CL2008003653A1 - Uso de un inhibidor de sglt derivado de glucopiranosilo y un inhibidor de dppiv seleccionado para tratar la diabetes; y composicion farmaceutica. - Google Patents
Uso de un inhibidor de sglt derivado de glucopiranosilo y un inhibidor de dppiv seleccionado para tratar la diabetes; y composicion farmaceutica.Info
- Publication number
- CL2008003653A1 CL2008003653A1 CL2008003653A CL2008003653A CL2008003653A1 CL 2008003653 A1 CL2008003653 A1 CL 2008003653A1 CL 2008003653 A CL2008003653 A CL 2008003653A CL 2008003653 A CL2008003653 A CL 2008003653A CL 2008003653 A1 CL2008003653 A1 CL 2008003653A1
- Authority
- CL
- Chile
- Prior art keywords
- inhibitor
- glucopyranosyl
- derived
- pharmaceutical composition
- treat diabetes
- Prior art date
Links
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
- A61K31/706—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/401—Proline; Derivatives thereof, e.g. captopril
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
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- A—HUMAN NECESSITIES
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- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/4985—Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
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- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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- A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H7/00—Compounds containing non-saccharide radicals linked to saccharide radicals by a carbon-to-carbon bond
- C07H7/04—Carbocyclic radicals
Abstract
Un método para tratar o prevenir la diabetes o una afección relacionada con diabetes, que comprende el uso de un inhibidor de sglt y un inhibidor dpp4.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US2177708P | 2008-01-17 | 2008-01-17 |
Publications (1)
Publication Number | Publication Date |
---|---|
CL2008003653A1 true CL2008003653A1 (es) | 2010-03-05 |
Family
ID=40433628
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CL2008003653A CL2008003653A1 (es) | 2008-01-17 | 2008-12-09 | Uso de un inhibidor de sglt derivado de glucopiranosilo y un inhibidor de dppiv seleccionado para tratar la diabetes; y composicion farmaceutica. |
Country Status (14)
Country | Link |
---|---|
US (2) | US8853385B2 (es) |
EP (1) | EP2252289B1 (es) |
JP (3) | JP5204849B2 (es) |
KR (1) | KR101257554B1 (es) |
CN (2) | CN103599539A (es) |
AR (1) | AR070193A1 (es) |
AU (1) | AU2009205060C1 (es) |
BR (1) | BRPI0906735A2 (es) |
CA (1) | CA2712614C (es) |
CL (1) | CL2008003653A1 (es) |
ES (1) | ES2763239T3 (es) |
MX (1) | MX2010007818A (es) |
TW (1) | TWI437996B (es) |
WO (1) | WO2009091082A1 (es) |
Families Citing this family (62)
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US7407955B2 (en) | 2002-08-21 | 2008-08-05 | Boehringer Ingelheim Pharma Gmbh & Co., Kg | 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions |
US7772191B2 (en) | 2005-05-10 | 2010-08-10 | Boehringer Ingelheim International Gmbh | Processes for preparing of glucopyranosyl-substituted benzyl-benzene derivatives and intermediates therein |
PE20080697A1 (es) | 2006-05-03 | 2008-08-05 | Boehringer Ingelheim Int | Derivados de benzonitrilo sustituidos con glucopiranosilo, composiciones farmaceuticas que contienen compuestos de este tipo, su uso y procedimiento para su fabricacion |
PE20110235A1 (es) | 2006-05-04 | 2011-04-14 | Boehringer Ingelheim Int | Combinaciones farmaceuticas que comprenden linagliptina y metmorfina |
EP1852108A1 (en) | 2006-05-04 | 2007-11-07 | Boehringer Ingelheim Pharma GmbH & Co.KG | DPP IV inhibitor formulations |
EA015687B1 (ru) | 2006-05-04 | 2011-10-31 | Бёрингер Ингельхайм Интернациональ Гмбх | Полиморфы |
PE20090938A1 (es) | 2007-08-16 | 2009-08-08 | Boehringer Ingelheim Int | Composicion farmaceutica que comprende un derivado de benceno sustituido con glucopiranosilo |
ME03072B (me) | 2007-09-10 | 2019-01-20 | Janssen Pharmaceutica Nv | Postupak za dobijanje jedinjenja која su korisna као inhibiтori sgl т |
CL2008003653A1 (es) * | 2008-01-17 | 2010-03-05 | Mitsubishi Tanabe Pharma Corp | Uso de un inhibidor de sglt derivado de glucopiranosilo y un inhibidor de dppiv seleccionado para tratar la diabetes; y composicion farmaceutica. |
JP2009196984A (ja) * | 2008-01-25 | 2009-09-03 | Mitsubishi Tanabe Pharma Corp | 医薬組成物 |
PE20091730A1 (es) | 2008-04-03 | 2009-12-10 | Boehringer Ingelheim Int | Formulaciones que comprenden un inhibidor de dpp4 |
KR20200118243A (ko) | 2008-08-06 | 2020-10-14 | 베링거 인겔하임 인터내셔날 게엠베하 | 메트포르민 요법이 부적합한 환자에서의 당뇨병 치료 |
EA018492B1 (ru) | 2008-08-28 | 2013-08-30 | Пфайзер Инк. | Диоксабицикло[3.2.1]октан-2,3,4-триольные производные |
US20200155558A1 (en) | 2018-11-20 | 2020-05-21 | Boehringer Ingelheim International Gmbh | Treatment for diabetes in patients with insufficient glycemic control despite therapy with an oral antidiabetic drug |
US9056850B2 (en) | 2008-10-17 | 2015-06-16 | Janssen Pharmaceutica N.V. | Process for the preparation of compounds useful as inhibitors of SGLT |
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WO2011039108A2 (en) | 2009-09-30 | 2011-04-07 | Boehringer Ingelheim International Gmbh | Processes for preparing of glucopyranosyl-substituted benzyl-benzene derivatives |
US10610489B2 (en) | 2009-10-02 | 2020-04-07 | Boehringer Ingelheim International Gmbh | Pharmaceutical composition, pharmaceutical dosage form, process for their preparation, methods for treating and uses thereof |
JP5833011B2 (ja) | 2009-10-14 | 2015-12-16 | ヤンセン ファーマシューティカ エヌ.ベー. | Sglt2の阻害物質として有用な化合物の調製プロセス |
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CN107115530A (zh) | 2009-11-27 | 2017-09-01 | 勃林格殷格翰国际有限公司 | 基因型糖尿病患者利用dpp‑iv抑制剂例如利拉利汀的治疗 |
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WO2011107494A1 (de) | 2010-03-03 | 2011-09-09 | Sanofi | Neue aromatische glykosidderivate, diese verbindungen enthaltende arzneimittel und deren verwendung |
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-
2008
- 2008-12-09 CL CL2008003653A patent/CL2008003653A1/es unknown
-
2009
- 2009-01-16 ES ES09701670T patent/ES2763239T3/es active Active
- 2009-01-16 CN CN201310475934.6A patent/CN103599539A/zh active Pending
- 2009-01-16 US US12/863,429 patent/US8853385B2/en not_active Expired - Fee Related
- 2009-01-16 CA CA2712614A patent/CA2712614C/en not_active Expired - Fee Related
- 2009-01-16 MX MX2010007818A patent/MX2010007818A/es active IP Right Grant
- 2009-01-16 CN CN200980102300.8A patent/CN101932321B/zh active Active
- 2009-01-16 EP EP09701670.3A patent/EP2252289B1/en active Active
- 2009-01-16 WO PCT/JP2009/051023 patent/WO2009091082A1/en active Application Filing
- 2009-01-16 JP JP2010528230A patent/JP5204849B2/ja active Active
- 2009-01-16 AU AU2009205060A patent/AU2009205060C1/en not_active Ceased
- 2009-01-16 AR ARP090100146A patent/AR070193A1/es not_active Application Discontinuation
- 2009-01-16 BR BRPI0906735-3A patent/BRPI0906735A2/pt not_active Application Discontinuation
- 2009-01-16 KR KR1020107018132A patent/KR101257554B1/ko active IP Right Grant
- 2009-01-17 TW TW098101763A patent/TWI437996B/zh not_active IP Right Cessation
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2012
- 2012-12-27 JP JP2012284625A patent/JP5646588B2/ja active Active
-
2014
- 2014-08-28 US US14/472,037 patent/US20140371162A1/en not_active Abandoned
- 2014-11-05 JP JP2014225301A patent/JP5908563B2/ja active Active
Also Published As
Publication number | Publication date |
---|---|
MX2010007818A (es) | 2010-08-09 |
AU2009205060B2 (en) | 2013-06-27 |
KR20100103874A (ko) | 2010-09-28 |
TWI437996B (zh) | 2014-05-21 |
JP2013091654A (ja) | 2013-05-16 |
US8853385B2 (en) | 2014-10-07 |
AU2009205060C1 (en) | 2013-12-19 |
BRPI0906735A2 (pt) | 2015-07-07 |
EP2252289B1 (en) | 2019-10-23 |
JP2015044845A (ja) | 2015-03-12 |
CA2712614A1 (en) | 2009-07-23 |
CA2712614C (en) | 2014-05-27 |
ES2763239T3 (es) | 2020-05-27 |
CN101932321A (zh) | 2010-12-29 |
AR070193A1 (es) | 2010-03-17 |
US20140371162A1 (en) | 2014-12-18 |
CN101932321B (zh) | 2016-05-18 |
JP5204849B2 (ja) | 2013-06-05 |
JP5908563B2 (ja) | 2016-04-26 |
TW200932249A (en) | 2009-08-01 |
RU2010134362A (ru) | 2012-02-27 |
EP2252289A1 (en) | 2010-11-24 |
WO2009091082A1 (en) | 2009-07-23 |
KR101257554B1 (ko) | 2013-04-23 |
CN103599539A (zh) | 2014-02-26 |
AU2009205060A1 (en) | 2009-07-23 |
JP5646588B2 (ja) | 2014-12-24 |
US20110059912A1 (en) | 2011-03-10 |
JP2011509922A (ja) | 2011-03-31 |
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