CZ295145B6 - Derivát chinazolinu - Google Patents

Derivát chinazolinu Download PDF

Info

Publication number
CZ295145B6
CZ295145B6 CZ19972067A CZ206797A CZ295145B6 CZ 295145 B6 CZ295145 B6 CZ 295145B6 CZ 19972067 A CZ19972067 A CZ 19972067A CZ 206797 A CZ206797 A CZ 206797A CZ 295145 B6 CZ295145 B6 CZ 295145B6
Authority
CZ
Czechia
Prior art keywords
hydrocarbyl
carbon atoms
group
methoxyethoxy
halogen
Prior art date
Application number
CZ19972067A
Other languages
Czech (cs)
English (en)
Inventor
Rodney Caughren Schnur
Lee Daniel Arnold
Original Assignee
Osi Pharmaceuticals, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=23636708&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CZ295145(B6) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Osi Pharmaceuticals, Inc. filed Critical Osi Pharmaceuticals, Inc.
Publication of CZ295145B6 publication Critical patent/CZ295145B6/cs

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/94—Nitrogen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/08—Drugs for disorders of the urinary system of the prostate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Urology & Nephrology (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
CZ19972067A 1995-03-30 1996-03-29 Derivát chinazolinu CZ295145B6 (cs)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US41330095A 1995-03-30 1995-03-30
PCT/IB1995/000436 WO1996030347A1 (en) 1995-03-30 1995-06-06 Quinazoline derivatives

Publications (1)

Publication Number Publication Date
CZ295145B6 true CZ295145B6 (cs) 2005-06-15

Family

ID=23636708

Family Applications (2)

Application Number Title Priority Date Filing Date
CZ19972067A CZ295145B6 (cs) 1995-03-30 1996-03-29 Derivát chinazolinu
CZ1996931A CZ294967B6 (cs) 1995-03-30 1996-03-29 4-(Substituovaný fenylamino)chinazolinové deriváty, způsob jejich výroby a použití a farmaceutické prostředky na jejich bázi

Family Applications After (1)

Application Number Title Priority Date Filing Date
CZ1996931A CZ294967B6 (cs) 1995-03-30 1996-03-29 4-(Substituovaný fenylamino)chinazolinové deriváty, způsob jejich výroby a použití a farmaceutické prostředky na jejich bázi

Country Status (43)

Country Link
EP (5) EP3103799B1 (h)
JP (1) JP3088018B2 (h)
KR (1) KR100232335B1 (h)
CN (1) CN1066142C (h)
AP (1) AP735A (h)
AR (1) AR002723A1 (h)
AT (2) ATE446955T1 (h)
AU (2) AU703638B2 (h)
BR (1) BR9601200B1 (h)
CA (1) CA2216796C (h)
CO (1) CO4410333A1 (h)
CZ (2) CZ295145B6 (h)
DE (3) DE122005000053I2 (h)
DK (1) DK0817775T3 (h)
EG (1) EG24229A (h)
ES (2) ES2332984T3 (h)
FI (1) FI120646B (h)
FR (1) FR06C0010I2 (h)
GR (1) GR3037070T3 (h)
HR (1) HRP960147B1 (h)
HU (2) HU229120B1 (h)
IL (7) IL189037A (h)
LU (1) LU91209I2 (h)
MA (1) MA23831A1 (h)
MX (1) MX9707453A (h)
MY (1) MY117896A (h)
NL (1) NL300214I2 (h)
NO (2) NO308740B1 (h)
NZ (1) NZ286263A (h)
OA (1) OA10277A (h)
PE (1) PE43897A1 (h)
PL (1) PL186843B1 (h)
PT (1) PT817775E (h)
RU (2) RU2694252C2 (h)
SA (1) SA96160707B1 (h)
SG (1) SG43262A1 (h)
SI (1) SI9600102A (h)
SK (2) SK283762B6 (h)
TR (1) TR199600265A1 (h)
TW (1) TW454000B (h)
UA (1) UA44254C2 (h)
WO (1) WO1996030347A1 (h)
ZA (1) ZA962522B (h)

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EP3103799A1 (en) 2016-12-14
RU2174977C2 (ru) 2001-10-20
KR100232335B1 (ko) 1999-12-01
EP3103799B1 (en) 2018-06-06
DE69522717D1 (de) 2001-10-18
JP3088018B2 (ja) 2000-09-18
BR9601200A (pt) 1998-01-06

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