IL129995A - Alkoxy-substituted 4-hydroxyquinazolines - Google Patents

Alkoxy-substituted 4-hydroxyquinazolines

Info

Publication number
IL129995A
IL129995A IL12999596A IL12999596A IL129995A IL 129995 A IL129995 A IL 129995A IL 12999596 A IL12999596 A IL 12999596A IL 12999596 A IL12999596 A IL 12999596A IL 129995 A IL129995 A IL 129995A
Authority
IL
Israel
Prior art keywords
hydroxyquinazolines
alkoxy
substituted
Prior art date
Application number
IL12999596A
Other languages
English (en)
Original Assignee
Pfizer Prod Inc
Osi Pharm Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=23636708&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IL129995(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer Prod Inc, Osi Pharm Inc filed Critical Pfizer Prod Inc
Publication of IL129995A publication Critical patent/IL129995A/xx

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/94—Nitrogen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/08—Drugs for disorders of the urinary system of the prostate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Dermatology (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
IL12999596A 1995-03-30 1996-03-21 Alkoxy-substituted 4-hydroxyquinazolines IL129995A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US41330095A 1995-03-30 1995-03-30
PCT/IB1995/000436 WO1996030347A1 (en) 1995-03-30 1995-06-06 Quinazoline derivatives
IL11759896A IL117598A (en) 1995-03-30 1996-03-21 Quinazoline derivatives, process for their preparation and pharmaceutical compositions containing them

Publications (1)

Publication Number Publication Date
IL129995A true IL129995A (en) 2005-11-20

Family

ID=23636708

Family Applications (7)

Application Number Title Priority Date Filing Date
IL129994A IL129994A (en) 1995-03-30 1996-03-21 4 - Chloroquinozolines are converted to alkoxy
IL11759896A IL117598A (en) 1995-03-30 1996-03-21 Quinazoline derivatives, process for their preparation and pharmaceutical compositions containing them
IL12999596A IL129995A (en) 1995-03-30 1996-03-21 Alkoxy-substituted 4-hydroxyquinazolines
IL189037A IL189037A (en) 1995-03-30 1996-03-21 4-Chloroquinazolines are converted to alkoxy
IL12999599A IL129995A0 (en) 1995-03-30 1999-05-17 Quinazoline derivatives
IL12999699A IL129996A0 (en) 1995-03-30 1999-05-17 Quinazoline derivative intermediates
IL12999499A IL129994A0 (en) 1995-03-30 1999-05-17 Quinazoline derivatives

Family Applications Before (2)

Application Number Title Priority Date Filing Date
IL129994A IL129994A (en) 1995-03-30 1996-03-21 4 - Chloroquinozolines are converted to alkoxy
IL11759896A IL117598A (en) 1995-03-30 1996-03-21 Quinazoline derivatives, process for their preparation and pharmaceutical compositions containing them

Family Applications After (4)

Application Number Title Priority Date Filing Date
IL189037A IL189037A (en) 1995-03-30 1996-03-21 4-Chloroquinazolines are converted to alkoxy
IL12999599A IL129995A0 (en) 1995-03-30 1999-05-17 Quinazoline derivatives
IL12999699A IL129996A0 (en) 1995-03-30 1999-05-17 Quinazoline derivative intermediates
IL12999499A IL129994A0 (en) 1995-03-30 1999-05-17 Quinazoline derivatives

Country Status (44)

Country Link
EP (5) EP3103799B1 (uk)
JP (1) JP3088018B2 (uk)
KR (1) KR100232335B1 (uk)
CN (1) CN1066142C (uk)
AP (1) AP735A (uk)
AR (1) AR002723A1 (uk)
AT (2) ATE446955T1 (uk)
AU (2) AU703638B2 (uk)
BR (1) BR9601200B1 (uk)
CA (1) CA2216796C (uk)
CO (1) CO4410333A1 (uk)
CZ (2) CZ294967B6 (uk)
DE (3) DE122005000053I2 (uk)
DK (1) DK0817775T3 (uk)
EG (1) EG24229A (uk)
ES (2) ES2332984T3 (uk)
FI (1) FI120646B (uk)
FR (1) FR06C0010I2 (uk)
GR (1) GR3037070T3 (uk)
HK (1) HK1038740A1 (uk)
HR (1) HRP960147B1 (uk)
HU (2) HU229120B1 (uk)
IL (7) IL129994A (uk)
LU (1) LU91209I2 (uk)
MA (1) MA23831A1 (uk)
MX (1) MX9707453A (uk)
MY (1) MY117896A (uk)
NL (1) NL300214I2 (uk)
NO (2) NO308740B1 (uk)
NZ (1) NZ286263A (uk)
OA (1) OA10277A (uk)
PE (1) PE43897A1 (uk)
PL (1) PL186843B1 (uk)
PT (1) PT817775E (uk)
RU (2) RU2694252C2 (uk)
SA (1) SA96160707B1 (uk)
SG (1) SG43262A1 (uk)
SI (1) SI9600102A (uk)
SK (2) SK283763B6 (uk)
TR (1) TR199600265A1 (uk)
TW (1) TW454000B (uk)
UA (1) UA44254C2 (uk)
WO (1) WO1996030347A1 (uk)
ZA (1) ZA962522B (uk)

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