OA10277A - Quinazoline derivatives - Google Patents

Quinazoline derivatives Download PDF

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Publication number
OA10277A
OA10277A OA60807A OA60807A OA10277A OA 10277 A OA10277 A OA 10277A OA 60807 A OA60807 A OA 60807A OA 60807 A OA60807 A OA 60807A OA 10277 A OA10277 A OA 10277A
Authority
OA
OAPI
Prior art keywords
amine
quinazolin
phenyl
ethynyl
alkyl
Prior art date
Application number
OA60807A
Other languages
English (en)
Inventor
Rodney Caughren Schnur
Lee Daniel Arnold
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=23636708&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=OA10277(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer filed Critical Pfizer
Publication of OA10277A publication Critical patent/OA10277A/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/86Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/94Nitrogen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/08Drugs for disorders of the urinary system of the prostate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/06Antipsoriatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Dermatology (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
OA60807A 1995-03-30 1996-03-29 Quinazoline derivatives OA10277A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US41330095A 1995-03-30 1995-03-30

Publications (1)

Publication Number Publication Date
OA10277A true OA10277A (en) 1997-10-07

Family

ID=23636708

Family Applications (1)

Application Number Title Priority Date Filing Date
OA60807A OA10277A (en) 1995-03-30 1996-03-29 Quinazoline derivatives

Country Status (44)

Country Link
EP (5) EP3103799B1 (uk)
JP (1) JP3088018B2 (uk)
KR (1) KR100232335B1 (uk)
CN (1) CN1066142C (uk)
AP (1) AP735A (uk)
AR (1) AR002723A1 (uk)
AT (2) ATE446955T1 (uk)
AU (2) AU703638B2 (uk)
BR (1) BR9601200B1 (uk)
CA (1) CA2216796C (uk)
CO (1) CO4410333A1 (uk)
CZ (2) CZ294967B6 (uk)
DE (3) DE122005000053I2 (uk)
DK (1) DK0817775T3 (uk)
EG (1) EG24229A (uk)
ES (2) ES2332984T3 (uk)
FI (1) FI120646B (uk)
FR (1) FR06C0010I2 (uk)
GR (1) GR3037070T3 (uk)
HK (1) HK1038740A1 (uk)
HR (1) HRP960147B1 (uk)
HU (2) HU229120B1 (uk)
IL (7) IL129994A (uk)
LU (1) LU91209I2 (uk)
MA (1) MA23831A1 (uk)
MX (1) MX9707453A (uk)
MY (1) MY117896A (uk)
NL (1) NL300214I2 (uk)
NO (2) NO308740B1 (uk)
NZ (1) NZ286263A (uk)
OA (1) OA10277A (uk)
PE (1) PE43897A1 (uk)
PL (1) PL186843B1 (uk)
PT (1) PT817775E (uk)
RU (2) RU2694252C2 (uk)
SA (1) SA96160707B1 (uk)
SG (1) SG43262A1 (uk)
SI (1) SI9600102A (uk)
SK (2) SK283763B6 (uk)
TR (1) TR199600265A1 (uk)
TW (1) TW454000B (uk)
UA (1) UA44254C2 (uk)
WO (1) WO1996030347A1 (uk)
ZA (1) ZA962522B (uk)

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