TWI292317B - Tamper-resistant oral opioid agonist formulations - Google Patents

Tamper-resistant oral opioid agonist formulations Download PDF

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Publication number
TWI292317B
TWI292317B TW090102735A TW90102735A TWI292317B TW I292317 B TWI292317 B TW I292317B TW 090102735 A TW090102735 A TW 090102735A TW 90102735 A TW90102735 A TW 90102735A TW I292317 B TWI292317 B TW I292317B
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TW
Taiwan
Prior art keywords
formulation
antagonist
interference
opioid
agonist
Prior art date
Application number
TW090102735A
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English (en)
Chinese (zh)
Inventor
Benjamin Oshlack
Curtis Wright
David Haddox J
Original Assignee
Euro Celtique Sa
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Application filed by Euro Celtique Sa filed Critical Euro Celtique Sa
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Publication of TWI292317B publication Critical patent/TWI292317B/zh

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    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5084—Mixtures of one or more drugs in different galenical forms, at least one of which being granules, microcapsules or (coated) microparticles according to A61K9/16 or A61K9/50, e.g. for obtaining a specific release pattern or for combining different drugs
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  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
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TW090102735A 2000-02-08 2001-04-17 Tamper-resistant oral opioid agonist formulations TWI292317B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US18136900P 2000-02-08 2000-02-08

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TWI292317B true TWI292317B (en) 2008-01-11

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TW090102735A TWI292317B (en) 2000-02-08 2001-04-17 Tamper-resistant oral opioid agonist formulations

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US (15) US6696088B2 (enExample)
EP (6) EP2092936B1 (enExample)
JP (10) JP2003522146A (enExample)
KR (2) KR20020071032A (enExample)
CN (3) CN1423559A (enExample)
AP (1) AP1665A (enExample)
AT (1) ATE431145T1 (enExample)
AU (2) AU776904B2 (enExample)
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SI1041987T1 (sl) * 1997-12-22 2006-10-31 Euro Celtique Sa Farmacevtska oralna dozirna oblika, ki obsega kombinacijo opioidnega agonista in naltreksona
AU755790B2 (en) * 1997-12-22 2002-12-19 Euro-Celtique S.A. A method of preventing abuse of opioid dosage forms
US6375957B1 (en) 1997-12-22 2002-04-23 Euro-Celtique, S.A. Opioid agonist/opioid antagonist/acetaminophen combinations
US10179130B2 (en) 1999-10-29 2019-01-15 Purdue Pharma L.P. Controlled release hydrocodone formulations
ES2374717T3 (es) 1999-10-29 2012-02-21 Euro-Celtique S.A. Formulaciones de hidrocodona de liberación controlada.
ATE431145T1 (de) 2000-02-08 2009-05-15 Euro Celtique Sa Missbrauchssichere orale opioid-agonist zubereitungen
AU2002227383B2 (en) 2000-10-30 2004-07-08 Euro-Celtique S.A. Controlled release hydrocodone formulations
US7858118B2 (en) * 2001-04-11 2010-12-28 Galephar Pharmaceutical Research, Inc. Extended release composition containing Tramadol
CA2446738C (en) * 2001-05-11 2012-05-29 Endo Pharmaceuticals, Inc. Abuse-resistant opioid dosage form
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