JP5478244B2 - Ｄｐｐ ｉｖインヒビター製剤 - Google Patents

Ｄｐｐ ｉｖインヒビター製剤 Download PDF

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JP5478244B2
JP5478244B2 JP2009508327A JP2009508327A JP5478244B2 JP 5478244 B2 JP5478244 B2 JP 5478244B2 JP 2009508327 A JP2009508327 A JP 2009508327A JP 2009508327 A JP2009508327 A JP 2009508327A JP 5478244 B2 JP5478244 B2 JP 5478244B2
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methyl
pharmaceutical composition
amino
xanthine
tablet
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JP2009535376A6 (ja
JP2009535376A (ja
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アーニャ コールラウシュ
パトリック ローマー
ゲルト ザイフェルト
Original Assignee
ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52—Purines, e.g. adenine
    • A61K31/522—Purines, e.g. adenine having oxo groups directly attached to the heterocyclic ring, e.g. hypoxanthine, guanine, acyclovir
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/34—Macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyesters, polyamino acids, polysiloxanes, polyphosphazines, copolymers of polyalkylene glycol or poloxamers
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    • A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Inorganic Chemistry (AREA)
  • Diabetes (AREA)
  • Immunology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Transplantation (AREA)
  • Child & Adolescent Psychology (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
JP2009508327A 2006-05-04 2007-04-30 Ｄｐｐ ｉｖインヒビター製剤 Active JP5478244B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP06009201.2 2006-05-04
EP06009201A EP1852108A1 (en) 2006-05-04 2006-05-04 DPP IV inhibitor formulations
PCT/EP2007/054204 WO2007128724A1 (en) 2006-05-04 2007-04-30 Dpp iv inhibitor formulations

Related Child Applications (2)

Application Number Title Priority Date Filing Date
JP2012000293A Division JP6100998B2 (ja) 2006-05-04 2012-01-04 Ｄｐｐｉｖインヒビター製剤
JP2013145188A Division JP2013227338A (ja) 2006-05-04 2013-07-11 Ｄｐｐｉｖインヒビター製剤

Publications (3)

Publication Number Publication Date
JP2009535376A JP2009535376A (ja) 2009-10-01
JP2009535376A6 JP2009535376A6 (ja) 2010-11-18
JP5478244B2 true JP5478244B2 (ja) 2014-04-23

Family

ID=36972901

Family Applications (8)

Application Number Title Priority Date Filing Date
JP2009508327A Active JP5478244B2 (ja) 2006-05-04 2007-04-30 Ｄｐｐ ｉｖインヒビター製剤
JP2012000293A Active JP6100998B2 (ja) 2006-05-04 2012-01-04 Ｄｐｐｉｖインヒビター製剤
JP2013145188A Pending JP2013227338A (ja) 2006-05-04 2013-07-11 Ｄｐｐｉｖインヒビター製剤
JP2016033423A Active JP6564720B2 (ja) 2006-05-04 2016-02-24 Ｄｐｐｉｖインヒビター製剤
JP2017217311A Active JP7084711B2 (ja) 2006-05-04 2017-11-10 Ｄｐｐ ｉｖインヒビター製剤
JP2020033173A Active JP6987908B2 (ja) 2006-05-04 2020-02-28 Ｄｐｐ ｉｖインヒビター製剤
JP2022040337A Pending JP2022075826A (ja) 2006-05-04 2022-03-15 Ｄｐｐ ｉｖインヒビター製剤
JP2024029844A Pending JP2024074800A (ja) 2006-05-04 2024-02-29 Ｄｐｐ ｉｖインヒビター製剤

Family Applications After (7)

Application Number Title Priority Date Filing Date
JP2012000293A Active JP6100998B2 (ja) 2006-05-04 2012-01-04 Ｄｐｐｉｖインヒビター製剤
JP2013145188A Pending JP2013227338A (ja) 2006-05-04 2013-07-11 Ｄｐｐｉｖインヒビター製剤
JP2016033423A Active JP6564720B2 (ja) 2006-05-04 2016-02-24 Ｄｐｐｉｖインヒビター製剤
JP2017217311A Active JP7084711B2 (ja) 2006-05-04 2017-11-10 Ｄｐｐ ｉｖインヒビター製剤
JP2020033173A Active JP6987908B2 (ja) 2006-05-04 2020-02-28 Ｄｐｐ ｉｖインヒビター製剤
JP2022040337A Pending JP2022075826A (ja) 2006-05-04 2022-03-15 Ｄｐｐ ｉｖインヒビター製剤
JP2024029844A Pending JP2024074800A (ja) 2006-05-04 2024-02-29 Ｄｐｐ ｉｖインヒビター製剤

Country Status (36)

Country Link
US (9) US20080107731A1 (enExample)
EP (5) EP1852108A1 (enExample)
JP (8) JP5478244B2 (enExample)
KR (5) KR101710881B1 (enExample)
CN (2) CN102526737B (enExample)
AR (2) AR060755A1 (enExample)
AT (1) ATE480228T1 (enExample)
AU (1) AU2007247193B2 (enExample)
BR (2) BRPI0722388B1 (enExample)
CA (1) CA2649922C (enExample)
CL (2) CL2012002521A1 (enExample)
CY (2) CY1111354T1 (enExample)
DE (1) DE602007009091D1 (enExample)
DK (3) DK2277509T5 (enExample)
EA (2) EA016559B1 (enExample)
EC (1) ECSP088800A (enExample)
ES (3) ES2527409T4 (enExample)
HR (2) HRP20100507T1 (enExample)
HU (1) HUE025210T2 (enExample)
IL (2) IL195030A (enExample)
ME (2) ME01941B (enExample)
MX (3) MX2008013958A (enExample)
MY (2) MY146969A (enExample)
NO (1) NO343067B1 (enExample)
NZ (3) NZ572862A (enExample)
PE (2) PE20110666A1 (enExample)
PL (3) PL2277509T3 (enExample)
PT (2) PT2023902E (enExample)
RS (2) RS53570B1 (enExample)
SG (1) SG171649A1 (enExample)
SI (2) SI2023902T1 (enExample)
TW (2) TWI520753B (enExample)
UA (1) UA94942C2 (enExample)
UY (1) UY30319A1 (enExample)
WO (1) WO2007128724A1 (enExample)
ZA (1) ZA200808361B (enExample)

Families Citing this family (120)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2530113B2 (ja) 1994-06-29 1996-09-04 インターナショナル・ビジネス・マシーンズ・コーポレイション デ―タ転送制御用インタ―フェ―ス回路及び磁気ディスク装置
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