MX2010009731A - Composiciones farmaceuticas de una combinacion de metformina y un inhibidor de dipeptidil peptidasa-iv. - Google Patents

Composiciones farmaceuticas de una combinacion de metformina y un inhibidor de dipeptidil peptidasa-iv.

Info

Publication number
MX2010009731A
MX2010009731A MX2010009731A MX2010009731A MX2010009731A MX 2010009731 A MX2010009731 A MX 2010009731A MX 2010009731 A MX2010009731 A MX 2010009731A MX 2010009731 A MX2010009731 A MX 2010009731A MX 2010009731 A MX2010009731 A MX 2010009731A
Authority
MX
Mexico
Prior art keywords
metformin
pharmaceutical compositions
inhibitor
combination
dipeptidyl peptidase
Prior art date
Application number
MX2010009731A
Other languages
English (en)
Inventor
Nazaneen Pourkavoos
Original Assignee
Merck Sharp & Dohme
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Sharp & Dohme filed Critical Merck Sharp & Dohme
Publication of MX2010009731A publication Critical patent/MX2010009731A/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/155—Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
    • A61K9/209—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics

Landscapes

  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Diabetes (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Se describen composiciones farmacéuticas que comprenden combinaciones de dosis fija de una forma de liberación prolongada de metformina, o una sal farmacéuticamente aceptable de la misma, recubierta con una forma de liberación inmediata del inhibidor de DPP-4 sitagliptina o una sal farmacéuticamente aceptable de la misma.
MX2010009731A 2008-03-04 2009-02-23 Composiciones farmaceuticas de una combinacion de metformina y un inhibidor de dipeptidil peptidasa-iv. MX2010009731A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US6801608P 2008-03-04 2008-03-04
PCT/US2009/034851 WO2009111200A1 (en) 2008-03-04 2009-02-23 Pharmaceutical compositions of a combination of metformin and a dipeptidyl peptidase-iv inhibitor

Publications (1)

Publication Number Publication Date
MX2010009731A true MX2010009731A (es) 2010-09-30

Family

ID=41056332

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2010009731A MX2010009731A (es) 2008-03-04 2009-02-23 Composiciones farmaceuticas de una combinacion de metformina y un inhibidor de dipeptidil peptidasa-iv.

Country Status (8)

Country Link
US (1) US20100323011A1 (es)
EP (1) EP2259676A4 (es)
JP (1) JP2011513408A (es)
CN (1) CN101959406A (es)
AU (1) AU2009220444A1 (es)
CA (1) CA2716130A1 (es)
MX (1) MX2010009731A (es)
WO (1) WO2009111200A1 (es)

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Also Published As

Publication number Publication date
CN101959406A (zh) 2011-01-26
US20100323011A1 (en) 2010-12-23
JP2011513408A (ja) 2011-04-28
WO2009111200A1 (en) 2009-09-11
EP2259676A4 (en) 2011-03-16
CA2716130A1 (en) 2009-09-11
EP2259676A1 (en) 2010-12-15
AU2009220444A1 (en) 2009-09-11

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