NO315162B1 - Forbindelser for anvendelse som lysosomale, enzymspaltbare antitumorlegemiddelkonjugater og fremgangsmåte for fremstilling derav - Google Patents
Forbindelser for anvendelse som lysosomale, enzymspaltbare antitumorlegemiddelkonjugater og fremgangsmåte for fremstilling derav Download PDFInfo
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- NO315162B1 NO315162B1 NO19941819A NO941819A NO315162B1 NO 315162 B1 NO315162 B1 NO 315162B1 NO 19941819 A NO19941819 A NO 19941819A NO 941819 A NO941819 A NO 941819A NO 315162 B1 NO315162 B1 NO 315162B1
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- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06008—Dipeptides with the first amino acid being neutral
- C07K5/06078—Dipeptides with the first amino acid being neutral and aromatic or cycloaliphatic
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
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- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Molecular Biology (AREA)
- Biochemistry (AREA)
- Genetics & Genomics (AREA)
- Biophysics (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Immunology (AREA)
- Epidemiology (AREA)
- Crystallography & Structural Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicinal Preparation (AREA)
- Peptides Or Proteins (AREA)
- Enzymes And Modification Thereof (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
- Polysaccharides And Polysaccharide Derivatives (AREA)
- Immobilizing And Processing Of Enzymes And Microorganisms (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US08/062,366 US6214345B1 (en) | 1993-05-14 | 1993-05-14 | Lysosomal enzyme-cleavable antitumor drug conjugates |
Publications (3)
Publication Number | Publication Date |
---|---|
NO941819D0 NO941819D0 (no) | 1994-05-13 |
NO941819L NO941819L (no) | 1994-11-15 |
NO315162B1 true NO315162B1 (no) | 2003-07-21 |
Family
ID=22042014
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO19941819A NO315162B1 (no) | 1993-05-14 | 1994-05-13 | Forbindelser for anvendelse som lysosomale, enzymspaltbare antitumorlegemiddelkonjugater og fremgangsmåte for fremstilling derav |
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- 1994-05-13 PT PT94107501T patent/PT624377E/pt unknown
- 1994-05-13 DE DE69429689T patent/DE69429689T2/de not_active Expired - Lifetime
- 1994-05-13 ES ES94107501T patent/ES2170755T3/es not_active Expired - Lifetime
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NZ260512A (en) | 1996-09-25 |
CN1100426A (zh) | 1995-03-22 |
HU9401507D0 (en) | 1994-09-28 |
PT624377E (pt) | 2002-07-31 |
DK0624377T3 (da) | 2002-05-06 |
RU94016384A (ru) | 1996-11-10 |
NO941819L (no) | 1994-11-15 |
EP0624377B1 (en) | 2002-01-23 |
CN1117760C (zh) | 2003-08-13 |
NO941819D0 (no) | 1994-05-13 |
US6214345B1 (en) | 2001-04-10 |
AU6302694A (en) | 1994-11-17 |
ATE212236T1 (de) | 2002-02-15 |
HUT66485A (en) | 1994-11-28 |
CA2123363A1 (en) | 1994-11-15 |
JPH0770175A (ja) | 1995-03-14 |
FI942237A0 (fi) | 1994-05-13 |
ES2170755T3 (es) | 2002-08-16 |
DE69429689T2 (de) | 2002-10-17 |
AU687795B2 (en) | 1998-03-05 |
CZ118794A3 (en) | 1994-11-16 |
EP0624377A3 (en) | 1995-11-15 |
FI942237A (fi) | 1994-11-15 |
CA2123363C (en) | 2005-04-12 |
FI116038B (fi) | 2005-09-15 |
HU224351B1 (hu) | 2005-08-29 |
DE69429689D1 (de) | 2002-03-14 |
JP3645283B2 (ja) | 2005-05-11 |
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