CN1423559A - 包含阿片样激动剂和拮抗剂的控释组合物 - Google Patents

包含阿片样激动剂和拮抗剂的控释组合物 Download PDF

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Publication number
CN1423559A
CN1423559A CN01807725A CN01807725A CN1423559A CN 1423559 A CN1423559 A CN 1423559A CN 01807725 A CN01807725 A CN 01807725A CN 01807725 A CN01807725 A CN 01807725A CN 1423559 A CN1423559 A CN 1423559A
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Prior art keywords
opioid
controlled release
opioid agonist
antagonists
agonist
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Pending
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CN01807725A
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English (en)
Chinese (zh)
Inventor
B·奥什拉克
C·赖特
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Euro Celtique SA
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Euro Celtique SA
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22663996&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CN1423559(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Euro Celtique SA filed Critical Euro Celtique SA
Publication of CN1423559A publication Critical patent/CN1423559A/zh
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    • A61K9/5084Mixtures of one or more drugs in different galenical forms, at least one of which being granules, microcapsules or (coated) microparticles according to A61K9/16 or A61K9/50, e.g. for obtaining a specific release pattern or for combining different drugs
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    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
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  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Dermatology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Emergency Medicine (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Otolaryngology (AREA)
  • Pain & Pain Management (AREA)
  • Addiction (AREA)
  • Physics & Mathematics (AREA)
  • Nanotechnology (AREA)
  • Optics & Photonics (AREA)
  • Inorganic Chemistry (AREA)
  • Rheumatology (AREA)
  • Psychiatry (AREA)
  • Toxicology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
CN01807725A 2000-02-08 2001-02-08 包含阿片样激动剂和拮抗剂的控释组合物 Pending CN1423559A (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US18136900P 2000-02-08 2000-02-08
US60/181,369 2000-02-08

Publications (1)

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CN1423559A true CN1423559A (zh) 2003-06-11

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Family Applications (3)

Application Number Title Priority Date Filing Date
CN2009102080743A Expired - Lifetime CN101703777B (zh) 2000-02-08 2001-02-08 抗破坏口服阿片样激动剂
CNB018065694A Expired - Lifetime CN100563656C (zh) 2000-02-08 2001-02-08 抗破坏口服阿片样激动剂
CN01807725A Pending CN1423559A (zh) 2000-02-08 2001-02-08 包含阿片样激动剂和拮抗剂的控释组合物

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Application Number Title Priority Date Filing Date
CN2009102080743A Expired - Lifetime CN101703777B (zh) 2000-02-08 2001-02-08 抗破坏口服阿片样激动剂
CNB018065694A Expired - Lifetime CN100563656C (zh) 2000-02-08 2001-02-08 抗破坏口服阿片样激动剂

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US (15) US6696088B2 (enExample)
EP (6) EP2517710B1 (enExample)
JP (10) JP2003522144A (enExample)
KR (2) KR20020071032A (enExample)
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IL (5) IL151057A0 (enExample)
ME (1) MEP48308A (enExample)
MX (2) MXPA02007686A (enExample)
NO (2) NO20023729L (enExample)
NZ (1) NZ520554A (enExample)
OA (1) OA12215A (enExample)
PL (1) PL210845B1 (enExample)
PT (6) PT2092936E (enExample)
RS (1) RS50407B (enExample)
SI (5) SI1299104T1 (enExample)
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Cited By (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN101622014A (zh) * 2007-03-01 2010-01-06 雷克特本克斯乐保健(英国)有限公司 包含丁丙诺啡和纳曲酮的改善的药用组合物
CN102068697A (zh) * 2010-12-30 2011-05-25 宜昌人福药业有限责任公司 含有阿片类镇痛剂和阿片受体拮抗剂的药用组合物
CN101023947B (zh) * 2006-02-24 2012-10-31 宝血纯化科技股份有限公司 用于杀菌、抑菌和抗炎的组合物及其方法
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CN101330903B (zh) * 2005-12-13 2015-07-08 生物递送科学国际公司 防滥用的经黏膜给药装置
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