AP2011005745A0 - Modulators of toll-like receptors. - Google Patents
Modulators of toll-like receptors.Info
- Publication number
- AP2011005745A0 AP2011005745A0 AP2011000745A AP2011000745A AP2011005745A0 AP 2011005745 A0 AP2011005745 A0 AP 2011005745A0 AP 2011000745 A AP2011000745 A AP 2011000745A AP 2011000745 A AP2011000745 A AP 2011000745A AP 2011005745 A0 AP2011005745 A0 AP 2011005745A0
- Authority
- AP
- ARIPO
- Prior art keywords
- toll
- modulators
- receptors
- Prior art date
Links
- 102000002689 Toll-like receptor Human genes 0.000 title 1
- 108020000411 Toll-like receptor Proteins 0.000 title 1
Classifications
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/527—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim spiro-condensed
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- A61K31/5375—1,4-Oxazines, e.g. morpholine
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- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
- A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
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- A61K31/573—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone substituted in position 21, e.g. cortisone, dexamethasone, prednisone or aldosterone
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- A61K31/708—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines containing purines, e.g. adenosine, adenylic acid having oxo groups directly attached to the purine ring system, e.g. guanosine, guanylic acid
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- C07D487/04—Ortho-condensed systems
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- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6561—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings
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- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Molecular Biology (AREA)
- Virology (AREA)
- Gastroenterology & Hepatology (AREA)
- Immunology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Pulmonology (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Zoology (AREA)
- Tropical Medicine & Parasitology (AREA)
- AIDS & HIV (AREA)
- Biotechnology (AREA)
- Biochemistry (AREA)
- Otolaryngology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Steroid Compounds (AREA)
- Pyrrole Compounds (AREA)
- Electrochromic Elements, Electrophoresis, Or Variable Reflection Or Absorption Elements (AREA)
- Devices For Checking Fares Or Tickets At Control Points (AREA)
- Digital Transmission Methods That Use Modulated Carrier Waves (AREA)
Applications Claiming Priority (5)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US12106108P | 2008-12-09 | 2008-12-09 | |
US17040409P | 2009-04-17 | 2009-04-17 | |
US22438609P | 2009-07-09 | 2009-07-09 | |
US22737809P | 2009-07-21 | 2009-07-21 | |
US24263509P | 2009-09-15 | 2009-09-15 |
Publications (1)
Publication Number | Publication Date |
---|---|
AP2011005745A0 true AP2011005745A0 (en) | 2011-06-30 |
Family
ID=41621203
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AP2011000745A AP2011005745A0 (en) | 2008-12-09 | 2009-12-07 | Modulators of toll-like receptors. |
Country Status (33)
Country | Link |
---|---|
US (8) | US8367670B2 (de) |
EP (3) | EP2818469B1 (de) |
JP (3) | JP5600116B2 (de) |
KR (2) | KR101787309B1 (de) |
CN (2) | CN102272134B (de) |
AP (1) | AP2011005745A0 (de) |
AR (1) | AR074506A1 (de) |
AU (1) | AU2009333559B2 (de) |
BR (1) | BRPI0923305B1 (de) |
CA (1) | CA2745295C (de) |
CL (1) | CL2011001392A1 (de) |
CO (1) | CO6362010A2 (de) |
CY (1) | CY1115176T1 (de) |
DK (1) | DK2364314T3 (de) |
EA (3) | EA201692167A1 (de) |
EC (2) | ECSP11011189A (de) |
ES (2) | ES2623794T3 (de) |
HK (2) | HK1161880A1 (de) |
HR (1) | HRP20140539T1 (de) |
IL (2) | IL213101A (de) |
MX (1) | MX2011006152A (de) |
NZ (2) | NZ593110A (de) |
PE (1) | PE20120106A1 (de) |
PL (1) | PL2364314T3 (de) |
PT (2) | PT2364314E (de) |
RS (1) | RS53347B (de) |
SG (1) | SG172060A1 (de) |
SI (1) | SI2364314T1 (de) |
SM (1) | SMT201400083B (de) |
TW (5) | TWI432436B (de) |
UY (1) | UY32306A (de) |
WO (1) | WO2010077613A1 (de) |
ZA (1) | ZA201104998B (de) |
Families Citing this family (237)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
PE20120106A1 (es) | 2008-12-09 | 2012-02-20 | Gilead Sciences Inc | Moduladores de receptores tipo toll |
DK2459216T3 (da) | 2009-09-02 | 2013-12-09 | Novartis Ag | Immunogene sammensætninger omfattende tlr-aktivitetsmodulatorer |
SI2477987T1 (en) * | 2009-09-14 | 2018-03-30 | Gilead Sciences, Inc. | MODULATORS TO TOLL OF LIKE RECEPTORS |
AU2010336509A1 (en) * | 2009-12-23 | 2012-07-19 | Elan Pharmaceuticals, Inc | Pteridinones as inhibitors of polo-like kinase |
JP5841998B2 (ja) | 2010-06-03 | 2016-01-13 | ファーマサイクリックス,インク. | ブルトン型チロシンキナーゼ(Btk)の阻害剤の使用 |
WO2012031140A1 (en) | 2010-09-01 | 2012-03-08 | Novartis Ag | Adsorption of immunopotentiators to insoluble metal salts |
WO2012087596A1 (en) | 2010-12-20 | 2012-06-28 | Gilead Sciences, Inc. | Combinations for treating hcv |
AU2012205486B2 (en) * | 2011-01-12 | 2017-02-02 | Array Biopharma, Inc. | Substituted benzoazepines as toll-like receptor modulators |
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