnancy & Childbirth (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
PE2003000444A 2002-05-08 2003-05-07 Pirazolopiridinas sustituidas con carbamato PE20040197A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE10220570A DE10220570A1 (de) 2002-05-08 2002-05-08 Carbamat-substituierte Pyrazolopyridine

Publications (1)

Publication Number Publication Date
PE20040197A1 true PE20040197A1 (es) 2004-04-22

Family

ID=29265155

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2003000444A PE20040197A1 (es) 2002-05-08 2003-05-07 Pirazolopiridinas sustituidas con carbamato

Country Status (38)

Country Link
US (1) US7173037B2 (OSRAM)
EP (1) EP1506193B3 (OSRAM)
JP (1) JP4455321B2 (OSRAM)
KR (1) KR101011864B1 (OSRAM)
CN (1) CN1330649C (OSRAM)
AR (1) AR039789A1 (OSRAM)
AT (1) ATE330957T1 (OSRAM)
AU (1) AU2003233061B2 (OSRAM)
BE (1) BE2014C030I2 (OSRAM)
BR (1) BRPI0309855B8 (OSRAM)
CA (1) CA2485143C (OSRAM)
CU (1) CU23453B7 (OSRAM)
CY (2) CY1105579T1 (OSRAM)
DE (2) DE10220570A1 (OSRAM)
DK (1) DK1506193T3 (OSRAM)
DO (1) DOP2003000639A (OSRAM)
EC (1) ECSP045414A (OSRAM)
ES (1) ES2268363T3 (OSRAM)
FR (1) FR14C0032I2 (OSRAM)
GT (1) GT200300101A (OSRAM)
HR (1) HRP20041166B1 (OSRAM)
IL (1) IL164958A (OSRAM)
LU (1) LU92419I2 (OSRAM)
MX (1) MXPA04011003A (OSRAM)
MY (1) MY136841A (OSRAM)
NL (1) NL300659I2 (OSRAM)
NO (3) NO329105B1 (OSRAM)
NZ (1) NZ536417A (OSRAM)
PE (1) PE20040197A1 (OSRAM)
PL (1) PL214985B1 (OSRAM)
PT (1) PT1506193E (OSRAM)
RU (1) RU2339638C9 (OSRAM)
SI (1) SI1506193T1 (OSRAM)
TW (1) TWI282792B (OSRAM)
UA (1) UA78314C2 (OSRAM)
UY (1) UY27793A1 (OSRAM)
WO (1) WO2003095451A1 (OSRAM)
ZA (1) ZA200408925B (OSRAM)

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DE102005031575A1 (de) * 2005-07-06 2007-01-11 Bayer Healthcare Ag Verwendung von Aktivatoren der löslichen Guanylatzyklase zur Förderung der Wundheilung
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DE102007054786A1 (de) 2007-11-16 2009-05-20 Bayer Healthcare Ag Trisubstituierte Furopyrimidine und ihre Verwendung
DE102007061766A1 (de) 2007-12-20 2009-06-25 Bayer Healthcare Ag 4-(4-Cyano-2-thioaryl)-dihydropyrimidinone und ihre Verwendung
DE102008052013A1 (de) 2008-10-17 2010-04-22 Bayer Schering Pharma Aktiengesellschaft 4-(4-Cyano-2-thioaryl)-dihydropyrimidinone und ihre Verwendung
DE102007061763A1 (de) * 2007-12-20 2009-06-25 Bayer Healthcare Ag Substituierte azabicyclische Verbindungen und ihre Verwendung
DE102007061756A1 (de) 2007-12-20 2009-06-25 Bayer Healthcare Ag Substituierte 4-Aminopyrimidin-5-carbonsäuren und ihre Verwendung
DE102007061764A1 (de) 2007-12-20 2009-06-25 Bayer Healthcare Ag Anellierte Cyanopyridine und ihre Verwendung
DE102007061757A1 (de) 2007-12-20 2009-06-25 Bayer Healthcare Ag Substituierte 2-Phenylpyrimidin-5-carbonsäuren und ihre Verwendung
DE102008022521A1 (de) 2008-05-07 2009-11-12 Bayer Schering Pharma Aktiengesellschaft 1,4-Diaryl-pyrimidopyridazin-2,5-dione und ihre Verwendung
DE102008007400A1 (de) 2008-02-04 2009-08-06 Bayer Healthcare Ag Substituierte Furane und ihre Verwendung
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DE102008060967A1 (de) 2008-12-06 2010-06-10 Bayer Schering Pharma Aktiengesellschaft Substituierte Phenylsulfonyltriazolone und ihre Verwendung
DE102008062566A1 (de) 2008-12-16 2010-06-17 Bayer Schering Pharma Aktiengesellschaft Aminosäureester-Prodrugs und ihre Verwendung
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EP1506193B1 (de) 2006-06-21
MY136841A (en) 2008-11-28
CA2485143C (en) 2011-04-19
HK1082247A1 (en) 2006-06-02
DK1506193T3 (da) 2006-10-09
CN1330649C (zh) 2007-08-08
US20060052397A1 (en) 2006-03-09
TWI282792B (en) 2007-06-21
WO2003095451A1 (de) 2003-11-20
NO2025058I1 (no) 2025-12-12
DE10220570A1 (de) 2003-11-20
NZ536417A (en) 2006-08-31
JP4455321B2 (ja) 2010-04-21
ZA200408925B (en) 2006-01-25
EP1506193A1 (de) 2005-02-16
AR039789A1 (es) 2005-03-02
CY2014018I2 (el) 2015-12-09
BE2014C030I2 (OSRAM) 2022-08-09
CU23453B7 (es) 2009-12-01
US7173037B2 (en) 2007-02-06
CY1105579T1 (el) 2010-07-28
NO2014018I2 (no) 2015-08-31
DE50303960D1 (de) 2006-08-03
TW200404797A (en) 2004-04-01
SI1506193T1 (sl) 2006-12-31
FR14C0032I2 (fr) 2014-11-21
AU2003233061B2 (en) 2009-09-03
UY27793A1 (es) 2003-12-31
DOP2003000639A (es) 2003-11-15
IL164958A (en) 2010-05-17
PT1506193E (pt) 2006-10-31
NL300659I2 (OSRAM) 2017-02-02
NO20045277L (no) 2004-12-01
PL373336A1 (pl) 2005-08-22
BRPI0309855B8 (pt) 2021-05-25
RU2339638C2 (ru) 2008-11-27
CN1665811A (zh) 2005-09-07
NO329105B1 (no) 2010-08-23
ES2268363T3 (es) 2007-03-16
ECSP045414A (es) 2005-01-03
BR0309855A (pt) 2005-03-01
IL164958A0 (en) 2005-12-18
CA2485143A1 (en) 2003-11-20
KR20050003415A (ko) 2005-01-10
NO2014018I1 (no) 2014-07-18
HRP20041166A2 (en) 2005-08-31
CY2014018I1 (el) 2015-12-09
ATE330957T1 (de) 2006-07-15
RU2339638C9 (ru) 2009-09-20
AU2003233061A1 (en) 2003-11-11
BRPI0309855B1 (pt) 2018-10-16
RU2004136277A (ru) 2005-06-27
GT200300101A (es) 2004-03-08
MXPA04011003A (es) 2005-02-14
HRP20041166B1 (hr) 2013-05-31
KR101011864B1 (ko) 2011-02-01
JP2005531553A (ja) 2005-10-20

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