ME01170B - Formulacije dpp iv inhibitora - Google Patents

Formulacije dpp iv inhibitora

Info

Publication number
ME01170B
ME01170B MEP-2010-172A MEP17210A ME01170B ME 01170 B ME01170 B ME 01170B ME P17210 A MEP17210 A ME P17210A ME 01170 B ME01170 B ME 01170B
Authority
ME
Montenegro
Prior art keywords
methyl
amino
xanthine
piperidin
butyn
Prior art date
Application number
MEP-2010-172A
Other languages
English (en)
French (fr)
Unknown language (me)
Inventor
Anja Kohlrausch
Patrick Romer
Gerd Seiffert
Original Assignee
Boehringer Ingelheim Int
Boehringer Ingelheim Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=36972901&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ME01170(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Boehringer Ingelheim Int, Boehringer Ingelheim Pharma filed Critical Boehringer Ingelheim Int
Publication of ME01170B publication Critical patent/ME01170B/me

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • A61K47/38—Cellulose; Derivatives thereof
    • A—HUMAN NECESSITIES
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52—Purines, e.g. adenine
    • A61K31/522—Purines, e.g. adenine having oxo groups directly attached to the heterocyclic ring, e.g. hypoxanthine, guanine, acyclovir
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    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/34—Macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyesters, polyamino acids, polysiloxanes, polyphosphazines, copolymers of polyalkylene glycol or poloxamers
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    • A61K9/2833—Organic macromolecular compounds
    • A61K9/2853—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers, poly(lactide-co-glycolide)
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    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
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    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Inorganic Chemistry (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Immunology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Rheumatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Transplantation (AREA)
  • Child & Adolescent Psychology (AREA)
  • Endocrinology (AREA)
  • Pain & Pain Management (AREA)
  • Emergency Medicine (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
MEP-2010-172A 2006-05-04 2007-04-30 Formulacije dpp iv inhibitora ME01170B (me)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP06009201A EP1852108A1 (en) 2006-05-04 2006-05-04 DPP IV inhibitor formulations
EP07728658A EP2023902B8 (en) 2006-05-04 2007-04-30 Dpp iv inhibitor formulations
PCT/EP2007/054204 WO2007128724A1 (en) 2006-05-04 2007-04-30 Dpp iv inhibitor formulations

Publications (1)

Publication Number Publication Date
ME01170B true ME01170B (me) 2013-03-20

Family

ID=36972901

Family Applications (2)

Application Number Title Priority Date Filing Date
MEP-2010-172A ME01170B (me) 2006-05-04 2007-04-30 Formulacije dpp iv inhibitora
MEP-2014-136A ME01941B (me) 2006-05-04 2007-04-30 Formulacije DPP IV inhibitora

Family Applications After (1)

Application Number Title Priority Date Filing Date
MEP-2014-136A ME01941B (me) 2006-05-04 2007-04-30 Formulacije DPP IV inhibitora

Country Status (36)

Country Link
US (9) US20080107731A1 (cg-RX-API-DMAC7.html)
EP (5) EP1852108A1 (cg-RX-API-DMAC7.html)
JP (8) JP5478244B2 (cg-RX-API-DMAC7.html)
KR (5) KR101710881B1 (cg-RX-API-DMAC7.html)
CN (2) CN101437493B (cg-RX-API-DMAC7.html)
AR (2) AR060755A1 (cg-RX-API-DMAC7.html)
AT (1) ATE480228T1 (cg-RX-API-DMAC7.html)
AU (1) AU2007247193B2 (cg-RX-API-DMAC7.html)
BR (2) BRPI0711179B1 (cg-RX-API-DMAC7.html)
CA (1) CA2649922C (cg-RX-API-DMAC7.html)
CL (2) CL2012002522A1 (cg-RX-API-DMAC7.html)
CY (2) CY1111354T1 (cg-RX-API-DMAC7.html)
DE (1) DE602007009091D1 (cg-RX-API-DMAC7.html)
DK (3) DK2277509T5 (cg-RX-API-DMAC7.html)
EA (2) EA016559B1 (cg-RX-API-DMAC7.html)
EC (1) ECSP088800A (cg-RX-API-DMAC7.html)
ES (3) ES2348576T3 (cg-RX-API-DMAC7.html)
HR (2) HRP20100507T1 (cg-RX-API-DMAC7.html)
HU (1) HUE025210T2 (cg-RX-API-DMAC7.html)
IL (2) IL195030A (cg-RX-API-DMAC7.html)
ME (2) ME01170B (cg-RX-API-DMAC7.html)
MX (3) MX358617B (cg-RX-API-DMAC7.html)
MY (2) MY146969A (cg-RX-API-DMAC7.html)
NO (1) NO343067B1 (cg-RX-API-DMAC7.html)
NZ (3) NZ595983A (cg-RX-API-DMAC7.html)
PE (2) PE20110666A1 (cg-RX-API-DMAC7.html)
PL (3) PL2283819T3 (cg-RX-API-DMAC7.html)
PT (2) PT2023902E (cg-RX-API-DMAC7.html)
RS (2) RS51466B (cg-RX-API-DMAC7.html)
SG (1) SG171649A1 (cg-RX-API-DMAC7.html)
SI (2) SI2023902T1 (cg-RX-API-DMAC7.html)
TW (2) TWI474843B (cg-RX-API-DMAC7.html)
UA (1) UA94942C2 (cg-RX-API-DMAC7.html)
UY (1) UY30319A1 (cg-RX-API-DMAC7.html)
WO (1) WO2007128724A1 (cg-RX-API-DMAC7.html)
ZA (1) ZA200808361B (cg-RX-API-DMAC7.html)

Families Citing this family (120)

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JP2530113B2 (ja) 1994-06-29 1996-09-04 インターナショナル・ビジネス・マシーンズ・コーポレイション デ―タ転送制御用インタ―フェ―ス回路及び磁気ディスク装置
US7407955B2 (en) 2002-08-21 2008-08-05 Boehringer Ingelheim Pharma Gmbh & Co., Kg 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions
US7495005B2 (en) * 2002-08-22 2009-02-24 Boehringer Ingelheim Pharma Gmbh & Co. Kg Xanthine derivatives, their preparation and their use in pharmaceutical compositions
US7482337B2 (en) * 2002-11-08 2009-01-27 Boehringer Ingelheim Pharma Gmbh & Co. Kg Xanthine derivatives, the preparation thereof and their use as pharmaceutical compositions
US7501426B2 (en) 2004-02-18 2009-03-10 Boehringer Ingelheim International Gmbh 8-[3-amino-piperidin-1-yl]-xanthines, their preparation and their use as pharmaceutical compositions
US7439370B2 (en) 2004-05-10 2008-10-21 Boehringer Ingelheim International Gmbh Imidazole derivatives, their preparation and their use as intermediates for the preparation of pharmaceutical compositions and pesticides
DE102004030502A1 (de) 2004-06-24 2006-01-12 Boehringer Ingelheim Pharma Gmbh & Co. Kg Neue Imidazole und Triazole, deren Herstellung und Verwendung als Arzneimittel
DE102004054054A1 (de) 2004-11-05 2006-05-11 Boehringer Ingelheim Pharma Gmbh & Co. Kg Verfahren zur Herstellung chiraler 8-(3-Amino-piperidin-1-yl)-xanthine
US7772191B2 (en) 2005-05-10 2010-08-10 Boehringer Ingelheim International Gmbh Processes for preparing of glucopyranosyl-substituted benzyl-benzene derivatives and intermediates therein
DE102005035891A1 (de) 2005-07-30 2007-02-08 Boehringer Ingelheim Pharma Gmbh & Co. Kg 8-(3-Amino-piperidin-1-yl)-xanthine, deren Herstellung und deren Verwendung als Arzneimittel
EP1852108A1 (en) 2006-05-04 2007-11-07 Boehringer Ingelheim Pharma GmbH & Co.KG DPP IV inhibitor formulations
JP5323684B2 (ja) * 2006-05-04 2013-10-23 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング 多形体
PE20080251A1 (es) 2006-05-04 2008-04-25 Boehringer Ingelheim Int Usos de inhibidores de dpp iv
US9255099B2 (en) 2006-06-06 2016-02-09 Intra-Cellular Therapies, Inc. Pyrazolo[3,4-D]pyrimidine-4,6(5H,7H)-diones as phosphodiesterase 1 inhibitors
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