EA029890B1 - Фармацевтическая композиция и фармацевтическая композиция в пероральной дозированной лекарственной форме на основе ингибитора dpp iv - Google Patents

Фармацевтическая композиция и фармацевтическая композиция в пероральной дозированной лекарственной форме на основе ингибитора dpp iv Download PDF

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Publication number
EA029890B1
EA029890B1 EA201100958A EA201100958A EA029890B1 EA 029890 B1 EA029890 B1 EA 029890B1 EA 201100958 A EA201100958 A EA 201100958A EA 201100958 A EA201100958 A EA 201100958A EA 029890 B1 EA029890 B1 EA 029890B1
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EA
Eurasian Patent Office
Prior art keywords
pharmaceutical composition
diluent
methyl
amount
composition according
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EA201100958A
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English (en)
Russian (ru)
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EA201100958A1 (ru
Inventor
Аня Кольрауш
Патрик Ромер
Герд Зайфферт
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Бёрингер Ингельхайм Интернациональ Гмбх
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Application filed by Бёрингер Ингельхайм Интернациональ Гмбх filed Critical Бёрингер Ингельхайм Интернациональ Гмбх
Publication of EA201100958A1 publication Critical patent/EA201100958A1/ru
Publication of EA029890B1 publication Critical patent/EA029890B1/ru

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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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  • Diabetes (AREA)
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  • Obesity (AREA)
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  • Pain & Pain Management (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
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EA201100958A 2006-05-04 2007-04-30 Фармацевтическая композиция и фармацевтическая композиция в пероральной дозированной лекарственной форме на основе ингибитора dpp iv EA029890B1 (ru)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP06009201A EP1852108A1 (en) 2006-05-04 2006-05-04 DPP IV inhibitor formulations

Publications (2)

Publication Number Publication Date
EA201100958A1 EA201100958A1 (ru) 2012-04-30
EA029890B1 true EA029890B1 (ru) 2018-05-31

Family

ID=36972901

Family Applications (2)

Application Number Title Priority Date Filing Date
EA201100958A EA029890B1 (ru) 2006-05-04 2007-04-30 Фармацевтическая композиция и фармацевтическая композиция в пероральной дозированной лекарственной форме на основе ингибитора dpp iv
EA200802184A EA016559B1 (ru) 2006-05-04 2007-04-30 Фармацевтические композиции с ингибиторами dpp iv

Family Applications After (1)

Application Number Title Priority Date Filing Date
EA200802184A EA016559B1 (ru) 2006-05-04 2007-04-30 Фармацевтические композиции с ингибиторами dpp iv

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Country Link
US (9) US20080107731A1 (enExample)
EP (5) EP1852108A1 (enExample)
JP (8) JP5478244B2 (enExample)
KR (5) KR101855323B1 (enExample)
CN (2) CN101437493B (enExample)
AR (2) AR060755A1 (enExample)
AT (1) ATE480228T1 (enExample)
AU (1) AU2007247193B2 (enExample)
BR (2) BRPI0722388B1 (enExample)
CA (1) CA2649922C (enExample)
CL (2) CL2012002522A1 (enExample)
CY (2) CY1111354T1 (enExample)
DE (1) DE602007009091D1 (enExample)
DK (3) DK2283819T3 (enExample)
EA (2) EA029890B1 (enExample)
EC (1) ECSP088800A (enExample)
ES (3) ES2348576T3 (enExample)
HR (2) HRP20100507T1 (enExample)
HU (1) HUE025210T2 (enExample)
IL (2) IL195030A (enExample)
ME (2) ME01941B (enExample)
MX (3) MX2008013958A (enExample)
MY (2) MY146969A (enExample)
NO (1) NO343067B1 (enExample)
NZ (3) NZ595983A (enExample)
PE (2) PE20110666A1 (enExample)
PL (3) PL2283819T3 (enExample)
PT (2) PT2023902E (enExample)
RS (2) RS53570B1 (enExample)
SG (1) SG171649A1 (enExample)
SI (2) SI2023902T1 (enExample)
TW (2) TWI474843B (enExample)
UA (1) UA94942C2 (enExample)
UY (1) UY30319A1 (enExample)
WO (1) WO2007128724A1 (enExample)
ZA (1) ZA200808361B (enExample)

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JP2530113B2 (ja) 1994-06-29 1996-09-04 インターナショナル・ビジネス・マシーンズ・コーポレイション デ―タ転送制御用インタ―フェ―ス回路及び磁気ディスク装置
US7407955B2 (en) 2002-08-21 2008-08-05 Boehringer Ingelheim Pharma Gmbh & Co., Kg 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions
US7495005B2 (en) * 2002-08-22 2009-02-24 Boehringer Ingelheim Pharma Gmbh & Co. Kg Xanthine derivatives, their preparation and their use in pharmaceutical compositions
US7482337B2 (en) * 2002-11-08 2009-01-27 Boehringer Ingelheim Pharma Gmbh & Co. Kg Xanthine derivatives, the preparation thereof and their use as pharmaceutical compositions
US7501426B2 (en) 2004-02-18 2009-03-10 Boehringer Ingelheim International Gmbh 8-[3-amino-piperidin-1-yl]-xanthines, their preparation and their use as pharmaceutical compositions
US7439370B2 (en) 2004-05-10 2008-10-21 Boehringer Ingelheim International Gmbh Imidazole derivatives, their preparation and their use as intermediates for the preparation of pharmaceutical compositions and pesticides
DE102004030502A1 (de) 2004-06-24 2006-01-12 Boehringer Ingelheim Pharma Gmbh & Co. Kg Neue Imidazole und Triazole, deren Herstellung und Verwendung als Arzneimittel
DE102004054054A1 (de) 2004-11-05 2006-05-11 Boehringer Ingelheim Pharma Gmbh & Co. Kg Verfahren zur Herstellung chiraler 8-(3-Amino-piperidin-1-yl)-xanthine
US7772191B2 (en) 2005-05-10 2010-08-10 Boehringer Ingelheim International Gmbh Processes for preparing of glucopyranosyl-substituted benzyl-benzene derivatives and intermediates therein
DE102005035891A1 (de) 2005-07-30 2007-02-08 Boehringer Ingelheim Pharma Gmbh & Co. Kg 8-(3-Amino-piperidin-1-yl)-xanthine, deren Herstellung und deren Verwendung als Arzneimittel
EP2540725A1 (de) 2006-05-04 2013-01-02 Boehringer Ingelheim International GmbH Polymorphe von 1-((4-Methyl-chinazolin-2-yl)methyl)-3-methyl-7-(2-butin-1-yl)-8-(3-(R)-amino-piperidin-1-yl)xanthin
EP1852108A1 (en) 2006-05-04 2007-11-07 Boehringer Ingelheim Pharma GmbH & Co.KG DPP IV inhibitor formulations
PE20080251A1 (es) 2006-05-04 2008-04-25 Boehringer Ingelheim Int Usos de inhibidores de dpp iv
WO2007143705A2 (en) 2006-06-06 2007-12-13 Intra-Cellular Therapies, Inc. Organic compounds
EP2057160A1 (en) 2006-08-08 2009-05-13 Boehringer Ingelheim International GmbH Pyrrolo [3, 2 -d]pyrimidines as dpp-iv inhibitors for the treatment of diabetes mellitus
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